EA200600318A1 - DERIVATIVES 3-NITROPYRAZOLO [1,5-a] PYRIMIDINES, METHOD OF THEIR PRODUCTION, MEDICATION (OPTIONS) AND METHOD OF TREATMENT OR PREVENTION OF DISEASE - Google Patents

DERIVATIVES 3-NITROPYRAZOLO [1,5-a] PYRIMIDINES, METHOD OF THEIR PRODUCTION, MEDICATION (OPTIONS) AND METHOD OF TREATMENT OR PREVENTION OF DISEASE

Info

Publication number
EA200600318A1
EA200600318A1 EA200600318A EA200600318A EA200600318A1 EA 200600318 A1 EA200600318 A1 EA 200600318A1 EA 200600318 A EA200600318 A EA 200600318A EA 200600318 A EA200600318 A EA 200600318A EA 200600318 A1 EA200600318 A1 EA 200600318A1
Authority
EA
Eurasian Patent Office
Prior art keywords
prevention
treatment
nitropyrazolo
pyrimidines
medication
Prior art date
Application number
EA200600318A
Other languages
Russian (ru)
Inventor
Луис Англада
Антонио Гугльетта
Альберт Паломер
Марта Принсеп
Original Assignee
Феррер Интернасионал, С.А.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Феррер Интернасионал, С.А. filed Critical Феррер Интернасионал, С.А.
Priority claimed from PCT/EP2004/008207 external-priority patent/WO2005014596A1/en
Publication of EA200600318A1 publication Critical patent/EA200600318A1/en

Links

Abstract

Настоящее изобретение относится к соединениям формулы (I)где Rимеет значение, как определено в описании изобретения. Соединения проявляют специфическую аффинность к рецептору ГАМКи, следовательно, их можно использовать для лечения и профилактики заболеваний, связанных с модуляцией рецептора α-ГАМКи α-ГАМК.The present invention relates to compounds of formula (I) where R has the meaning as defined in the description. The compounds exhibit specific affinity for the GABA receptor, therefore, they can be used for the treatment and prevention of diseases associated with the modulation of the α-GABA and α-GABA receptor.

EA200600318A 2003-07-24 2004-07-22 DERIVATIVES 3-NITROPYRAZOLO [1,5-a] PYRIMIDINES, METHOD OF THEIR PRODUCTION, MEDICATION (OPTIONS) AND METHOD OF TREATMENT OR PREVENTION OF DISEASE EA200600318A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
ES200301747A ES2222814B1 (en) 2003-07-24 2003-07-24 3-NITRO-PIRAZOLO (1,5-A) PYRIMIDINS 7-REPLACED AND RELATED COMPOSITIONS AND METHODS.
ES200401696A ES2245893B1 (en) 2003-07-24 2004-07-12 IMPROVEMENTS IN THE OBJECT OF THE INVENTION PATENT N.P200301747 REFERRING TO "3-NITRO-PIRAZOLO (1,5-A) 7-REPLACED PYRIMIDINES AND RELATED COMPOSITIONS AND METHODS".
PCT/EP2004/008207 WO2005014596A1 (en) 2003-07-24 2004-07-22 7-substituted 3-nitro-pyrazolo `1,5-a! pyrimidines

Publications (1)

Publication Number Publication Date
EA200600318A1 true EA200600318A1 (en) 2006-06-30

Family

ID=34354826

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200600318A EA200600318A1 (en) 2003-07-24 2004-07-22 DERIVATIVES 3-NITROPYRAZOLO [1,5-a] PYRIMIDINES, METHOD OF THEIR PRODUCTION, MEDICATION (OPTIONS) AND METHOD OF TREATMENT OR PREVENTION OF DISEASE

Country Status (11)

Country Link
CN (1) CN1829720A (en)
AR (1) AR045088A1 (en)
CL (1) CL2004001813A1 (en)
EA (1) EA200600318A1 (en)
ES (2) ES2222814B1 (en)
IL (1) IL173347A0 (en)
MA (1) MA27945A1 (en)
PA (1) PA8607401A1 (en)
PE (1) PE20050722A1 (en)
TN (1) TNSN05324A1 (en)
ZA (1) ZA200600471B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006084835A1 (en) * 2005-02-10 2006-08-17 Ferrer Internacional, S. A. N-(3-(imidazo [1,5-a]pyrimidin-4-yl)phenyl]-sulfonamides and n-[3-(imidazo[1,5-a]pyrimidin-4-yl)-phenyl]-carboxamides and their use as gabaa receptor modulators

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4626538A (en) * 1983-06-23 1986-12-02 American Cyanamid Company [7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidines
NZ208554A (en) * 1983-06-23 1987-06-30 American Cyanamid Co (aryl and heteroaryl)-(7-(aryl and heteroaryl)-pyrazolo (1,5-a) pyrimidin-3-yl)-methanone derivatives and pharmaceutical compositions

Also Published As

Publication number Publication date
ES2245893B1 (en) 2006-12-01
IL173347A0 (en) 2006-06-11
ES2222814A1 (en) 2005-02-01
TNSN05324A1 (en) 2007-07-10
CN1829720A (en) 2006-09-06
CL2004001813A1 (en) 2005-06-03
ES2222814B1 (en) 2005-12-01
MA27945A1 (en) 2006-06-01
PE20050722A1 (en) 2005-09-14
PA8607401A1 (en) 2006-08-03
ZA200600471B (en) 2007-04-25
AR045088A1 (en) 2005-10-12
ES2245893A1 (en) 2006-01-16

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