SK52393A3 - Novel pilocarpine erivatives and process for their preparation - Google Patents
Novel pilocarpine erivatives and process for their preparation Download PDFInfo
- Publication number
- SK52393A3 SK52393A3 SK523-93A SK52393A SK52393A3 SK 52393 A3 SK52393 A3 SK 52393A3 SK 52393 A SK52393 A SK 52393A SK 52393 A3 SK52393 A3 SK 52393A3
- Authority
- SK
- Slovakia
- Prior art keywords
- formula
- acid
- compound
- defined above
- pilocarpine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Ophthalmology & Optometry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FI905930A FI98815C (fi) | 1990-11-30 | 1990-11-30 | Menetelmä uusien, farmakologisesti käyttökelpoisten bispilokarpiinihapon esterijohdannaisten valmistamiseksi |
PCT/FI1991/000359 WO1992009583A1 (en) | 1990-11-30 | 1991-11-27 | Novel pilocarpine derivatives and process for their preparation |
Publications (1)
Publication Number | Publication Date |
---|---|
SK52393A3 true SK52393A3 (en) | 1994-01-12 |
Family
ID=8531500
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SK523-93A SK52393A3 (en) | 1990-11-30 | 1991-11-27 | Novel pilocarpine erivatives and process for their preparation |
Country Status (19)
Country | Link |
---|---|
EP (1) | EP0559700B1 (fi) |
JP (1) | JP3094232B2 (fi) |
KR (1) | KR930703264A (fi) |
AT (1) | ATE192144T1 (fi) |
AU (1) | AU664958B2 (fi) |
CA (1) | CA2096444A1 (fi) |
CZ (1) | CZ282229B6 (fi) |
DE (1) | DE69132143T2 (fi) |
EE (1) | EE9400143A (fi) |
FI (1) | FI98815C (fi) |
HU (1) | HUT67273A (fi) |
LT (1) | LT3532B (fi) |
LV (1) | LV10094B (fi) |
NO (1) | NO304228B1 (fi) |
NZ (1) | NZ240781A (fi) |
PL (2) | PL167773B1 (fi) |
RU (1) | RU2100352C1 (fi) |
SK (1) | SK52393A3 (fi) |
WO (1) | WO1992009583A1 (fi) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0642501A1 (en) * | 1992-05-29 | 1995-03-15 | Leiras Oy | Novel pilocarpine derivatives and process for their preparation |
GB9310965D0 (en) * | 1993-05-27 | 1993-07-14 | Ucb Sa | 2-hydroxy-3-(1h-imidazol-4-yl)alkyl)benzenecarboximidamides |
SE501482C2 (sv) | 1993-06-24 | 1995-02-27 | Leiras Oy | Komposition för topisk administration av bispilokarpinsyradiestrar till ögat i form av en vattenlösning |
SE9302201D0 (sv) | 1993-06-24 | 1993-06-24 | Leiras Oy | Composition for ophthalmic use |
AU6973094A (en) * | 1993-06-24 | 1995-01-17 | Leiras Oy | Composition for ophthalmic use |
DE4334135A1 (de) * | 1993-10-07 | 1995-04-13 | Merck Patent Gmbh | Verfahren zur Herstellung von Pilocarpin-Derivaten |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4061722A (en) | 1976-04-26 | 1977-12-06 | Interx Research Corporation | Selected quaternary ammonium salts of pilocarpine useful in reducing intraocular pressure in warm-blooded animals |
IL69593A (en) * | 1982-09-17 | 1988-09-30 | Bundegaard Hans | Pilocarpine prodrugs,their preparation and pharmaceutical compositions containing them |
-
1990
- 1990-11-30 FI FI905930A patent/FI98815C/fi not_active IP Right Cessation
-
1991
- 1991-11-27 PL PL91299375A patent/PL167773B1/pl unknown
- 1991-11-27 RU RU93041054/04A patent/RU2100352C1/ru not_active IP Right Cessation
- 1991-11-27 CA CA002096444A patent/CA2096444A1/en not_active Abandoned
- 1991-11-27 JP JP04500392A patent/JP3094232B2/ja not_active Expired - Fee Related
- 1991-11-27 HU HU9301569A patent/HUT67273A/hu unknown
- 1991-11-27 SK SK523-93A patent/SK52393A3/sk unknown
- 1991-11-27 WO PCT/FI1991/000359 patent/WO1992009583A1/en active IP Right Grant
- 1991-11-27 EP EP91920512A patent/EP0559700B1/en not_active Expired - Lifetime
- 1991-11-27 DE DE69132143T patent/DE69132143T2/de not_active Expired - Fee Related
- 1991-11-27 CZ CS931025A patent/CZ282229B6/cs not_active IP Right Cessation
- 1991-11-27 PL PL91308270A patent/PL168715B1/pl unknown
- 1991-11-27 KR KR1019930701611A patent/KR930703264A/ko not_active Application Discontinuation
- 1991-11-27 AU AU89398/91A patent/AU664958B2/en not_active Ceased
- 1991-11-27 AT AT91920512T patent/ATE192144T1/de not_active IP Right Cessation
- 1991-11-28 NZ NZ240781A patent/NZ240781A/xx unknown
-
1993
- 1993-05-28 LV LVP-93-436A patent/LV10094B/en unknown
- 1993-05-28 LT LTIP577A patent/LT3532B/lt not_active IP Right Cessation
- 1993-05-28 NO NO931960A patent/NO304228B1/no not_active IP Right Cessation
-
1994
- 1994-11-16 EE EE9400143A patent/EE9400143A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
LV10094A (lv) | 1994-05-10 |
CZ282229B6 (cs) | 1997-06-11 |
FI905930A0 (fi) | 1990-11-30 |
LV10094B (en) | 1995-02-20 |
CZ102593A3 (en) | 1994-04-13 |
NO931960L (no) | 1993-05-28 |
FI98815C (fi) | 1997-08-25 |
PL168715B1 (pl) | 1996-03-29 |
ATE192144T1 (de) | 2000-05-15 |
LT3532B (en) | 1995-11-27 |
NO304228B1 (no) | 1998-11-16 |
CA2096444A1 (en) | 1992-05-31 |
DE69132143D1 (de) | 2000-05-31 |
EP0559700A1 (en) | 1993-09-15 |
FI98815B (fi) | 1997-05-15 |
HU9301569D0 (en) | 1993-09-28 |
AU8939891A (en) | 1992-06-25 |
HUT67273A (en) | 1995-03-28 |
EE9400143A (et) | 1995-12-15 |
PL167773B1 (pl) | 1995-11-30 |
NO931960D0 (no) | 1993-05-28 |
KR930703264A (ko) | 1993-11-29 |
WO1992009583A1 (en) | 1992-06-11 |
EP0559700B1 (en) | 2000-04-26 |
AU664958B2 (en) | 1995-12-07 |
RU2100352C1 (ru) | 1997-12-27 |
JPH06504270A (ja) | 1994-05-19 |
JP3094232B2 (ja) | 2000-10-03 |
FI905930A (fi) | 1992-05-31 |
DE69132143T2 (de) | 2000-12-14 |
LTIP577A (en) | 1994-12-27 |
NZ240781A (en) | 1993-12-23 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
US6589959B1 (en) | Crystalline bis[(e)-7-[4-(4-fluorophenyl)-6-isopropyl-2-[methyl(methylsulfonyl)amino]pyrimidin-5-yl](3R,5S)-3,5-dihydroxyhept-6-enoic acid]calcium salt | |
CZ300410B6 (cs) | 1,4-Benzothiazepin-1,1-dioxidové deriváty, tyto deriváty pro použití jako léciva, léciva tyto deriváty obsahující, zpusob prípravy techto léciv a použití techto derivátu pro prípravu léciv | |
SU1138024A3 (ru) | Способ получени аминопроизводных пиридазина | |
WO2010105910A1 (en) | Fosfluconazole derivatives, synthesis, and use in long acting formulations | |
SK52393A3 (en) | Novel pilocarpine erivatives and process for their preparation | |
EP0087378B1 (fr) | Ethers-oximes d'alcoylaminoalcools comme médicaments, produits nouveaux et procédés pour leur préparation | |
JP2013545728A (ja) | 抗菌性ポリエーテルおよびポリオール化合物 | |
JPH026497A (ja) | ホスホノアルキルプリン誘導体類 | |
JPS6119620B2 (fi) | ||
KR900006124B1 (ko) | Gem-디할로 및 테트라할로-1,12-디아미노-4,9-디아자-도데칸 및 이들의 제조방법 | |
KR900006132B1 (ko) | 젬-디할로-1,8-디아미노-4-아자-옥탄 및 이의 제조방법 | |
JPS6218545B2 (fi) | ||
US5436350A (en) | Bispilocarpic acid ester derivatives and process for their preparation | |
FI98910C (fi) | Menetelmä farmaseuttisesti käyttökelpoisten pilokarpiinijohdannaisten valmistamiseksi | |
WO2010100199A1 (en) | Fluconazole carboxylic ester derivatives, synthesis, and use in long acting formulations | |
LV10257B (en) | Novel pilocarpine derivatives and process for their preparation | |
GB1565021A (en) | Pharmaceutical compositions containing alkylamine deratives | |
HU189439B (en) | Process for producing triazol compounds | |
SU963470A3 (ru) | Способ получени N @ -четвертичных производных 10-бромаймалина и 10-бромизоаймалина | |
JP2602887B2 (ja) | 新規含フッ素3−ニトロ−1,2,4−トリアゾールおよびそれを含む放射線増感剤 | |
EA027979B1 (ru) | N-оксидированный сополимер n-винилпирролидона и 2-метил-5-винилпиридина | |
NO161736B (no) | Analogifremgangsmaate for fremstilling av nye derivater av1-alkylamin-3(4(p-alkyloksybenzamid)fenoksy)-2-propanol med beta-sympatolytisk aktivitet. | |
JPH08104680A (ja) | 2−アリール−1−(1h−1,2,4−トリアゾー ル−1−イル)ブタン−2−オール誘導体 |