UY30805A1 - Moduladores no esteroides de receptores de progesterona - Google Patents
Moduladores no esteroides de receptores de progesteronaInfo
- Publication number
- UY30805A1 UY30805A1 UY30805A UY30805A UY30805A1 UY 30805 A1 UY30805 A1 UY 30805A1 UY 30805 A UY30805 A UY 30805A UY 30805 A UY30805 A UY 30805A UY 30805 A1 UY30805 A1 UY 30805A1
- Authority
- UY
- Uruguay
- Prior art keywords
- therapy
- modulators
- prevention
- progesterone receptors
- progesterone receptor
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/02—1,2-Oxazines; Hydrogenated 1,2-oxazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Abstract
La presente invencion se refiere a moduladores no esteroides del receptor de la progesterona de la formula general I, al uso de moduladores del receptor de Progesterona para la preparacion de medicamentos, así como a composiciones farmacéuticas que contienen estos compuestos. Los compuestos segun la invencion son apropiados para la terapia y la prevencion de enfermedades ginecologicas tales como endometriosis, leiomiomas de utero, hemorragias disfuncionales y dismenorrea y para la terapia y la prevencion de tumores dependientes de hormonas y para el uso para el control de la fertilidad femenina y para la terapia de reemplazo hormonal.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE102006061913A DE102006061913A1 (de) | 2006-12-21 | 2006-12-21 | Nichtsteroidale Progesteronrezeptor-Modulatoren |
DE102007023614A DE102007023614A1 (de) | 2007-05-21 | 2007-05-21 | Nichtsteroidale Progesteronrezeptor-Modulatoren |
Publications (1)
Publication Number | Publication Date |
---|---|
UY30805A1 true UY30805A1 (es) | 2008-07-31 |
Family
ID=39456752
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY30805A UY30805A1 (es) | 2006-12-21 | 2007-12-18 | Moduladores no esteroides de receptores de progesterona |
Country Status (5)
Country | Link |
---|---|
AR (1) | AR064478A1 (es) |
PE (1) | PE20081397A1 (es) |
TW (1) | TW200835498A (es) |
UY (1) | UY30805A1 (es) |
WO (1) | WO2008077647A2 (es) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN103288669B (zh) * | 2013-07-01 | 2015-06-24 | 南开大学 | 一种阿卓乳酸酰胺衍生物及应用 |
Family Cites Families (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8617652D0 (en) * | 1986-07-18 | 1986-08-28 | Ici Plc | Acylanilide derivatives |
GB8617653D0 (en) * | 1986-07-18 | 1986-08-28 | Ici Plc | Amide derivatives |
IE922316A1 (en) * | 1991-07-17 | 1993-01-27 | Smithkline Beecham Corp | Retroviral protease inhibitors |
US5733882A (en) * | 1994-01-17 | 1998-03-31 | Smithkline Beecham Corporation | Retroviral protease inhibitors |
DE19723722A1 (de) * | 1997-05-30 | 1998-12-10 | Schering Ag | Nichtsteroidale Gestagene |
DE19856475A1 (de) * | 1998-11-27 | 2000-05-31 | Schering Ag | Nichtsteroidale Entzündungshemmer |
DE10038639A1 (de) * | 2000-07-28 | 2002-02-21 | Schering Ag | Nichtsteroidale Entzündungshemmer |
US6960581B2 (en) * | 2002-01-14 | 2005-11-01 | Boehringer Ingelheim Pharmaceuticals, Inc. | Glucocorticoid mimetics, methods of making them, pharmaceutical formulations, and uses thereof |
CN1652768A (zh) * | 2002-03-11 | 2005-08-10 | 舍林股份公司 | 用于节育和激素替代疗法的具有孕酮受体调节活性的5-{2-羟基-3-[′1-(3-三氟甲基苯基)-环丙基]-丙酰氨基}-2-苯并[c]呋喃酮及相关化合物 |
EP1344776A1 (en) * | 2002-03-11 | 2003-09-17 | Schering Aktiengesellschaft | 5- 2-hydroxy-3-[1-(3-trifluoromethylphenyl)-cyclopropyl]-propionylamino -phtalide and 6- 2-hydroxy-3-[1-(3-trifluoromethylphenyl)-cyclopropyl]-propionylamino -4-methyl-2,3-benzoxazin-1-one derivatives with progesterone receptor modulating activity for use in fertility control, hormone replacement therapy and the treatment of gynecological disorders |
KR20060027376A (ko) * | 2003-07-01 | 2006-03-27 | 쉐링 악티엔게젤샤프트 | 헤테로시클릭 치환된 펜탄올 유도체, 그의 제조 방법 및그의 항염증제로서 용도 |
ES2414479T3 (es) * | 2005-04-14 | 2013-07-19 | Glaxo Group Limited | Indazoles como ligandos del receptor de glucocorticoides |
DE102005030293A1 (de) * | 2005-06-24 | 2007-01-04 | Schering Ag | Verwendung von nichtsteroidale Progesteronrezeptor-Modulatoren |
DE102005030294A1 (de) * | 2005-06-24 | 2007-01-04 | Schering Ag | Nichtsteroidale Progesteronrezeptor-Modulatoren |
DE102005030292A1 (de) * | 2005-06-24 | 2007-01-11 | Schering Ag | Nichtsteroidale Progesteronrezeptor-Modulatoren |
-
2007
- 2007-12-18 UY UY30805A patent/UY30805A1/es not_active Application Discontinuation
- 2007-12-20 WO PCT/EP2007/011487 patent/WO2008077647A2/de active Application Filing
- 2007-12-20 AR ARP070105761A patent/AR064478A1/es unknown
- 2007-12-20 TW TW096149042A patent/TW200835498A/zh unknown
-
2008
- 2008-01-02 PE PE2008000016A patent/PE20081397A1/es not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
WO2008077647A2 (de) | 2008-07-03 |
TW200835498A (en) | 2008-09-01 |
AR064478A1 (es) | 2009-04-01 |
PE20081397A1 (es) | 2008-12-05 |
WO2008077647A3 (de) | 2008-10-16 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
109 | Application deemed to be withdrawn |
Effective date: 20170802 |