UY30285A1 - Derivados de aminometilpirina, su preparacion y su aplicacion en terapéutica - Google Patents

Derivados de aminometilpirina, su preparacion y su aplicacion en terapéutica

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Publication number
UY30285A1
UY30285A1 UY30285A UY30285A UY30285A1 UY 30285 A1 UY30285 A1 UY 30285A1 UY 30285 A UY30285 A UY 30285A UY 30285 A UY30285 A UY 30285A UY 30285 A1 UY30285 A1 UY 30285A1
Authority
UY
Uruguay
Prior art keywords
therapeutics
preparation
application
derivatives
aminometilipirine
Prior art date
Application number
UY30285A
Other languages
English (en)
Inventor
Barth Francis
Philippe Pointeau
Christian Congy
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of UY30285A1 publication Critical patent/UY30285A1/es

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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Abstract

Derivados de la aminometilpiridina que responden a la formula (I) en la que: Z; X; R1 y R2; R3 y R6; R4; R5; Ar1 y Ar2; n; Alk representan grupos químicos sustituyentes especificados en la descripcion del invento, y que se presentan también en forma de base o de sal de adicion, así como en forma de hidrato o de solvato. Se describen los métodos de prepracion y su aplicacion en terapéutica, particularmente destinados al tratamiento y prevencion de las enfermedades en las que están implicados los receptores de los cannabinoides CB1
UY30285A 2006-04-14 2007-04-13 Derivados de aminometilpirina, su preparacion y su aplicacion en terapéutica UY30285A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0603382A FR2899899A1 (fr) 2006-04-14 2006-04-14 Derives d'aminomethyl pyridine, leur preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
UY30285A1 true UY30285A1 (es) 2007-11-30

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UY30285A UY30285A1 (es) 2006-04-14 2007-04-13 Derivados de aminometilpirina, su preparacion y su aplicacion en terapéutica

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US (1) US20090203699A1 (es)
EP (1) EP2010492A2 (es)
JP (1) JP2009533400A (es)
KR (1) KR20080108540A (es)
CN (1) CN101421240A (es)
AR (1) AR060800A1 (es)
AU (1) AU2007239344A1 (es)
BR (1) BRPI0710741A2 (es)
CA (1) CA2645961A1 (es)
DO (1) DOP2007000067A (es)
FR (1) FR2899899A1 (es)
IL (1) IL194573A0 (es)
MX (1) MX2008013208A (es)
PE (1) PE20071224A1 (es)
RU (1) RU2008144952A (es)
TW (1) TW200813037A (es)
UY (1) UY30285A1 (es)
WO (1) WO2007119001A2 (es)

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EP2025674A1 (de) 2007-08-15 2009-02-18 sanofi-aventis Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
AU2011281132B2 (en) * 2010-07-20 2014-01-30 Council Of Scientific & Industrial Research Pyridin- 2 - YL sulfanyl acid esters and process for the preparation thereof
GB201103419D0 (es) 2011-02-28 2011-04-13 Univ Aberdeen
WO2012120054A1 (de) 2011-03-08 2012-09-13 Sanofi Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
EP2766349B1 (de) 2011-03-08 2016-06-01 Sanofi Mit carbozyklen oder heterozyklen substituierte oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung
EP2683700B1 (de) 2011-03-08 2015-02-18 Sanofi Tetrasubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
WO2012120053A1 (de) 2011-03-08 2012-09-13 Sanofi Verzweigte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
WO2012120055A1 (de) 2011-03-08 2012-09-13 Sanofi Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
US8809372B2 (en) 2011-09-30 2014-08-19 Asana Biosciences, Llc Pyridine derivatives
US9199975B2 (en) 2011-09-30 2015-12-01 Asana Biosciences, Llc Biaryl imidazole derivatives for regulating CYP17

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CA2479744A1 (en) * 2002-03-28 2003-10-09 Paul E. Finke Substituted 2,3-diphenyl pyridines
FR2838439B1 (fr) * 2002-04-11 2005-05-20 Sanofi Synthelabo Derives de terphenyle, leur preparation, les compositions pharmaceutqiues en contenant
FR2838438A1 (fr) * 2002-04-11 2003-10-17 Sanofi Synthelabo Derives de diphenylpyridine,leur preparation, les compositions pharmaceutiques en contenant
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RU2008144952A (ru) 2010-05-20
US20090203699A1 (en) 2009-08-13
TW200813037A (en) 2008-03-16
JP2009533400A (ja) 2009-09-17
KR20080108540A (ko) 2008-12-15
FR2899899A1 (fr) 2007-10-19
DOP2007000067A (es) 2007-10-31
CA2645961A1 (fr) 2007-10-25
AR060800A1 (es) 2008-07-16
MX2008013208A (es) 2008-10-27
CN101421240A (zh) 2009-04-29
PE20071224A1 (es) 2008-01-23
EP2010492A2 (fr) 2009-01-07
BRPI0710741A2 (pt) 2011-06-07

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