TH134759A - A new type of derivative of pyrazole steroid [3,2-C] with a measure of the chemical reactivity of glucocorticoids. - Google Patents

A new type of derivative of pyrazole steroid [3,2-C] with a measure of the chemical reactivity of glucocorticoids.

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Publication number
TH134759A
TH134759A TH1101002479A TH1101002479A TH134759A TH 134759 A TH134759 A TH 134759A TH 1101002479 A TH1101002479 A TH 1101002479A TH 1101002479 A TH1101002479 A TH 1101002479A TH 134759 A TH134759 A TH 134759A
Authority
TH
Thailand
Prior art keywords
glucocorticoids
pyrazole
steroid
derivative
measure
Prior art date
Application number
TH1101002479A
Other languages
Thai (th)
Other versions
TH134759B (en
Inventor
บลาดห์
เฮแคน
เบิร์กแคมป์
แฟรงค์
กาบอส
บาลินท์
ฮันเซน
ปีเตอร์
โรเบิร์ต
Original Assignee
นายธีรพล สุวรรณประทีป
นางสาวสยุมพร สุจินตัย
Filing date
Publication date
Application filed by นายธีรพล สุวรรณประทีป, นางสาวสยุมพร สุจินตัย filed Critical นายธีรพล สุวรรณประทีป
Publication of TH134759B publication Critical patent/TH134759B/en
Publication of TH134759A publication Critical patent/TH134759A/en

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Abstract

DC60 (12/02/55) การประดิษฐ์นี้จัดหาสารประกอบของสูตรผสม (I) (สูตรเคมี) (I) และสารผสมทางเภสัชกรรมที่มีสารดังกล่าวและการนำไปใช้รักษาโรค การประดิษฐ์นี้จัดหาสารประกอบของสูตรผสม(I) (สูตรเคมี) และสารผสมทางเภสัชกรรมที่มีสารดังกล่าวและการนำไปใช้รักษาโรค สิทธิบัตรยา DC60 (12/02/55) This invention provides compound formulation compounds (I) (chemical formulas) (I) and pharmaceutical mixtures containing such substances and their therapeutic use. This invention provides a compound (I) compound (chemical formula) and a pharmaceutical mixtures containing such substances and their therapeutic application.

Claims (1)

1.สารประกอบที่เลือกจากกลุ่มซึ่งประกอบด้วย: (1R,2R,3aS,3bS,10aS,10bR,11S,12aS)-10b-ฟลูออโร-1-{[(ฟลูออโรเมทอล)ซัลฟานิล] คาร์บอนิล}-7-(6-ฟลูออโรไพริดิน-3-อิล)-11-ไฮดรอกซี-2,10a,12a-ไตรเมทิล- 1,2,3,3a,3b,4,5,7,10,10a,10b,11,12,12a-เททราเดคาไฮโดรไซโคลเพนทา[5,6]แนพโท[1,2-f] อินดาซอล-1-อิล เมทอกซีอะซิเตท, (1R,2R,3aS,3bS,10aS,10bR,11S,12aS)-10b-ฟลูออโร-1-{[(ฟลูออโรเมทอล)ซัลฟานิล] คาร์บอนิล}-7-(6-ฟลูออโรไพริดิน-3-อิล)-11-ไฮดรอกซี-2,10a,12a-ไตรเมทิล- 1,2,3,3a,3b,4,5,7,1แท็ก : สิทธิบัตรยา1. Compounds selected from the group consisting of: (1R, 2R, 3aS, 3bS, 10aS, 10bR, 11S, 12aS) -10b-fluoro-1 - (((fluoromethol) sulfanyl. ] Carbonyl} -7- (6-fluoropyridin-3-il) -11-hydroxy -2,10a, 12a-trimethyl- 1,2,3,3a, 3b, 4,5,7,10,10a, 10b, 11,12,12a-tetradeca, hydrocyclopenta [5,6] naphtho [1,2-f] indasol. -1- il Methyl acetate, (1R, 2R, 3aS, 3bS, 10aS, 10bR, 11S, 12aS) -10b-fluoro-1 - (((fluoromethol) sulfanyl) kha Carbonyl) -7- (6-fluoropyridin-3-il) -11-hydroxy -2,10a, 12a-trimethyl-1,2,3,3a, 3b, 4,5,7,1 Tag: Drug Patents
TH1101002479A 2010-04-01 A new type of derivative of pyrazole steroid [3,2-C] with a measure of the chemical reactivity of glucocorticoids. TH134759A (en)

Publications (2)

Publication Number Publication Date
TH134759B TH134759B (en) 2014-06-11
TH134759A true TH134759A (en) 2014-06-11

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