TR200002804T2 - MRP1 inhibe etmek için yöntemler - Google Patents
MRP1 inhibe etmek için yöntemlerInfo
- Publication number
- TR200002804T2 TR200002804T2 TR2000/02804T TR200002804T TR200002804T2 TR 200002804 T2 TR200002804 T2 TR 200002804T2 TR 2000/02804 T TR2000/02804 T TR 2000/02804T TR 200002804 T TR200002804 T TR 200002804T TR 200002804 T2 TR200002804 T2 TR 200002804T2
- Authority
- TR
- Turkey
- Prior art keywords
- methods
- mrp1
- inhibit
- inhibit mrp1
- wholly
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
Mevcut bulus, direncin kismen veya bütünüyle MRP1'den kaynaklandigi dirençli neoplazmalarin inhibe edilmesi için yararli olan bir formül (I) bilesigi ile ilgilidir.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US8108898P | 1998-04-08 | 1998-04-08 |
Publications (1)
Publication Number | Publication Date |
---|---|
TR200002804T2 true TR200002804T2 (tr) | 2001-02-21 |
Family
ID=22162031
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TR2000/02804T TR200002804T2 (tr) | 1998-04-08 | 1999-04-07 | MRP1 inhibe etmek için yöntemler |
Country Status (17)
Country | Link |
---|---|
US (1) | US6221876B1 (tr) |
EP (1) | EP1067932A4 (tr) |
JP (1) | JP2002510632A (tr) |
KR (1) | KR20010042481A (tr) |
CN (1) | CN1296410A (tr) |
AU (1) | AU3550299A (tr) |
BR (1) | BR9909446A (tr) |
CA (1) | CA2327452A1 (tr) |
EA (1) | EA200001035A1 (tr) |
HU (1) | HUP0102548A2 (tr) |
ID (1) | ID26804A (tr) |
IL (1) | IL138393A0 (tr) |
NO (1) | NO20005041L (tr) |
PL (1) | PL343320A1 (tr) |
SK (1) | SK14992000A3 (tr) |
TR (1) | TR200002804T2 (tr) |
WO (1) | WO1999051236A1 (tr) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2255294T3 (es) * | 1998-08-07 | 2006-06-16 | Chiron Corporation | Derivados de isoxazol sustituidos como moduladores del receptor de estrogenos. |
US6743794B2 (en) | 1999-12-22 | 2004-06-01 | Eli Lilly And Company | Methods and compounds for inhibiting MRP1 |
DE60016039T2 (de) * | 1999-12-22 | 2005-08-11 | Eli Lilly And Co., Indianapolis | Verfahren und verbindungen für die hemmung von mrp1 |
WO2001096346A1 (en) * | 2000-06-14 | 2001-12-20 | Eli Lilly And Company | Tricyclic compounds as mrp1-inhibitors |
US7064131B2 (en) | 2001-04-09 | 2006-06-20 | Eli Lilly And Company | Compounds and methods for inhibiting MRP1 |
CN1281210C (zh) * | 2003-11-29 | 2006-10-25 | 胡汛 | 五味子乙素在制备***药物中的应用 |
WO2005113004A2 (en) * | 2004-05-14 | 2005-12-01 | The Cleveland Clinic Founfation | Small molecule inhibitors for mrp1 and other multidrug transporters |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5182290A (en) * | 1991-08-27 | 1993-01-26 | Neurogen Corporation | Certain oxazoloquinolinones; a new class of GABA brain receptor ligands |
-
1999
- 1999-04-07 EP EP99917359A patent/EP1067932A4/en not_active Withdrawn
- 1999-04-07 BR BR9909446-0A patent/BR9909446A/pt not_active IP Right Cessation
- 1999-04-07 PL PL99343320A patent/PL343320A1/xx not_active Application Discontinuation
- 1999-04-07 CA CA002327452A patent/CA2327452A1/en not_active Abandoned
- 1999-04-07 IL IL13839399A patent/IL138393A0/xx unknown
- 1999-04-07 SK SK1499-2000A patent/SK14992000A3/sk unknown
- 1999-04-07 KR KR1020007011101A patent/KR20010042481A/ko not_active Application Discontinuation
- 1999-04-07 CN CN99804797A patent/CN1296410A/zh active Pending
- 1999-04-07 TR TR2000/02804T patent/TR200002804T2/tr unknown
- 1999-04-07 EA EA200001035A patent/EA200001035A1/ru unknown
- 1999-04-07 WO PCT/US1999/007615 patent/WO1999051236A1/en not_active Application Discontinuation
- 1999-04-07 ID IDW20002006A patent/ID26804A/id unknown
- 1999-04-07 HU HU0102548A patent/HUP0102548A2/hu unknown
- 1999-04-07 AU AU35502/99A patent/AU3550299A/en not_active Abandoned
- 1999-04-07 US US09/646,063 patent/US6221876B1/en not_active Expired - Fee Related
- 1999-04-07 JP JP2000542007A patent/JP2002510632A/ja not_active Withdrawn
-
2000
- 2000-10-06 NO NO20005041A patent/NO20005041L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
NO20005041D0 (no) | 2000-10-06 |
KR20010042481A (ko) | 2001-05-25 |
CA2327452A1 (en) | 1999-10-14 |
JP2002510632A (ja) | 2002-04-09 |
EP1067932A4 (en) | 2001-11-14 |
NO20005041L (no) | 2000-10-06 |
BR9909446A (pt) | 2000-12-12 |
SK14992000A3 (sk) | 2001-06-11 |
AU3550299A (en) | 1999-10-25 |
US6221876B1 (en) | 2001-04-24 |
IL138393A0 (en) | 2001-10-31 |
CN1296410A (zh) | 2001-05-23 |
HUP0102548A2 (hu) | 2001-11-28 |
ID26804A (id) | 2001-02-08 |
PL343320A1 (en) | 2001-08-13 |
WO1999051236A1 (en) | 1999-10-14 |
EA200001035A1 (ru) | 2001-04-23 |
EP1067932A1 (en) | 2001-01-17 |
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