ZA200406191B - N-ä5-Ä4-94-methyl-piperazino-methyl)-benzoylamidoÜ-2-methyphenylü-4-(3-pyridyl)-2-pyrimidine-amine coated stents - Google Patents

N-ä5-Ä4-94-methyl-piperazino-methyl)-benzoylamidoÜ-2-methyphenylü-4-(3-pyridyl)-2-pyrimidine-amine coated stents Download PDF

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Publication number: ZA200406191B
Authority: ZA; South Africa
Prior art keywords: methyl; pharmaceutically acceptable; inhibitor; pyrimidine; piperazino
Prior art date: 2002-02-28

Application number

ZA200406191A

Other languages

English (en)

Inventor

Margaret F Prescott

David L Feldman

Original Assignee

Novartis Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-02-28

Filing date

2004-08-03

Publication date

2006-05-31

2004-08-03 Application filed by Novartis Ag filed Critical Novartis Ag

2006-05-31 Publication of ZA200406191B publication Critical patent/ZA200406191B/en

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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
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Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical & Material Sciences (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Veterinary Medicine (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
Epidemiology (AREA)
Pharmacology & Pharmacy (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Bioinformatics & Cheminformatics (AREA)
General Chemical & Material Sciences (AREA)
Molecular Biology (AREA)
Heart & Thoracic Surgery (AREA)
Biomedical Technology (AREA)
Vascular Medicine (AREA)
Surgery (AREA)
Diabetes (AREA)
Hematology (AREA)
Dermatology (AREA)
Oral & Maxillofacial Surgery (AREA)
Transplantation (AREA)
Immunology (AREA)
Cardiology (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Endocrinology (AREA)
Emergency Medicine (AREA)
Obesity (AREA)
Urology & Nephrology (AREA)
Gastroenterology & Hepatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Materials For Medical Uses (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

ZA200406191A 2002-02-28 2004-08-03 N-ä5-Ä4-94-methyl-piperazino-methyl)-benzoylamidoÜ-2-methyphenylü-4-(3-pyridyl)-2-pyrimidine-amine coated stents ZA200406191B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US36025402P	2002-02-28	2002-02-28

Publications (1)

Publication Number	Publication Date
ZA200406191B true ZA200406191B (en)	2006-05-31

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ID=27766209

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ZA200406191A ZA200406191B (en)	2002-02-28	2004-08-03	N-ä5-Ä4-94-methyl-piperazino-methyl)-benzoylamidoÜ-2-methyphenylü-4-(3-pyridyl)-2-pyrimidine-amine coated stents

Country Status (18)

Country	Link
US (1)	US20050209244A1 (ru)
EP (1)	EP1480688A1 (ru)
JP (1)	JP2005519080A (ru)
KR (1)	KR20040093058A (ru)
CN (1)	CN1326577C (ru)
AU (1)	AU2003214079B2 (ru)
BR (1)	BR0308053A (ru)
CA (1)	CA2477558A1 (ru)
CO (1)	CO5611172A2 (ru)
EC (1)	ECSP045240A (ru)
IL (1)	IL163771A0 (ru)
MX (1)	MXPA04008361A (ru)
NO (1)	NO20044093L (ru)
NZ (1)	NZ534544A (ru)
PL (1)	PL371466A1 (ru)
RU (1)	RU2341266C2 (ru)
WO (1)	WO2003072159A1 (ru)
ZA (1)	ZA200406191B (ru)

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2003
- 2003-02-27 CN CNB038047888A patent/CN1326577C/zh not_active Expired - Fee Related
- 2003-02-27 CA CA002477558A patent/CA2477558A1/en not_active Abandoned
- 2003-02-27 EP EP03709729A patent/EP1480688A1/en not_active Withdrawn
- 2003-02-27 JP JP2003570902A patent/JP2005519080A/ja active Pending
- 2003-02-27 IL IL16377103A patent/IL163771A0/xx unknown
- 2003-02-27 BR BR0308053-6A patent/BR0308053A/pt not_active IP Right Cessation
- 2003-02-27 AU AU2003214079A patent/AU2003214079B2/en not_active Ceased
- 2003-02-27 KR KR10-2004-7012608A patent/KR20040093058A/ko not_active Application Discontinuation
- 2003-02-27 WO PCT/EP2003/002028 patent/WO2003072159A1/en active IP Right Grant
- 2003-02-27 NZ NZ534544A patent/NZ534544A/en unknown
- 2003-02-27 PL PL03371466A patent/PL371466A1/xx not_active Application Discontinuation
- 2003-02-27 RU RU2004129281/15A patent/RU2341266C2/ru not_active IP Right Cessation
- 2003-02-27 MX MXPA04008361A patent/MXPA04008361A/es unknown
- 2003-02-27 US US10/505,398 patent/US20050209244A1/en not_active Abandoned
2004
- 2004-08-03 ZA ZA200406191A patent/ZA200406191B/en unknown
- 2004-08-20 EC EC2004005240A patent/ECSP045240A/es unknown
- 2004-09-21 CO CO04093663A patent/CO5611172A2/es not_active Application Discontinuation
- 2004-09-27 NO NO20044093A patent/NO20044093L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
ECSP045240A (es)	2004-09-28
NO20044093L (no)	2004-11-24
CA2477558A1 (en)	2003-09-04
CN1638823A (zh)	2005-07-13
KR20040093058A (ko)	2004-11-04
IL163771A0 (en)	2005-12-18
RU2004129281A (ru)	2005-09-10
RU2341266C2 (ru)	2008-12-20
PL371466A1 (en)	2005-06-13
AU2003214079B2 (en)	2007-05-31
US20050209244A1 (en)	2005-09-22
EP1480688A1 (en)	2004-12-01
CN1326577C (zh)	2007-07-18
AU2003214079A1 (en)	2003-09-09
NZ534544A (en)	2007-05-31
CO5611172A2 (es)	2006-02-28
JP2005519080A (ja)	2005-06-30
BR0308053A (pt)	2004-12-28
WO2003072159A1 (en)	2003-09-04
MXPA04008361A (es)	2004-11-26

Publication	Publication Date	Title
ZA200406191B (en)	2006-05-31	N-ä5-Ä4-94-methyl-piperazino-methyl)-benzoylamidoÜ-2-methyphenylü-4-(3-pyridyl)-2-pyrimidine-amine coated stents
ZA200405118B (en)	2005-06-21	Drug delivery systems for the prevention and treatment of vascular diseases comprising rapamycin and derivatives thereof.
TWI435724B (zh)	2014-05-01	組合物、系統、套組及使用醫藥裝置施加雷帕黴素（ｒａｐａｍｙｃｉｎ）類似物及紫杉醇之方法
US20110305742A1 (en)	2011-12-15	Pharmaceutical compositions
AU2003283399B2 (en)	2007-04-19	Drug delivery system
JP2005519080A5 (ru)	2006-05-25
AU2005229566A1 (en)	2005-10-13	VEGF receptor tyrosine kinase inhibitor coated stent
JP2010500404A (ja)	2010-01-07	ラパマイシン類似体及びパクリタキセルを含む組成物及び薬物送達システム
Tedesco-Silva et al.	2022	An overview of the efficacy and safety of everolimus in adult solid organ transplant recipients
WO2005099695A1 (en)	2005-10-27	Drug delivery systems for the prevention and treatment of vascular diseases
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