TNSN05324A1 - 7-substituted 3-nitro-pyrazolo `1,5-a! pyrimidines - Google Patents

7-substituted 3-nitro-pyrazolo `1,5-a! pyrimidines

Info

Publication number
TNSN05324A1
TNSN05324A1 TNP2005000324A TNSN05324A TNSN05324A1 TN SN05324 A1 TNSN05324 A1 TN SN05324A1 TN P2005000324 A TNP2005000324 A TN P2005000324A TN SN05324 A TNSN05324 A TN SN05324A TN SN05324 A1 TNSN05324 A1 TN SN05324A1
Authority
TN
Tunisia
Prior art keywords
pyrazolo
pyrimidines
nitro
substituted
compounds
Prior art date
Application number
TNP2005000324A
Inventor
Luis Anglada
Albert Palomer
Marta Princep
Antonio Guglietta
Original Assignee
Ferrer Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/EP2004/008207 external-priority patent/WO2005014596A1/en
Application filed by Ferrer Int filed Critical Ferrer Int
Publication of TNSN05324A1 publication Critical patent/TNSN05324A1/en

Links

Landscapes

  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

The present invention relates to compounds of Formula (I): wherein R1 is as defined in the claims. The compounds have specific affinity for the GABAA receptor and are therefore useful in the treatment and prevention of diseases modulated by the alpha1- and alpha 2- GABAA receptors.
TNP2005000324A 2003-07-24 2005-12-22 7-substituted 3-nitro-pyrazolo `1,5-a! pyrimidines TNSN05324A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ES200301747A ES2222814B1 (en) 2003-07-24 2003-07-24 3-NITRO-PIRAZOLO (1,5-A) PYRIMIDINS 7-REPLACED AND RELATED COMPOSITIONS AND METHODS.
PCT/EP2004/008207 WO2005014596A1 (en) 2003-07-24 2004-07-22 7-substituted 3-nitro-pyrazolo `1,5-a! pyrimidines

Publications (1)

Publication Number Publication Date
TNSN05324A1 true TNSN05324A1 (en) 2007-07-10

Family

ID=34354826

Family Applications (1)

Application Number Title Priority Date Filing Date
TNP2005000324A TNSN05324A1 (en) 2003-07-24 2005-12-22 7-substituted 3-nitro-pyrazolo `1,5-a! pyrimidines

Country Status (11)

Country Link
CN (1) CN1829720A (en)
AR (1) AR045088A1 (en)
CL (1) CL2004001813A1 (en)
EA (1) EA200600318A1 (en)
ES (2) ES2222814B1 (en)
IL (1) IL173347A0 (en)
MA (1) MA27945A1 (en)
PA (1) PA8607401A1 (en)
PE (1) PE20050722A1 (en)
TN (1) TNSN05324A1 (en)
ZA (1) ZA200600471B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006084835A1 (en) * 2005-02-10 2006-08-17 Ferrer Internacional, S. A. N-(3-(imidazo [1,5-a]pyrimidin-4-yl)phenyl]-sulfonamides and n-[3-(imidazo[1,5-a]pyrimidin-4-yl)-phenyl]-carboxamides and their use as gabaa receptor modulators

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4626538A (en) * 1983-06-23 1986-12-02 American Cyanamid Company [7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidines
NZ208554A (en) * 1983-06-23 1987-06-30 American Cyanamid Co (aryl and heteroaryl)-(7-(aryl and heteroaryl)-pyrazolo (1,5-a) pyrimidin-3-yl)-methanone derivatives and pharmaceutical compositions

Also Published As

Publication number Publication date
CL2004001813A1 (en) 2005-06-03
CN1829720A (en) 2006-09-06
EA200600318A1 (en) 2006-06-30
ES2222814A1 (en) 2005-02-01
ES2245893B1 (en) 2006-12-01
IL173347A0 (en) 2006-06-11
PA8607401A1 (en) 2006-08-03
ES2222814B1 (en) 2005-12-01
AR045088A1 (en) 2005-10-12
MA27945A1 (en) 2006-06-01
ES2245893A1 (en) 2006-01-16
PE20050722A1 (en) 2005-09-14
ZA200600471B (en) 2007-04-25

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