AR034277A1 - Proceso para la produccion de una preparacion liofilizada de pantoprazol, preparacion liofilizada de pantoprazol obtenida, inyeccion de pantoprazol obtenida por reconstitucion en un disolvente y kit de inyeccion - Google Patents

Proceso para la produccion de una preparacion liofilizada de pantoprazol, preparacion liofilizada de pantoprazol obtenida, inyeccion de pantoprazol obtenida por reconstitucion en un disolvente y kit de inyeccion

Info

Publication number
AR034277A1
AR034277A1 ARP010105391A ARP010105391A AR034277A1 AR 034277 A1 AR034277 A1 AR 034277A1 AR P010105391 A ARP010105391 A AR P010105391A AR P010105391 A ARP010105391 A AR P010105391A AR 034277 A1 AR034277 A1 AR 034277A1
Authority
AR
Argentina
Prior art keywords
pantoprazol
preparation
injection
liophilized
pantoprazole
Prior art date
Application number
ARP010105391A
Other languages
English (en)
Original Assignee
Altana Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8170452&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR034277(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Altana Pharma Ag filed Critical Altana Pharma Ag
Publication of AR034277A1 publication Critical patent/AR034277A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • A61K47/183Amino acids, e.g. glycine, EDTA or aspartame
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/19Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Inorganic Chemistry (AREA)
  • Dermatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Proceso para la producción de una preparación liofilizada que comprende 5-difluorometoxi-2-[(3,4-dimetoxi-2-pirimidinil)metilsulfinil]-1-H-bencimidazol (pantoprazol), una sal del mismo, un solvato de pantoprazol o una sal del mismo, que comprende liofilizar una solución acuosa de pantroprazol, una sal del mismo, un solvato de pantoprazol o una sal del mismo, ácido etilenodiaminotetraacético y/o una sal de adecuada del mismo, e hidróxido de sodio y/o carbonato de sodio.Se describe una preparación liofilizada de pantoprazol, así como una inyección obtenible por reconstitución de la preparación liofilizada de pantoprazol en un disolvente adecuado y un kit para inyección.
ARP010105391A 2000-11-22 2001-11-19 Proceso para la produccion de una preparacion liofilizada de pantoprazol, preparacion liofilizada de pantoprazol obtenida, inyeccion de pantoprazol obtenida por reconstitucion en un disolvente y kit de inyeccion AR034277A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP00125569 2000-11-22

Publications (1)

Publication Number Publication Date
AR034277A1 true AR034277A1 (es) 2004-02-18

Family

ID=8170452

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP010105391A AR034277A1 (es) 2000-11-22 2001-11-19 Proceso para la produccion de una preparacion liofilizada de pantoprazol, preparacion liofilizada de pantoprazol obtenida, inyeccion de pantoprazol obtenida por reconstitucion en un disolvente y kit de inyeccion
ARP130102967A AR092374A2 (es) 2000-11-22 2013-08-21 Preparacion liofilizada de 5-difluorometoxi-2-[(3,4-dimetoxi-2-piridinil)metilsulfinil]-1h-bencimidazol (pantoprazol)

Family Applications After (1)

Application Number Title Priority Date Filing Date
ARP130102967A AR092374A2 (es) 2000-11-22 2013-08-21 Preparacion liofilizada de 5-difluorometoxi-2-[(3,4-dimetoxi-2-piridinil)metilsulfinil]-1h-bencimidazol (pantoprazol)

Country Status (40)

Country Link
US (3) US6780881B2 (es)
EP (2) EP1762249A3 (es)
JP (1) JP4886158B2 (es)
KR (2) KR100910606B1 (es)
CN (1) CN1250292C (es)
AR (2) AR034277A1 (es)
AT (1) ATE381946T1 (es)
AU (2) AU1604202A (es)
BG (1) BG66329B1 (es)
BR (1) BRPI0115483B8 (es)
CA (2) CA2428870C (es)
CY (1) CY1107896T1 (es)
CZ (1) CZ304348B6 (es)
DE (1) DE60132108T2 (es)
DK (1) DK1339430T3 (es)
EA (1) EA007602B1 (es)
EC (1) ECSP034613A (es)
EE (1) EE05236B1 (es)
ES (1) ES2298295T3 (es)
GE (1) GEP20053461B (es)
HK (1) HK1060848A1 (es)
HR (1) HRP20030410B1 (es)
HU (1) HUP0303278A3 (es)
IL (2) IL155601A0 (es)
IS (1) IS2971B (es)
ME (1) ME00556B (es)
MX (1) MXPA03004548A (es)
MY (1) MY137726A (es)
NO (1) NO332937B1 (es)
NZ (1) NZ525911A (es)
PE (1) PE20020582A1 (es)
PL (1) PL201188B1 (es)
PT (1) PT1339430E (es)
RS (1) RS52024B (es)
SI (1) SI1339430T1 (es)
SK (1) SK287993B6 (es)
TW (1) TWI284041B (es)
UA (1) UA80961C2 (es)
WO (1) WO2002041919A1 (es)
ZA (1) ZA200303593B (es)

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US20050004172A1 (en) * 2003-05-19 2005-01-06 Pliva-Istrazivacki Institut D.O.O. Solid state forms of 5-(difluoro-methoxy)-2-((3,4-dimethoxy-2-pyridinyl)-methyl) sulfinyl]-1H-benzimidazole sodium aquo complexes
AR045258A1 (es) 2003-08-21 2005-10-19 Altana Pharma Ag Un producto farmaceutico para inyeccion
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DE102004007854A1 (de) * 2004-02-17 2005-09-01 Hexal Ag Stabile, wässrige Formulierung für Benzimidazole
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CN102000034B (zh) * 2010-10-13 2011-12-21 江苏奥赛康药业股份有限公司 一种供注射用的s-泮托拉唑钠组合物及其制备方法
CN102225063B (zh) * 2011-05-10 2012-10-10 江苏奥赛康药业股份有限公司 一种供注射用的泮托拉唑钠组合物
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CN104582687A (zh) * 2012-06-27 2015-04-29 武田药品工业株式会社 用盐稳定的胺和有机酸的液体制剂
CN104000786A (zh) * 2013-02-25 2014-08-27 杭州赛利药物研究所有限公司 泮托拉唑钠冻干制剂及其制备方法
CN104414979A (zh) * 2013-08-21 2015-03-18 哈药集团三精制药股份有限公司 一种泮托拉唑钠冻干粉针剂及其制备方法
CN104019635B (zh) * 2014-06-19 2015-05-27 上海慈瑞医药科技有限公司 一种兰索拉唑原料药化合物及其干燥工艺
CN104055791A (zh) * 2014-07-10 2014-09-24 北京人福军威医药技术开发有限公司 西地碘治疗眼角结膜炎的用途
CN104055792A (zh) * 2014-07-10 2014-09-24 北京人福军威医药技术开发有限公司 西地碘治疗中耳炎的用途
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Also Published As

Publication number Publication date
AU2002216042B2 (en) 2006-08-03
PL201188B1 (pl) 2009-03-31
UA80961C2 (en) 2007-11-26
CA2541946A1 (en) 2002-05-30
PT1339430E (pt) 2008-03-27
CZ20031416A3 (cs) 2003-09-17
BG66329B1 (bg) 2013-06-28
EA007602B1 (ru) 2006-12-29
EE05236B1 (et) 2009-12-15
CN1476335A (zh) 2004-02-18
TWI284041B (en) 2007-07-21
IL155601A (en) 2008-12-29
IS6820A (is) 2003-05-19
JP4886158B2 (ja) 2012-02-29
YU37703A (sh) 2006-05-25
IS2971B (is) 2017-05-15
HRP20030410B1 (en) 2011-02-28
NO20032303L (no) 2003-05-21
HUP0303278A2 (hu) 2004-01-28
ES2298295T3 (es) 2008-05-16
ATE381946T1 (de) 2008-01-15
US20030003058A1 (en) 2003-01-02
ME00556A (en) 2011-12-20
AU1604202A (en) 2002-06-03
CA2428870C (en) 2006-05-23
HK1060848A1 (en) 2004-08-27
MXPA03004548A (es) 2003-09-10
IL155601A0 (en) 2003-11-23
NO332937B1 (no) 2013-02-04
WO2002041919A1 (en) 2002-05-30
BR0115483A (pt) 2003-10-21
PL361118A1 (en) 2004-09-20
EE200300182A (et) 2003-06-16
MY137726A (en) 2009-03-31
US20090093522A1 (en) 2009-04-09
EP1762249A2 (en) 2007-03-14
ECSP034613A (es) 2003-08-29
US8754108B2 (en) 2014-06-17
ZA200303593B (en) 2004-04-23
JP2004513970A (ja) 2004-05-13
CA2428870A1 (en) 2002-05-30
PE20020582A1 (es) 2002-07-06
NZ525911A (en) 2004-11-26
CZ304348B6 (cs) 2014-03-19
RS52024B (sr) 2012-04-30
SK6062003A3 (en) 2003-10-07
CN1250292C (zh) 2006-04-12
ME00556B (me) 2011-12-20
KR20080003010A (ko) 2008-01-04
SK287993B6 (sk) 2012-09-03
CY1107896T1 (el) 2013-09-04
US7351723B2 (en) 2008-04-01
EP1339430A1 (en) 2003-09-03
GEP20053461B (en) 2005-02-25
US20040220228A1 (en) 2004-11-04
KR100910606B1 (ko) 2009-08-04
KR100910607B1 (ko) 2009-08-04
HRP20030410A2 (en) 2005-04-30
KR20030055308A (ko) 2003-07-02
SI1339430T1 (sl) 2008-06-30
HUP0303278A3 (en) 2007-08-28
DE60132108T2 (de) 2008-12-11
DK1339430T3 (da) 2008-05-13
BG107828A (bg) 2004-07-30
EA200300501A1 (ru) 2003-12-25
BRPI0115483B8 (pt) 2021-05-25
AR092374A2 (es) 2015-04-15
EP1762249A3 (en) 2014-05-14
US6780881B2 (en) 2004-08-24
EP1339430B1 (en) 2007-12-26
BRPI0115483B1 (pt) 2017-05-09
NO20032303D0 (no) 2003-05-21
DE60132108D1 (de) 2008-02-07

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