AR028576A1 - Derivados de b-carbolina utiles como inhibidores de fosfodiesterasa - Google Patents

Derivados de b-carbolina utiles como inhibidores de fosfodiesterasa

Info

Publication number
AR028576A1
AR028576A1 ARP010102326A ARP010102326A AR028576A1 AR 028576 A1 AR028576 A1 AR 028576A1 AR P010102326 A ARP010102326 A AR P010102326A AR P010102326 A ARP010102326 A AR P010102326A AR 028576 A1 AR028576 A1 AR 028576A1
Authority
AR
Argentina
Prior art keywords
phosphodesterase
inhibitors
useful
carboline derivatives
carboline
Prior art date
Application number
ARP010102326A
Other languages
English (en)
Original Assignee
Ortho Mcneil Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ortho Mcneil Pharm Inc filed Critical Ortho Mcneil Pharm Inc
Publication of AR028576A1 publication Critical patent/AR028576A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
ARP010102326A 2000-05-17 2001-05-16 Derivados de b-carbolina utiles como inhibidores de fosfodiesterasa AR028576A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US20466700P 2000-05-17 2000-05-17
US09/847,767 US6492358B2 (en) 2000-05-17 2001-05-02 β-carboline derivatives useful as inhibitors of phosphodiesterase

Publications (1)

Publication Number Publication Date
AR028576A1 true AR028576A1 (es) 2003-05-14

Family

ID=22758909

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP010102326A AR028576A1 (es) 2000-05-17 2001-05-16 Derivados de b-carbolina utiles como inhibidores de fosfodiesterasa

Country Status (32)

Country Link
US (2) US6492358B2 (es)
EP (1) EP1289985B1 (es)
JP (1) JP5014551B2 (es)
KR (1) KR20030031482A (es)
CN (1) CN1255403C (es)
AR (1) AR028576A1 (es)
AT (1) ATE256127T1 (es)
AU (2) AU2001261167B2 (es)
BG (1) BG66141B1 (es)
CA (1) CA2409715C (es)
CZ (1) CZ20023934A3 (es)
DE (1) DE60101479T2 (es)
DK (1) DK1289985T3 (es)
ES (1) ES2211806T3 (es)
GE (1) GEP20053511B (es)
HK (1) HK1051368A1 (es)
HR (1) HRP20020910B1 (es)
HU (1) HUP0302412A3 (es)
IL (2) IL152873A0 (es)
MX (1) MXPA02011426A (es)
MY (1) MY128479A (es)
NO (1) NO324251B1 (es)
NZ (1) NZ522731A (es)
PL (1) PL205507B1 (es)
PT (1) PT1289985E (es)
RU (1) RU2271358C2 (es)
SK (1) SK16972002A3 (es)
TR (1) TR200302309T4 (es)
TW (1) TWI286553B (es)
UA (1) UA74826C2 (es)
WO (1) WO2001087038A2 (es)
ZA (1) ZA200210111B (es)

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Also Published As

Publication number Publication date
GEP20053511B (en) 2005-05-10
HUP0302412A2 (hu) 2003-11-28
HK1051368A1 (en) 2003-08-01
ATE256127T1 (de) 2003-12-15
PT1289985E (pt) 2004-03-31
HRP20020910B1 (en) 2011-02-28
IL152873A0 (en) 2003-06-24
BG107285A (bg) 2003-07-31
ES2211806T3 (es) 2004-07-16
NO324251B1 (no) 2007-09-17
IL152873A (en) 2012-01-31
UA74826C2 (en) 2006-02-15
ZA200210111B (en) 2004-03-12
DK1289985T3 (da) 2004-04-05
US20020010189A1 (en) 2002-01-24
NO20025527L (no) 2003-01-16
US6864253B2 (en) 2005-03-08
PL365445A1 (en) 2005-01-10
AU6116701A (en) 2001-11-26
US20030166641A1 (en) 2003-09-04
HRP20020910A2 (en) 2004-12-31
MY128479A (en) 2007-02-28
NZ522731A (en) 2004-09-24
TWI286553B (en) 2007-09-11
AU2001261167B2 (en) 2006-10-05
MXPA02011426A (es) 2004-09-06
PL205507B1 (pl) 2010-04-30
JP2003533453A (ja) 2003-11-11
EP1289985B1 (en) 2003-12-10
US6492358B2 (en) 2002-12-10
JP5014551B2 (ja) 2012-08-29
TR200302309T4 (tr) 2004-02-23
HUP0302412A3 (en) 2007-02-28
WO2001087038A2 (en) 2001-11-22
SK16972002A3 (sk) 2003-11-04
CA2409715A1 (en) 2001-11-22
KR20030031482A (ko) 2003-04-21
DE60101479D1 (en) 2004-01-22
CA2409715C (en) 2010-09-14
NO20025527D0 (no) 2002-11-18
RU2271358C2 (ru) 2006-03-10
CZ20023934A3 (cs) 2003-10-15
CN1446217A (zh) 2003-10-01
BG66141B1 (bg) 2011-07-29
WO2001087038A3 (en) 2002-05-16
DE60101479T2 (de) 2005-04-28
EP1289985A2 (en) 2003-03-12
CN1255403C (zh) 2006-05-10

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