TNSN05324A1 - 7-substituted 3-nitro-pyrazolo `1,5-a! pyrimidines - Google Patents
7-substituted 3-nitro-pyrazolo `1,5-a! pyrimidinesInfo
- Publication number
- TNSN05324A1 TNSN05324A1 TNP2005000324A TNSN05324A TNSN05324A1 TN SN05324 A1 TNSN05324 A1 TN SN05324A1 TN P2005000324 A TNP2005000324 A TN P2005000324A TN SN05324 A TNSN05324 A TN SN05324A TN SN05324 A1 TNSN05324 A1 TN SN05324A1
- Authority
- TN
- Tunisia
- Prior art keywords
- pyrazolo
- pyrimidines
- nitro
- substituted
- compounds
- Prior art date
Links
Landscapes
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
The present invention relates to compounds of Formula (I): wherein R1 is as defined in the claims. The compounds have specific affinity for the GABAA receptor and are therefore useful in the treatment and prevention of diseases modulated by the alpha1- and alpha 2- GABAA receptors.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ES200301747A ES2222814B1 (en) | 2003-07-24 | 2003-07-24 | 3-NITRO-PIRAZOLO (1,5-A) PYRIMIDINS 7-REPLACED AND RELATED COMPOSITIONS AND METHODS. |
PCT/EP2004/008207 WO2005014596A1 (en) | 2003-07-24 | 2004-07-22 | 7-substituted 3-nitro-pyrazolo `1,5-a! pyrimidines |
Publications (1)
Publication Number | Publication Date |
---|---|
TNSN05324A1 true TNSN05324A1 (en) | 2007-07-10 |
Family
ID=34354826
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TNP2005000324A TNSN05324A1 (en) | 2003-07-24 | 2005-12-22 | 7-substituted 3-nitro-pyrazolo `1,5-a! pyrimidines |
Country Status (11)
Country | Link |
---|---|
CN (1) | CN1829720A (en) |
AR (1) | AR045088A1 (en) |
CL (1) | CL2004001813A1 (en) |
EA (1) | EA200600318A1 (en) |
ES (2) | ES2222814B1 (en) |
IL (1) | IL173347A0 (en) |
MA (1) | MA27945A1 (en) |
PA (1) | PA8607401A1 (en) |
PE (1) | PE20050722A1 (en) |
TN (1) | TNSN05324A1 (en) |
ZA (1) | ZA200600471B (en) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2006084835A1 (en) * | 2005-02-10 | 2006-08-17 | Ferrer Internacional, S. A. | N-(3-(imidazo [1,5-a]pyrimidin-4-yl)phenyl]-sulfonamides and n-[3-(imidazo[1,5-a]pyrimidin-4-yl)-phenyl]-carboxamides and their use as gabaa receptor modulators |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4626538A (en) * | 1983-06-23 | 1986-12-02 | American Cyanamid Company | [7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidines |
NZ208554A (en) * | 1983-06-23 | 1987-06-30 | American Cyanamid Co | (aryl and heteroaryl)-(7-(aryl and heteroaryl)-pyrazolo (1,5-a) pyrimidin-3-yl)-methanone derivatives and pharmaceutical compositions |
-
2003
- 2003-07-24 ES ES200301747A patent/ES2222814B1/en not_active Expired - Fee Related
-
2004
- 2004-07-12 ES ES200401696A patent/ES2245893B1/en not_active Expired - Fee Related
- 2004-07-20 CL CL200401813A patent/CL2004001813A1/en unknown
- 2004-07-20 PA PA8607401A patent/PA8607401A1/en unknown
- 2004-07-22 CN CN 200480021467 patent/CN1829720A/en active Pending
- 2004-07-22 EA EA200600318A patent/EA200600318A1/en unknown
- 2004-07-22 ZA ZA200600471A patent/ZA200600471B/en unknown
- 2004-07-23 PE PE2004000711A patent/PE20050722A1/en not_active Application Discontinuation
- 2004-07-23 AR ARP040102618 patent/AR045088A1/en unknown
-
2005
- 2005-12-22 TN TNP2005000324A patent/TNSN05324A1/en unknown
-
2006
- 2006-01-24 IL IL173347A patent/IL173347A0/en unknown
- 2006-02-13 MA MA28798A patent/MA27945A1/en unknown
Also Published As
Publication number | Publication date |
---|---|
CL2004001813A1 (en) | 2005-06-03 |
CN1829720A (en) | 2006-09-06 |
EA200600318A1 (en) | 2006-06-30 |
ES2222814A1 (en) | 2005-02-01 |
ES2245893B1 (en) | 2006-12-01 |
IL173347A0 (en) | 2006-06-11 |
PA8607401A1 (en) | 2006-08-03 |
ES2222814B1 (en) | 2005-12-01 |
AR045088A1 (en) | 2005-10-12 |
MA27945A1 (en) | 2006-06-01 |
ES2245893A1 (en) | 2006-01-16 |
PE20050722A1 (en) | 2005-09-14 |
ZA200600471B (en) | 2007-04-25 |
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