ZA200102588B - Aryl-substituted propanolamine derivatives, methods for their production, medicaments containing said compounds and their use. - Google Patents

Aryl-substituted propanolamine derivatives, methods for their production, medicaments containing said compounds and their use.

Info

Publication number
ZA200102588B
ZA200102588B ZA200102588A ZA200102588A ZA200102588B ZA 200102588 B ZA200102588 B ZA 200102588B ZA 200102588 A ZA200102588 A ZA 200102588A ZA 200102588 A ZA200102588 A ZA 200102588A ZA 200102588 B ZA200102588 B ZA 200102588B
Authority
ZA
South Africa
Prior art keywords
aryl
compounds
production
methods
medicaments containing
Prior art date
Application number
ZA200102588A
Other languages
English (en)
Inventor
Wendelin Frick
Reinhard Kirsch
Heiner Glombik
Werner Kramer
Hans-Ludwig Schaefer
Original Assignee
Aventis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Gmbh filed Critical Aventis Pharma Gmbh
Publication of ZA200102588B publication Critical patent/ZA200102588B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/18—Acyclic radicals, substituted by carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biochemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Peptides Or Proteins (AREA)
  • Pyridine Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
ZA200102588A 1998-10-02 2001-03-29 Aryl-substituted propanolamine derivatives, methods for their production, medicaments containing said compounds and their use. ZA200102588B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19845405A DE19845405C2 (de) 1998-10-02 1998-10-02 Arylsubstituierte Propanolaminderivate und deren Verwendung

Publications (1)

Publication Number Publication Date
ZA200102588B true ZA200102588B (en) 2002-01-30

Family

ID=7883186

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200102588A ZA200102588B (en) 1998-10-02 2001-03-29 Aryl-substituted propanolamine derivatives, methods for their production, medicaments containing said compounds and their use.

Country Status (23)

Country Link
US (4) US6245744B1 (es)
EP (1) EP1117645B1 (es)
JP (1) JP3794618B2 (es)
KR (1) KR100600425B1 (es)
CN (1) CN1135223C (es)
AR (1) AR021844A1 (es)
AT (1) ATE266005T1 (es)
AU (1) AU757871B2 (es)
BR (1) BR9915967A (es)
CA (1) CA2345369C (es)
CZ (1) CZ299828B6 (es)
DE (2) DE19845405C2 (es)
DK (1) DK1117645T3 (es)
ES (1) ES2219110T3 (es)
HK (1) HK1040708B (es)
HU (1) HU228987B1 (es)
ID (1) ID27762A (es)
PL (1) PL347107A1 (es)
PT (1) PT1117645E (es)
RU (1) RU2226532C2 (es)
TR (1) TR200100894T2 (es)
WO (1) WO2000020392A1 (es)
ZA (1) ZA200102588B (es)

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US7208504B2 (en) * 2002-10-12 2007-04-24 Sanofi-Aventis Deutschland Gmbh Bicyclic inhibitors of hormone sensitive lipase
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US7196114B2 (en) * 2003-02-17 2007-03-27 Sanofi-Aventis Deutschland Gmbh Substituted 3-(benzoylureido) thiophene derivatives, processes for preparing them and their use
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Also Published As

Publication number Publication date
EP1117645B1 (de) 2004-05-06
JP3794618B2 (ja) 2006-07-05
ATE266005T1 (de) 2004-05-15
DE19845405A1 (de) 2000-04-20
HK1040708B (zh) 2004-06-18
PL347107A1 (en) 2002-03-25
DE59909418D1 (de) 2004-06-09
RU2226532C2 (ru) 2004-04-10
ID27762A (id) 2001-04-26
CZ20011175A3 (cs) 2001-07-11
CA2345369A1 (en) 2000-04-13
US6569835B2 (en) 2003-05-27
HU228987B1 (hu) 2013-07-29
KR100600425B1 (ko) 2006-07-13
HUP0103877A3 (en) 2002-10-28
TR200100894T2 (tr) 2001-10-22
US20020042381A1 (en) 2002-04-11
US20020177610A1 (en) 2002-11-28
AU757871B2 (en) 2003-03-06
KR20010103592A (ko) 2001-11-23
CN1321148A (zh) 2001-11-07
WO2000020392A1 (de) 2000-04-13
US6245744B1 (en) 2001-06-12
EP1117645A1 (de) 2001-07-25
DK1117645T3 (da) 2004-08-02
ES2219110T3 (es) 2004-11-16
BR9915967A (pt) 2001-08-28
CA2345369C (en) 2009-12-29
US6566340B2 (en) 2003-05-20
PT1117645E (pt) 2004-09-30
DE19845405C2 (de) 2000-07-13
JP2002526529A (ja) 2002-08-20
AR021844A1 (es) 2002-08-07
AU5979599A (en) 2000-04-26
CN1135223C (zh) 2004-01-21
US6897198B2 (en) 2005-05-24
US20030195145A1 (en) 2003-10-16
HK1040708A1 (en) 2002-06-21
CZ299828B6 (cs) 2008-12-10
HUP0103877A2 (hu) 2002-02-28

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