UY35359A - 7-OXO-PIRIDO[2,3-d]PIRIMIDINAS SUSTITUIDAS Y MÉTODOS DE USO - Google Patents

7-OXO-PIRIDO[2,3-d]PIRIMIDINAS SUSTITUIDAS Y MÉTODOS DE USO

Info

Publication number
UY35359A
UY35359A UY0001035359A UY35359A UY35359A UY 35359 A UY35359 A UY 35359A UY 0001035359 A UY0001035359 A UY 0001035359A UY 35359 A UY35359 A UY 35359A UY 35359 A UY35359 A UY 35359A
Authority
UY
Uruguay
Prior art keywords
methods
pirido
pyrimidins
oxo
substituted
Prior art date
Application number
UY0001035359A
Other languages
English (en)
Spanish (es)
Inventor
Brown James
Thomas T Nguyen
Jian J Chen
Hong Fang-Tsao
Ryan Wurz
Andrew Tasker
Seifu Tadesse
Liping H Pettus
Bradley J Herberich
Harrington Essa
Original Assignee
Amgen Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Amgen Inc filed Critical Amgen Inc
Publication of UY35359A publication Critical patent/UY35359A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
UY0001035359A 2013-03-01 2014-02-28 7-OXO-PIRIDO[2,3-d]PIRIMIDINAS SUSTITUIDAS Y MÉTODOS DE USO UY35359A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361771582P 2013-03-01 2013-03-01
US201361900156P 2013-11-05 2013-11-05

Publications (1)

Publication Number Publication Date
UY35359A true UY35359A (es) 2014-09-30

Family

ID=50288304

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001035359A UY35359A (es) 2013-03-01 2014-02-28 7-OXO-PIRIDO[2,3-d]PIRIMIDINAS SUSTITUIDAS Y MÉTODOS DE USO

Country Status (7)

Country Link
EP (1) EP2961750A1 (fr)
JP (1) JP2016510029A (fr)
AU (1) AU2014223396A1 (fr)
CA (1) CA2903040A1 (fr)
TW (1) TW201522332A (fr)
UY (1) UY35359A (fr)
WO (1) WO2014134308A1 (fr)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP6631616B2 (ja) 2014-07-26 2020-01-15 ノース・アンド・サウス・ブラザー・ファーマシー・インベストメント・カンパニー・リミテッド CDK阻害剤としての2−アミノ−ピリド[2,3−d]ピリミジン−7(8H)−オン誘導体及びその使用
EP3294737A4 (fr) * 2015-05-12 2018-10-03 Kalyra Pharmaceuticals, Inc. Composés bicycliques
CN106632313B (zh) * 2016-03-04 2021-04-09 上海贤鼎生物科技有限公司 一种抗癌药帕博昔布重要中间体及合成工艺
IL276802B2 (en) 2018-03-09 2023-09-01 Recurium Ip Holdings Llc Transduced 2,1-dihydro-3h-pyrazolo[4,3-d]pyrimidine-3-ones
KR102328435B1 (ko) * 2018-09-11 2021-11-18 재단법인 대구경북첨단의료산업진흥재단 신규 피리도-피리미딘 유도체, 이의 제조방법 및 이를 유효성분으로 함유하는 단백질 키나아제 관련 질환의 예방 또는 치료용 약학적 조성물
EP4065578A1 (fr) 2019-11-26 2022-10-05 Theravance Biopharma R&D IP, LLC Composés de pyrimidine pyridinone fusionnés en tant qu'inhibiteurs de jak
AU2022234998A1 (en) * 2021-03-08 2023-10-12 Jinan University Pyridopyrimidine compounds and applications thereof
CN114210238A (zh) * 2021-12-02 2022-03-22 上海旭东海普南通药业有限公司 一种氟尿嘧啶精制方法及装置

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2711249T3 (es) * 2008-06-27 2019-04-30 Celgene Car Llc Compuestos de heteroarilo y usos de los mismos
US8619856B2 (en) 2008-10-03 2013-12-31 Qualcomm Incorporated Video coding with large macroblocks
WO2010129053A2 (fr) * 2009-05-05 2010-11-11 Dana Farber Cancer Institute Inhibiteurs d'egfr et procédés de traitement de troubles
EP2637502B1 (fr) 2010-11-10 2018-01-10 Celgene CAR LLC Inhibiteurs d'egfr sélectifs d'un mutant et leurs utilisations
CN102816162B (zh) * 2011-06-10 2016-04-27 中国科学院广州生物医药与健康研究院 嘧啶并嘧啶酮类化合物及其药用组合物和应用
WO2013170671A1 (fr) * 2012-05-14 2013-11-21 华东理工大学 Dérivé de ptéridine cétone et ses applications en tant qu'inhibiteur d'egfr, de blk et de flt3
CN103012399B (zh) * 2012-11-22 2015-06-17 中国科学院广州生物医药与健康研究院 7-氧代吡啶并嘧啶类化合物及其药用组合物和应用

Also Published As

Publication number Publication date
EP2961750A1 (fr) 2016-01-06
TW201522332A (zh) 2015-06-16
CA2903040A1 (fr) 2014-09-04
JP2016510029A (ja) 2016-04-04
WO2014134308A1 (fr) 2014-09-04
AU2014223396A1 (en) 2015-08-27

Similar Documents

Publication Publication Date Title
DOP2015000274A (es) Compuestos químicos
CR20150472A (es) USO DE DERIVADOS DE PIRAZOLOPIRIMIDINA PARA EL TRATAMIENTO DE TRANSTORNOS RELACIONADOS CON LA PI3Kd
CY1123953T1 (el) Καθυστερημενης απελευθερωσης συνθεσεις λινακλοτιδης
UY35359A (es) 7-OXO-PIRIDO[2,3-d]PIRIMIDINAS SUSTITUIDAS Y MÉTODOS DE USO
DOP2015000158A (es) Inhibidores de prmt5 y sus usos
SV2018005687A (es) Derivados de dihidroimidazopirazinona usados en el tratamiento del cancer
CU20160052A7 (es) Amino-heteroaril-benzamidas como inhibidores de cinasa
CR20150628A (es) Derivados de la pirazolopirrolidina y su uso en el tratamiento de enfermedades
CL2016001895A1 (es) Compuestos
CL2015002767A1 (es) Compuestos terapéuticos y composiciones
UY35663A (es) Derivados de piperidinil-indol como inhibidores del factor de complemento b y usos de los mismos
UY34750A (es) ?compuestos para el tratamiento del hiv, composiciones,métodos de preparación, intermediarios y métodos terapéuticos?.
CU20160192A7 (es) Derivados de indano e indolina útiles como activadores de la guanilato ciclasa soluble
CL2016002091A1 (es) Compuesto de triazina y su uso para fines medicinales
ECSP16074478A (es) Compuestos novedosos
UY36875A (es) Composiciones inhibidoras de bromodominios para el tratamiento de diversas enfermedades
CL2019002900A1 (es) Análogos de benzoazepina como agentes inhibidores de la tirosina cinasa de bruton.
DOP2017000107A (es) Diamino-quinoleina 2,4 sustituida como nuevos agentes anticancerigenos
ECSP16008797A (es) Derivados de heterobicicloaril como inhibidores rorc2 y métodos de uso de los mismos
CL2015003195A1 (es) Derivados de purina como agonistas del receptor cb2.
CR20160016A (es) Pirazolpiridinas sustituidas
CL2017000827A1 (es) Inhibidores de aldosterona sintasa
DOP2016000297A (es) Composiciones farmacéuticas útiles para tratar enfermedades infecciosas
UY36124A (es) Derivados de carboxamida
DOP2018000049A (es) Compuestos para uso en aplicaciones antibacterianas

Legal Events

Date Code Title Description
104 Application deemed to be withdrawn (no substantive examination fee paid)

Effective date: 20150710