SI0683170T1 - Glucopyranoside benzothiophenes - Google Patents

Glucopyranoside benzothiophenes

Info

Publication number
SI0683170T1
SI0683170T1 SI9530336T SI9530336T SI0683170T1 SI 0683170 T1 SI0683170 T1 SI 0683170T1 SI 9530336 T SI9530336 T SI 9530336T SI 9530336 T SI9530336 T SI 9530336T SI 0683170 T1 SI0683170 T1 SI 0683170T1
Authority
SI
Slovenia
Prior art keywords
benzothiophenes
glucopyranoside
chem
solvate
processes
Prior art date
Application number
SI9530336T
Other languages
English (en)
Slovenian (sl)
Inventor
Jeffrey Alan Dodge
Charles Alan Frolik
Terry Donald Lindstrom
Charles Willis Lugar Iii
Gilbert Stanley Staten
Original Assignee
Eli Lilly And Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly And Company filed Critical Eli Lilly And Company
Publication of SI0683170T1 publication Critical patent/SI0683170T1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/26—Acyclic or carbocyclic radicals, substituted by hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/10—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Steroid Compounds (AREA)
  • Networks Using Active Elements (AREA)
  • Photoreceptors In Electrophotography (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
SI9530336T 1994-05-20 1995-05-16 Glucopyranoside benzothiophenes SI0683170T1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US24665594A 1994-05-20 1994-05-20
EP95303265A EP0683170B1 (en) 1994-05-20 1995-05-16 Glucopyranoside benzothiophenes

Publications (1)

Publication Number Publication Date
SI0683170T1 true SI0683170T1 (en) 2000-02-29

Family

ID=22931623

Family Applications (1)

Application Number Title Priority Date Filing Date
SI9530336T SI0683170T1 (en) 1994-05-20 1995-05-16 Glucopyranoside benzothiophenes

Country Status (27)

Country Link
US (2) US6723739B1 (xx)
EP (1) EP0683170B1 (xx)
JP (1) JPH07316180A (xx)
KR (1) KR950032183A (xx)
CN (1) CN1039013C (xx)
AT (1) ATE184880T1 (xx)
AU (1) AU683734B2 (xx)
BR (1) BR9502079A (xx)
CA (1) CA2149501A1 (xx)
CO (1) CO4650137A1 (xx)
CZ (1) CZ126295A3 (xx)
DE (1) DE69512310T2 (xx)
DK (1) DK0683170T3 (xx)
ES (1) ES2136799T3 (xx)
FI (1) FI952420A (xx)
GR (1) GR3032142T3 (xx)
HU (1) HU219335B (xx)
IL (1) IL113780A (xx)
NO (1) NO304694B1 (xx)
NZ (1) NZ272131A (xx)
PE (1) PE23396A1 (xx)
PL (1) PL308635A1 (xx)
RU (1) RU95107655A (xx)
SI (1) SI0683170T1 (xx)
TW (1) TW323285B (xx)
YU (1) YU31995A (xx)
ZA (1) ZA953975B (xx)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR19980701933A (ko) * 1995-02-06 1998-06-25 피터 쥐. 스트링거 인터루킨-6의 작용의 억제 방법
US20040167080A1 (en) * 1995-03-15 2004-08-26 Dodge Jeffrey A. Glucopyranoside benzothiophenes
CZ300341B6 (cs) 1996-03-26 2009-04-22 Eli Lilly And Company Farmaceutická kompozice obsahující raloxifen
US6458811B1 (en) 1996-03-26 2002-10-01 Eli Lilly And Company Benzothiophenes formulations containing same and methods
DK1175433T3 (da) 1999-05-04 2005-09-19 Strakan Int Ltd Androgenglycosider og androgen aktivitet deraf
DK1212335T3 (da) * 1999-09-13 2006-03-20 Wyeth Corp Glucopyranosid-konjugater af 2-(4-hydroxyphenyl)-1-[4-(2-amin-1-ylethoxy)-benzyl]-1H-indol-5-oler
US6380166B1 (en) 1999-09-13 2002-04-30 American Home Products Corporation Glucopyranosides conjugates of 2-(4-hydroxy-phenyl)-3-methyl-1-[4-(2-amin-1-yl-ethoxy)-benzyl]-1H-indol-5-ols
WO2001027127A1 (en) * 1999-10-08 2001-04-19 Strakan Group Plc Tamoxifen and tamoxifen analogue glycosides and uses thereof
WO2001027129A1 (en) * 1999-10-08 2001-04-19 Strakan Limited Glycosides and orthoester glycosides of raloxifene and analogues and the use thereof
WO2011029088A2 (en) * 2009-09-07 2011-03-10 Dr. Reddy's Laboratories Ltd. Preparation of raloxifene and its salts

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4133814A (en) 1975-10-28 1979-01-09 Eli Lilly And Company 2-Phenyl-3-aroylbenzothiophenes useful as antifertility agents
US4418068A (en) * 1981-04-03 1983-11-29 Eli Lilly And Company Antiestrogenic and antiandrugenic benzothiophenes
TW366342B (en) * 1992-07-28 1999-08-11 Lilly Co Eli The use of 2-phenyl-3-aroylbenzothiophenes in inhibiting bone loss

Also Published As

Publication number Publication date
PL308635A1 (en) 1995-11-27
CZ126295A3 (en) 1995-12-13
ATE184880T1 (de) 1999-10-15
CN1116626A (zh) 1996-02-14
US6723739B1 (en) 2004-04-20
EP0683170A1 (en) 1995-11-22
AU683734B2 (en) 1997-11-20
IL113780A0 (en) 1995-08-31
ZA953975B (en) 1996-11-18
FI952420A (fi) 1995-11-21
CA2149501A1 (en) 1995-11-21
HU219335B (en) 2001-03-28
DE69512310T2 (de) 2000-02-03
DE69512310D1 (de) 1999-10-28
FI952420A0 (fi) 1995-05-18
ES2136799T3 (es) 1999-12-01
HUT73788A (en) 1996-09-30
YU31995A (sh) 1998-12-23
DK0683170T3 (da) 1999-12-20
AU2012195A (en) 1995-11-30
US5567820A (en) 1996-10-22
NZ272131A (en) 1996-11-26
EP0683170B1 (en) 1999-09-22
TW323285B (xx) 1997-12-21
IL113780A (en) 1999-06-20
RU95107655A (ru) 1997-02-10
NO951954L (no) 1995-11-21
BR9502079A (pt) 1996-03-05
PE23396A1 (es) 1996-06-15
KR950032183A (ko) 1995-12-20
HU9501466D0 (en) 1995-06-28
GR3032142T3 (en) 2000-04-27
NO304694B1 (no) 1999-02-01
CN1039013C (zh) 1998-07-08
NO951954D0 (no) 1995-05-18
JPH07316180A (ja) 1995-12-05
CO4650137A1 (es) 1998-09-03

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