ATE259346T1 - Benflumentolderivative und ihre verwendung gegen parasitäre protozoen und trematoden - Google Patents

Benflumentolderivative und ihre verwendung gegen parasitäre protozoen und trematoden

Info

Publication number
ATE259346T1
ATE259346T1 AT99931151T AT99931151T ATE259346T1 AT E259346 T1 ATE259346 T1 AT E259346T1 AT 99931151 T AT99931151 T AT 99931151T AT 99931151 T AT99931151 T AT 99931151T AT E259346 T1 ATE259346 T1 AT E259346T1
Authority
AT
Austria
Prior art keywords
trematodes
benflumentol
derivatives
use against
against parasitic
Prior art date
Application number
AT99931151T
Other languages
English (en)
Inventor
Thomas Allmendinger
Walther Helmut Wernsdorfer
Original Assignee
Novartis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Pharma Gmbh filed Critical Novartis Pharma Gmbh
Application granted granted Critical
Publication of ATE259346T1 publication Critical patent/ATE259346T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C215/00Compounds containing amino and hydroxy groups bound to the same carbon skeleton
    • C07C215/02Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C215/22Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated
    • C07C215/28Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings
    • C07C215/38Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings with rings other than six-membered aromatic rings being part of the carbon skeleton
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/06Antimalarials
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C217/00Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
    • C07C217/02Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C217/04Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
    • C07C217/06Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted
    • C07C217/08Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted the oxygen atom of the etherified hydroxy group being further bound to an acyclic carbon atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00Systems containing at least three condensed rings
    • C07C2603/02Ortho- or ortho- and peri-condensed systems
    • C07C2603/04Ortho- or ortho- and peri-condensed systems containing three rings
    • C07C2603/06Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members
    • C07C2603/10Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings
    • C07C2603/12Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings only one five-membered ring
    • C07C2603/18Fluorenes; Hydrogenated fluorenes

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
AT99931151T 1998-06-25 1999-06-23 Benflumentolderivative und ihre verwendung gegen parasitäre protozoen und trematoden ATE259346T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH135198 1998-06-25
PCT/EP1999/004355 WO1999067197A1 (en) 1998-06-25 1999-06-23 Benflumetol derivatives, intermediates thereof and their use against parasitical protozoa and trematodes

Publications (1)

Publication Number Publication Date
ATE259346T1 true ATE259346T1 (de) 2004-02-15

Family

ID=4208448

Family Applications (1)

Application Number Title Priority Date Filing Date
AT99931151T ATE259346T1 (de) 1998-06-25 1999-06-23 Benflumentolderivative und ihre verwendung gegen parasitäre protozoen und trematoden

Country Status (17)

Country Link
US (1) US6329552B2 (de)
EP (1) EP1089961B1 (de)
JP (1) JP4355450B2 (de)
CN (1) CN1183097C (de)
AT (1) ATE259346T1 (de)
AU (1) AU4776399A (de)
BR (1) BRPI9912208B8 (de)
CA (1) CA2335685C (de)
CO (1) CO5040050A1 (de)
ES (1) ES2216528T3 (de)
HK (1) HK1035712A1 (de)
ID (1) ID27500A (de)
MY (1) MY117662A (de)
PE (1) PE20000703A1 (de)
PT (1) PT1089961E (de)
TW (2) TWI250141B (de)
WO (1) WO1999067197A1 (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN108148186A (zh) * 2012-01-31 2018-06-12 剑桥显示技术有限公司 聚合物
JP7375343B2 (ja) 2019-06-25 2023-11-08 味の素株式会社 樹脂組成物
CN111320547B (zh) * 2020-04-03 2022-05-20 南京昊绿生物科技有限公司 一种苯芴醇-d9的合成方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1029680C (zh) * 1988-11-10 1995-09-06 军事医学科学院微生物流行病研究所 抗疟新药苯芴醇的合成新工艺
CN1058717A (zh) * 1990-08-08 1992-02-19 中国人民解放军军事医学科学院微生物流行病研究所 抗疟新药—复方蒿甲醚及其制备方法

Also Published As

Publication number Publication date
HK1035712A1 (en) 2001-12-07
BRPI9912208B1 (pt) 2016-04-19
CO5040050A1 (es) 2001-05-29
ID27500A (id) 2001-04-12
US20010014699A1 (en) 2001-08-16
BR9912208A (pt) 2001-04-10
EP1089961A1 (de) 2001-04-11
JP2002518467A (ja) 2002-06-25
JP4355450B2 (ja) 2009-11-04
PE20000703A1 (es) 2000-08-23
CN1183097C (zh) 2005-01-05
CA2335685C (en) 2009-08-11
WO1999067197A1 (en) 1999-12-29
TW200528419A (en) 2005-09-01
TWI250141B (en) 2006-03-01
EP1089961B1 (de) 2004-02-11
US6329552B2 (en) 2001-12-11
AU4776399A (en) 2000-01-10
BRPI9912208B8 (pt) 2021-05-25
CA2335685A1 (en) 1999-12-29
MY117662A (en) 2004-07-31
ES2216528T3 (es) 2004-10-16
PT1089961E (pt) 2004-06-30
CN1312794A (zh) 2001-09-12

Similar Documents

Publication Publication Date Title
DK0931788T3 (da) Metalloproteasehæmmere
TR200000065T2 (tr) Epotilon türevleri.
ATE491703T1 (de) Phthalazinonderivate
ATE430563T1 (de) Cyano-substituierte oleanolsäure als inhibitor der no-produktion
DE69705874T2 (de) Verwendung von Östrogenantagonisten und - agonisten zur Hemmung pathologischer Zustände
ES8401031A1 (es) Una tetrahidroftalimida.
EA199800141A1 (ru) Гетероциклические соединения
BR0313686A (pt) Compostos quìmicos
HUP0101688A2 (hu) Heterociklussal szubsztituált amidok és alkalmazásuk gyógyszerkészítmények előállítására
EA200100310A1 (ru) Кислородсодержащие гетероциклические соединения
DE60014043D1 (de) Flouride von 4-substituierten piperidin-derivaten
DK1706414T3 (da) Fremgangsmåde til fluorcytidinderivater
DE69824450D1 (de) Biphenylamidin-derivate
EA200301317A1 (ru) Производные аминохинолина и его применение в качестве лигандов аденозина a3
ATE550332T1 (de) 4-imidazolin-2-onverbindungen als p38-map- kinaseinhibitors
DE60034577D1 (de) In 4-stellung substituierte piperidinderivate
ATE71619T1 (de) Pyridazinon-derivate.
ES2160158T3 (es) Derivados de 4-indol-1-il acido butirico, su preparacion y su utilizacion como inhibidores de receptores alfa1-adrenergicos y testosterona 5alfa-reductasas.
ATE259346T1 (de) Benflumentolderivative und ihre verwendung gegen parasitäre protozoen und trematoden
EA200001036A1 (ru) Способы ингибирования mrp1
BR0013409B1 (pt) compostos fungicidas possuindo uma porção flúorvinil ou fluorpropenil-oxifeniloxima e processo para preparação dos mesmos.
DE60221250D1 (de) Bis(5-aryl-2-pyridyl)derivate
ATE284379T1 (de) Aminderivate
ATE340175T1 (de) Imidazo(4,5-böchinolinderivate und ihre verwendung als inhibitoren der induzierbaren no- synthase
ECSP993035A (es) Compuestos organicos

Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification

Ref document number: 1089961

Country of ref document: EP