AR012098A1 - Derivados de acidos succinicos, maleicos y fumaricos con sustituyentes heterociclicos como antagonistas del receptor endotelial, procedimiento paraprepararlos, medicamentos y preparaciones farmaceuticas que los contienen y un procedimiento para obtener estas preparaciones farmaceuticas - Google Patents
Derivados de acidos succinicos, maleicos y fumaricos con sustituyentes heterociclicos como antagonistas del receptor endotelial, procedimiento paraprepararlos, medicamentos y preparaciones farmaceuticas que los contienen y un procedimiento para obtener estas preparaciones farmaceuticasInfo
- Publication number
- AR012098A1 AR012098A1 ARP980101216A ARP980101216A AR012098A1 AR 012098 A1 AR012098 A1 AR 012098A1 AR P980101216 A ARP980101216 A AR P980101216A AR P980101216 A ARP980101216 A AR P980101216A AR 012098 A1 AR012098 A1 AR 012098A1
- Authority
- AR
- Argentina
- Prior art keywords
- nha
- hal
- atoms
- naa
- independently represent
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/14—Thiadiazoles; Hydrogenated thiadiazoles condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
- C07D271/12—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
- C07D317/50—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to atoms of the carbocyclic ring
- C07D317/60—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D319/10—1,4-Dioxanes; Hydrogenated 1,4-dioxanes
- C07D319/14—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
- C07D319/16—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D319/18—Ethylenedioxybenzenes, not substituted on the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19711428A DE19711428A1 (de) | 1997-03-19 | 1997-03-19 | Endothelin-Rezeptor-Antagonisten |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR012098A1 true AR012098A1 (es) | 2000-09-27 |
Family
ID=7823886
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP980101216A AR012098A1 (es) | 1997-03-19 | 1998-03-18 | Derivados de acidos succinicos, maleicos y fumaricos con sustituyentes heterociclicos como antagonistas del receptor endotelial, procedimiento paraprepararlos, medicamentos y preparaciones farmaceuticas que los contienen y un procedimiento para obtener estas preparaciones farmaceuticas |
Country Status (5)
| Country | Link |
|---|---|
| AR (1) | AR012098A1 (fr) |
| AU (1) | AU6826698A (fr) |
| DE (1) | DE19711428A1 (fr) |
| WO (1) | WO1998041521A1 (fr) |
| ZA (1) | ZA982299B (fr) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10155076A1 (de) * | 2001-11-09 | 2003-05-22 | Merck Patent Gmbh | Verwendung von Endothelin-Rezeptor-Antagonisten zur Behandlung von Tumorerkrankungen |
| RU2462450C2 (ru) * | 2005-09-22 | 2012-09-27 | Мейдзи Сейка Кайся, Лтд. | ИНГИБИТОРЫ МЕТАЛЛО-β-ЛАКТАМАЗЫ |
| WO2008140251A2 (fr) * | 2007-05-14 | 2008-11-20 | University-Industry Cooperation Group Of Kyung Hee University | Inhibiteurs de la cyclooxygénase-2 |
| CN101538256B (zh) * | 2009-04-28 | 2014-05-21 | 沈阳药科大学 | 3，4-二芳基呋喃-2，5-二酮类衍生物与3，4-二芳基-1h-吡咯-2，5-二酮类衍生物及其用途 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1994002474A1 (fr) * | 1992-07-17 | 1994-02-03 | Smithkline Beecham Corporation | Antagonistes du recepteur de l'endotheline |
| KR960703901A (ko) * | 1993-08-19 | 1996-08-31 | 로즈 암스트롱 | 치환된 2(5H)푸라논, 2(5H)티오페논 및 2(5H)피롤론 유도체, 그의 제조 방법 및 엔도텔린 길항제로서의 그의 용도(Substituted 2(5H)Furanone, 2(5H)Thiophenone and 2(5H)Pyrrolone Derivatives, Their Preparation and Their Use as Endothelin antagonists) |
-
1997
- 1997-03-19 DE DE19711428A patent/DE19711428A1/de not_active Withdrawn
-
1998
- 1998-03-04 WO PCT/EP1998/001207 patent/WO1998041521A1/fr active Application Filing
- 1998-03-04 AU AU68266/98A patent/AU6826698A/en not_active Abandoned
- 1998-03-18 ZA ZA982299A patent/ZA982299B/xx unknown
- 1998-03-18 AR ARP980101216A patent/AR012098A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AU6826698A (en) | 1998-10-12 |
| ZA982299B (en) | 1998-09-28 |
| DE19711428A1 (de) | 1998-09-24 |
| WO1998041521A1 (fr) | 1998-09-24 |
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