EA200600318A1 - DERIVATIVES 3-NITROPYRAZOLO [1,5-a] PYRIMIDINES, METHOD OF THEIR PRODUCTION, MEDICATION (OPTIONS) AND METHOD OF TREATMENT OR PREVENTION OF DISEASE - Google Patents
DERIVATIVES 3-NITROPYRAZOLO [1,5-a] PYRIMIDINES, METHOD OF THEIR PRODUCTION, MEDICATION (OPTIONS) AND METHOD OF TREATMENT OR PREVENTION OF DISEASEInfo
- Publication number
- EA200600318A1 EA200600318A1 EA200600318A EA200600318A EA200600318A1 EA 200600318 A1 EA200600318 A1 EA 200600318A1 EA 200600318 A EA200600318 A EA 200600318A EA 200600318 A EA200600318 A EA 200600318A EA 200600318 A1 EA200600318 A1 EA 200600318A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- prevention
- treatment
- nitropyrazolo
- pyrimidines
- medication
- Prior art date
Links
Abstract
Настоящее изобретение относится к соединениям формулы (I)где Rимеет значение, как определено в описании изобретения. Соединения проявляют специфическую аффинность к рецептору ГАМКи, следовательно, их можно использовать для лечения и профилактики заболеваний, связанных с модуляцией рецептора α-ГАМКи α-ГАМК.The present invention relates to compounds of formula (I) where R has the meaning as defined in the description. The compounds exhibit specific affinity for the GABA receptor, therefore, they can be used for the treatment and prevention of diseases associated with the modulation of the α-GABA and α-GABA receptor.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ES200301747A ES2222814B1 (en) | 2003-07-24 | 2003-07-24 | 3-NITRO-PIRAZOLO (1,5-A) PYRIMIDINS 7-REPLACED AND RELATED COMPOSITIONS AND METHODS. |
ES200401696A ES2245893B1 (en) | 2003-07-24 | 2004-07-12 | IMPROVEMENTS IN THE OBJECT OF THE INVENTION PATENT N.P200301747 REFERRING TO "3-NITRO-PIRAZOLO (1,5-A) 7-REPLACED PYRIMIDINES AND RELATED COMPOSITIONS AND METHODS". |
PCT/EP2004/008207 WO2005014596A1 (en) | 2003-07-24 | 2004-07-22 | 7-substituted 3-nitro-pyrazolo `1,5-a! pyrimidines |
Publications (1)
Publication Number | Publication Date |
---|---|
EA200600318A1 true EA200600318A1 (en) | 2006-06-30 |
Family
ID=34354826
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200600318A EA200600318A1 (en) | 2003-07-24 | 2004-07-22 | DERIVATIVES 3-NITROPYRAZOLO [1,5-a] PYRIMIDINES, METHOD OF THEIR PRODUCTION, MEDICATION (OPTIONS) AND METHOD OF TREATMENT OR PREVENTION OF DISEASE |
Country Status (11)
Country | Link |
---|---|
CN (1) | CN1829720A (en) |
AR (1) | AR045088A1 (en) |
CL (1) | CL2004001813A1 (en) |
EA (1) | EA200600318A1 (en) |
ES (2) | ES2222814B1 (en) |
IL (1) | IL173347A0 (en) |
MA (1) | MA27945A1 (en) |
PA (1) | PA8607401A1 (en) |
PE (1) | PE20050722A1 (en) |
TN (1) | TNSN05324A1 (en) |
ZA (1) | ZA200600471B (en) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2006084835A1 (en) * | 2005-02-10 | 2006-08-17 | Ferrer Internacional, S. A. | N-(3-(imidazo [1,5-a]pyrimidin-4-yl)phenyl]-sulfonamides and n-[3-(imidazo[1,5-a]pyrimidin-4-yl)-phenyl]-carboxamides and their use as gabaa receptor modulators |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4626538A (en) * | 1983-06-23 | 1986-12-02 | American Cyanamid Company | [7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidines |
NZ208554A (en) * | 1983-06-23 | 1987-06-30 | American Cyanamid Co | (aryl and heteroaryl)-(7-(aryl and heteroaryl)-pyrazolo (1,5-a) pyrimidin-3-yl)-methanone derivatives and pharmaceutical compositions |
-
2003
- 2003-07-24 ES ES200301747A patent/ES2222814B1/en not_active Expired - Fee Related
-
2004
- 2004-07-12 ES ES200401696A patent/ES2245893B1/en not_active Expired - Fee Related
- 2004-07-20 PA PA8607401A patent/PA8607401A1/en unknown
- 2004-07-20 CL CL200401813A patent/CL2004001813A1/en unknown
- 2004-07-22 CN CN 200480021467 patent/CN1829720A/en active Pending
- 2004-07-22 EA EA200600318A patent/EA200600318A1/en unknown
- 2004-07-22 ZA ZA200600471A patent/ZA200600471B/en unknown
- 2004-07-23 AR ARP040102618 patent/AR045088A1/en unknown
- 2004-07-23 PE PE2004000711A patent/PE20050722A1/en not_active Application Discontinuation
-
2005
- 2005-12-22 TN TNP2005000324A patent/TNSN05324A1/en unknown
-
2006
- 2006-01-24 IL IL173347A patent/IL173347A0/en unknown
- 2006-02-13 MA MA28798A patent/MA27945A1/en unknown
Also Published As
Publication number | Publication date |
---|---|
ES2245893B1 (en) | 2006-12-01 |
IL173347A0 (en) | 2006-06-11 |
ES2222814A1 (en) | 2005-02-01 |
TNSN05324A1 (en) | 2007-07-10 |
CN1829720A (en) | 2006-09-06 |
CL2004001813A1 (en) | 2005-06-03 |
ES2222814B1 (en) | 2005-12-01 |
MA27945A1 (en) | 2006-06-01 |
PE20050722A1 (en) | 2005-09-14 |
PA8607401A1 (en) | 2006-08-03 |
ZA200600471B (en) | 2007-04-25 |
AR045088A1 (en) | 2005-10-12 |
ES2245893A1 (en) | 2006-01-16 |
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