UY34626A - Proceso para la preparación estereoselectiva de pirazol carboxamida y compuestos intermediarios - Google Patents

Proceso para la preparación estereoselectiva de pirazol carboxamida y compuestos intermediarios

Info

Publication number
UY34626A
UY34626A UY0001034626A UY34626A UY34626A UY 34626 A UY34626 A UY 34626A UY 0001034626 A UY0001034626 A UY 0001034626A UY 34626 A UY34626 A UY 34626A UY 34626 A UY34626 A UY 34626A
Authority
UY
Uruguay
Prior art keywords
pirazol
carboxamide
intermediate compounds
stereoselective preparation
stereoselective
Prior art date
Application number
UY0001034626A
Other languages
English (en)
Inventor
Smejkal Tomas
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of UY34626A publication Critical patent/UY34626A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C249/00—Preparation of compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C249/04—Preparation of compounds containing nitrogen atoms doubly-bound to a carbon skeleton of oximes
    • C07C249/08—Preparation of compounds containing nitrogen atoms doubly-bound to a carbon skeleton of oximes by reaction of hydroxylamines with carbonyl compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/32—Oximes
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/32—Oximes
    • C07C251/34—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • C07C251/44—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atom of at least one of the oxyimino groups being part of a ring other than a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/32—Oximes
    • C07C251/62—Oximes having oxygen atoms of oxyimino groups esterified
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/32—Oximes
    • C07C251/62—Oximes having oxygen atoms of oxyimino groups esterified
    • C07C251/64—Oximes having oxygen atoms of oxyimino groups esterified by carboxylic acids
    • C07C251/66—Oximes having oxygen atoms of oxyimino groups esterified by carboxylic acids with the esterifying carboxyl groups bound to hydrogen atoms, to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/527—Unsaturated compounds containing keto groups bound to rings other than six-membered aromatic rings
    • C07C49/573—Unsaturated compounds containing keto groups bound to rings other than six-membered aromatic rings containing hydroxy groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/587—Unsaturated compounds containing a keto groups being part of a ring
    • C07C49/687—Unsaturated compounds containing a keto groups being part of a ring containing halogen
    • C07C49/693—Unsaturated compounds containing a keto groups being part of a ring containing halogen polycyclic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/587—Unsaturated compounds containing a keto groups being part of a ring
    • C07C49/703—Unsaturated compounds containing a keto groups being part of a ring containing hydroxy groups
    • C07C49/743—Unsaturated compounds containing a keto groups being part of a ring containing hydroxy groups having unsaturation outside the rings, e.g. humulones, lupulones
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/56—Ring systems containing bridged rings
    • C07C2603/58—Ring systems containing bridged rings containing three rings
    • C07C2603/60—Ring systems containing bridged rings containing three rings containing at least one ring with less than six members
    • C07C2603/66—Ring systems containing bridged rings containing three rings containing at least one ring with less than six members containing five-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Catalysts (AREA)

Abstract

La presente invención se refiere a un proceso para la preparación enantioselectiva de la ((1S,4R)-9- 5 diclorometilen-1,2,3,4-tetrahidro-1,4-metanonaftalen-5-il)amida del ácido 3-difluorometil-1-metil-1H-pirazol-4-carboxílico de fórmula Ib
UY0001034626A 2012-02-15 2013-02-14 Proceso para la preparación estereoselectiva de pirazol carboxamida y compuestos intermediarios UY34626A (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP12155526 2012-02-15
EP12173642 2012-06-26
EP12177606 2012-07-24
EP12182799 2012-09-03

Publications (1)

Publication Number Publication Date
UY34626A true UY34626A (es) 2013-09-30

Family

ID=47683767

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001034626A UY34626A (es) 2012-02-15 2013-02-14 Proceso para la preparación estereoselectiva de pirazol carboxamida y compuestos intermediarios

Country Status (21)

Country Link
US (1) US9120759B2 (es)
EP (1) EP2814813B1 (es)
JP (1) JP6216332B2 (es)
KR (1) KR102037942B1 (es)
CN (1) CN104114539B (es)
AP (1) AP4027A (es)
AR (1) AR089989A1 (es)
AU (1) AU2013220443B2 (es)
BR (1) BR112014020011B1 (es)
CA (1) CA2863725C (es)
CO (1) CO7030966A2 (es)
EA (1) EA026529B1 (es)
ES (1) ES2568638T3 (es)
HR (1) HRP20160381T1 (es)
HU (1) HUE028544T2 (es)
PL (1) PL2814813T3 (es)
RS (1) RS54672B1 (es)
TW (1) TWI510472B (es)
UY (1) UY34626A (es)
WO (1) WO2013120860A1 (es)
ZA (1) ZA201405565B (es)

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5093347A (en) 1991-01-28 1992-03-03 Monsanto Company 3-difluoromethylpyrazolecarboxamide fungicides, compositions and use
JP4004123B2 (ja) 1997-12-26 2007-11-07 独立行政法人科学技術振興機構 ルテニウム錯体を触媒とするアルコール化合物の製造方法
AU2002318538A1 (en) 2002-07-15 2004-02-02 Nippon Soda Co., Ltd. Ruthenium compounds, diamine ligands, and process for preparation of optically active alcohols
ITPD20040115A1 (it) 2004-05-04 2004-08-04 Univ Degli Studi Udine Complessi di rutenio con 2-(amminometil)piridine e fosfine, loro preparazione ed uso come catalizzatori
CN1331874C (zh) 2005-01-27 2007-08-15 中国科学院上海有机化学研究所 过渡金属络合物、合成方法及其用途
TWI374126B (en) 2005-10-25 2012-10-11 Syngenta Participations Ag Novel microbiocides
CN101328191B (zh) * 2008-06-13 2013-06-05 中国科学院上海有机化学研究所 一类含氮配体过渡金属络合物、合成方法及其用途
AU2009309884B2 (en) * 2008-10-27 2013-08-29 Syngenta Participations Ag Process for the preparation of benzonorbornenes
PL2462108T3 (pl) * 2009-08-06 2013-09-30 Syngenta Participations Ag Sposób otrzymywania amidów kwasów pirazolokarboksylowych
JP5685071B2 (ja) * 2010-04-28 2015-03-18 高砂香料工業株式会社 新規ルテニウム錯体及びこれを触媒とする光学活性アルコール化合物の製造方法
AR083987A1 (es) 2010-12-01 2013-04-10 Bayer Cropscience Ag Amidas de acido pirazolcarboxilico utiles para la reduccion de la contaminacion de micotoxina en las plantas
TWI534126B (zh) * 2011-01-25 2016-05-21 先正達合夥公司 用於製備吡唑羧酸醯胺之方法

Also Published As

Publication number Publication date
WO2013120860A1 (en) 2013-08-22
CN104114539B (zh) 2016-10-12
CO7030966A2 (es) 2014-08-21
CA2863725C (en) 2019-10-01
CN104114539A (zh) 2014-10-22
TWI510472B (zh) 2015-12-01
EP2814813B1 (en) 2016-02-10
AP4027A (en) 2017-02-04
AR089989A1 (es) 2014-10-01
EP2814813A1 (en) 2014-12-24
KR20140128429A (ko) 2014-11-05
EA201400904A1 (ru) 2015-01-30
JP6216332B2 (ja) 2017-10-18
KR102037942B1 (ko) 2019-10-29
AU2013220443B2 (en) 2016-10-27
US9120759B2 (en) 2015-09-01
BR112014020011A2 (es) 2017-06-20
EA026529B1 (ru) 2017-04-28
HRP20160381T1 (hr) 2016-05-20
ES2568638T3 (es) 2016-05-03
RS54672B1 (en) 2016-08-31
TW201345897A (zh) 2013-11-16
HUE028544T2 (en) 2016-12-28
ZA201405565B (en) 2016-01-27
PL2814813T3 (pl) 2016-07-29
BR112014020011B1 (pt) 2019-08-20
US20140364622A1 (en) 2014-12-11
AU2013220443A1 (en) 2014-08-28
AP2014007855A0 (en) 2014-08-31
BR112014020011A8 (pt) 2017-07-11
JP2015506997A (ja) 2015-03-05
CA2863725A1 (en) 2013-08-22

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