TR201722493A2 - Posakonazol i̇çeren kati farmasöti̇k kompozi̇syon - Google Patents
Posakonazol i̇çeren kati farmasöti̇k kompozi̇syon Download PDFInfo
- Publication number
- TR201722493A2 TR201722493A2 TR2017/22493A TR201722493A TR201722493A2 TR 201722493 A2 TR201722493 A2 TR 201722493A2 TR 2017/22493 A TR2017/22493 A TR 2017/22493A TR 201722493 A TR201722493 A TR 201722493A TR 201722493 A2 TR201722493 A2 TR 201722493A2
- Authority
- TR
- Turkey
- Prior art keywords
- pharmaceutical composition
- posaconazol
- composition containing
- solid pharmaceutical
- posaconazole
- Prior art date
Links
- RAGOYPUPXAKGKH-XAKZXMRKSA-N posaconazole Chemical compound O=C1N([C@H]([C@H](C)O)CC)N=CN1C1=CC=C(N2CCN(CC2)C=2C=CC(OC[C@H]3C[C@@](CN4N=CN=C4)(OC3)C=3C(=CC(F)=CC=3)F)=CC=2)C=C1 RAGOYPUPXAKGKH-XAKZXMRKSA-N 0.000 title abstract 3
- 229960001589 posaconazole Drugs 0.000 title abstract 3
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 239000007787 solid Substances 0.000 title 1
- 239000006185 dispersion Substances 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 239000012458 free base Substances 0.000 abstract 1
- 150000004677 hydrates Chemical class 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
Mevcut buluş, posakonazol serbest bazını veya posakonazolün farmasötik olarak kabul edilebilir tuzlarını, kristalin polimorflarını, solvatlarını, hidratlarını veya esterlerini ve bir dispersiyon taşıyıcı içeren bir farmasötik kompozisyonla ilgilidir. Üstelik, kompozisyon, etkili bir proses kullanılarak elde edilmektedir.
Priority Applications (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
TR2017/22493A TR201722493A2 (tr) | 2017-12-28 | 2017-12-28 | Posakonazol i̇çeren kati farmasöti̇k kompozi̇syon |
EP18918419.5A EP3731827A2 (en) | 2017-12-28 | 2018-12-26 | Oral pharmaceutical composition comprising posaconazole |
PCT/TR2018/050906 WO2019240698A2 (en) | 2017-12-28 | 2018-12-26 | Oral pharmaceutical composition comprising posaconazole |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
TR2017/22493A TR201722493A2 (tr) | 2017-12-28 | 2017-12-28 | Posakonazol i̇çeren kati farmasöti̇k kompozi̇syon |
Publications (1)
Publication Number | Publication Date |
---|---|
TR201722493A2 true TR201722493A2 (tr) | 2019-07-22 |
Family
ID=67900711
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TR2017/22493A TR201722493A2 (tr) | 2017-12-28 | 2017-12-28 | Posakonazol i̇çeren kati farmasöti̇k kompozi̇syon |
Country Status (3)
Country | Link |
---|---|
EP (1) | EP3731827A2 (tr) |
TR (1) | TR201722493A2 (tr) |
WO (1) | WO2019240698A2 (tr) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP4196096A1 (en) | 2020-08-13 | 2023-06-21 | Alfred E. Tiefenbacher (GmbH & Co. KG) | Gastro-resistant high-strength formulation containing posaconazole |
EP4091604B1 (en) | 2021-11-25 | 2024-04-03 | Alfred E. Tiefenbacher (GmbH & Co. KG) | Granules containing posaconazole |
WO2023012378A1 (en) | 2021-11-25 | 2023-02-09 | Alfred E. Tiefenbacher (Gmbh Und Co. Kg) | Granules containing posaconazole |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5703079A (en) | 1993-12-21 | 1997-12-30 | Schering Corporation | Tetrahydrofuran antifungals |
US5661151A (en) | 1993-12-21 | 1997-08-26 | Schering Corporation | Tetrahydrofuran antifungals |
ID29290A (id) | 1997-10-07 | 2001-08-16 | Schering Corp | Susunan kristal bentuk-banyak yang dapat membasmi jamur |
DE10014588A1 (de) * | 2000-03-27 | 2001-10-04 | Basf Ag | Wirkstoffhaltige Schwimmformen enthaltend Polyvinylacetat und Polyvinylpyrrolidon, deren Verwendung und Herstellung |
SG170047A1 (en) * | 2006-05-30 | 2011-04-29 | Elan Pharma Int Ltd | Nanoparticulate posaconazole formulations |
US20150231081A1 (en) * | 2014-02-20 | 2015-08-20 | Cadila Healthcare Limited | Delayed release posaconazole tablets |
EP3331501B1 (en) * | 2015-08-08 | 2019-09-11 | Alfred E. Tiefenbacher (GmbH & Co. KG) | Gastro-resistant formulation containing posaconazole |
TR201620462A2 (tr) * | 2016-12-31 | 2018-07-23 | Abdi Ibrahim Ilac Sanayi Ve Ticaret Anonim Sirketi | POSAKONAZOL İÇEREN FARMASÖTİK BİLEŞİMLER ve ÜRETİM YÖNTEMİ |
CN108066289B (zh) * | 2017-12-28 | 2021-01-26 | 广州玻思韬控释药业有限公司 | 一种泊沙康唑固体分散体及其制备方法和泊沙康唑肠溶制剂 |
CA3098306C (en) * | 2018-05-14 | 2024-04-16 | Capsugel Belgium Nv | Solid dosage forms with high active agent loading |
-
2017
- 2017-12-28 TR TR2017/22493A patent/TR201722493A2/tr unknown
-
2018
- 2018-12-26 EP EP18918419.5A patent/EP3731827A2/en active Pending
- 2018-12-26 WO PCT/TR2018/050906 patent/WO2019240698A2/en unknown
Also Published As
Publication number | Publication date |
---|---|
EP3731827A2 (en) | 2020-11-04 |
WO2019240698A2 (en) | 2019-12-19 |
WO2019240698A3 (en) | 2020-02-13 |
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