WO2016004280A3 - Inhibiteurs de tyrosine kinase de bruton - Google Patents
Inhibiteurs de tyrosine kinase de bruton Download PDFInfo
- Publication number
- WO2016004280A3 WO2016004280A3 PCT/US2015/038947 US2015038947W WO2016004280A3 WO 2016004280 A3 WO2016004280 A3 WO 2016004280A3 US 2015038947 W US2015038947 W US 2015038947W WO 2016004280 A3 WO2016004280 A3 WO 2016004280A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- inhibitors
- btk
- tyrosine kinase
- bruton
- irreversible
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4166—1,3-Diazoles having oxo groups directly attached to the heterocyclic ring, e.g. phenytoin
Abstract
L'invention concerne des composés hétéroaryle en tant qu'inhibiteurs de kinase. Des méthodes de synthèse de tels inhibiteurs et des méthodes d'utilisation de ces inhibiteurs dans le traitement de maladies sont également décrits.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201462019977P | 2014-07-02 | 2014-07-02 | |
US62/019,977 | 2014-07-02 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2016004280A2 WO2016004280A2 (fr) | 2016-01-07 |
WO2016004280A3 true WO2016004280A3 (fr) | 2016-03-10 |
Family
ID=55020101
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/US2015/038947 WO2016004280A2 (fr) | 2014-07-02 | 2015-07-02 | Inhibiteurs de tyrosine kinase de bruton |
Country Status (1)
Country | Link |
---|---|
WO (1) | WO2016004280A2 (fr) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TWI815137B (zh) * | 2018-06-15 | 2023-09-11 | 漢達生技醫藥股份有限公司 | 尼洛替尼十二烷基硫酸鹽之結晶 |
WO2020113094A1 (fr) | 2018-11-30 | 2020-06-04 | Nuvation Bio Inc. | Composés pyrrole et pyrazole et leurs procédés d'utilisation |
JP7475370B2 (ja) | 2019-05-10 | 2024-04-26 | 河南知微生物医薬有限公司 | ブルトン型チロシンキナーゼ阻害剤としての置換されている1-アミノ-1h-イミダゾール-5-カルボキサミド |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20030100768A1 (en) * | 2000-12-13 | 2003-05-29 | Han Amy Qi | Imidazolidinones and their related derivatives as hepatitis C virus NS3 protease inhibitors |
WO2014082598A1 (fr) * | 2012-11-30 | 2014-06-05 | Centaurus Biopharma Co., Ltd. | Inhibiteurs de la tyrosine kinase de bruton |
-
2015
- 2015-07-02 WO PCT/US2015/038947 patent/WO2016004280A2/fr active Application Filing
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20030100768A1 (en) * | 2000-12-13 | 2003-05-29 | Han Amy Qi | Imidazolidinones and their related derivatives as hepatitis C virus NS3 protease inhibitors |
WO2014082598A1 (fr) * | 2012-11-30 | 2014-06-05 | Centaurus Biopharma Co., Ltd. | Inhibiteurs de la tyrosine kinase de bruton |
Non-Patent Citations (1)
Title |
---|
HAHM ET AL.: "An Efficient Synthesis of Enantiomerically Pure Functionalized Imidazolidin-2-ones from Chiral Aziridines: Supplementary Information.", THE ROYAL SCIENCE OF CHEMISTRY, 2005, Retrieved from the Internet <URL:http://www.rsc.org/suppdata/cc/b5/b503750f/b503750f.pdf> [retrieved on 20150902] * |
Also Published As
Publication number | Publication date |
---|---|
WO2016004280A2 (fr) | 2016-01-07 |
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