CO4650137A1 - Benzotiofenos de glucopiranosido - Google Patents
Benzotiofenos de glucopiranosidoInfo
- Publication number
- CO4650137A1 CO4650137A1 CO95021224A CO95021224A CO4650137A1 CO 4650137 A1 CO4650137 A1 CO 4650137A1 CO 95021224 A CO95021224 A CO 95021224A CO 95021224 A CO95021224 A CO 95021224A CO 4650137 A1 CO4650137 A1 CO 4650137A1
- Authority
- CO
- Colombia
- Prior art keywords
- benzothiophenes
- glucopyranoside
- chem
- solvate
- processes
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/26—Acyclic or carbocyclic radicals, substituted by hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/10—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Steroid Compounds (AREA)
- Photoreceptors In Electrophotography (AREA)
- Networks Using Active Elements (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Abstract
REIVINDICACION NUMERO UN COMPUESTO DE FORMULA FIGURA 1 O UNA DE SUS SALES O SOLVATOS FARMACEUTICAMENTE ACEPTABLES". REIVINDICACION NUMERO UN PROCEDIMIENTO PARA LA PREPARACION DE UN COM- PUESTO DE FORMULA FIGURA 2 EN LA QUE R1 ES HIDROGENO O UN GRUPO DE FORMULA FIGURA 3 Y R2 ES HIDROGENO O UN GRUPO DE FORMULA FIGURA 4 O UNA DE SUS SALES O SOLVATOS, CON LA CONDICION DE QUE UNO DE R1 O R2 ES HIDROGENO, QUE COMPRENDE LA REACCION DE UN COMPUESTO DE FOR- MULA FIGURA 5 EN LA QUE R1, ES UN GRUPO PROTECTOR DE HIDROXI O UN GRUPO DE FORMULA FIGURA 6 O R2, ES UN GRUPO PROTECTOR DE HIDROXI O UN GRUPO DE FORMULA FIGURA 7 O UNA DE SUS SALES O SOLVATOS, CON LA CONDICION DE QUE UNO DE R1, Y R2, ES UN GRUPO PROTECTOR DE HI- DROXI, CON UNA BASE ADECUADA Y UN AGENTE DE SEPA- RACION DEL GRUPO PROTECTOR DE HIDROXI, EN UN DI- SOLVENTE ORGANICO POLAR ADECUADO, DURANTE UN TIEM- PO Y A UNA TEMPERATURA SUFICIENTES PARA PROPORCIO- NAR UN COMPUESTO DE LA FORMULA (II)".
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US24665594A | 1994-05-20 | 1994-05-20 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CO4650137A1 true CO4650137A1 (es) | 1998-09-03 |
Family
ID=22931623
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CO95021224A CO4650137A1 (es) | 1994-05-20 | 1995-05-18 | Benzotiofenos de glucopiranosido |
Country Status (27)
| Country | Link |
|---|---|
| US (2) | US6723739B1 (es) |
| EP (1) | EP0683170B1 (es) |
| JP (1) | JPH07316180A (es) |
| KR (1) | KR950032183A (es) |
| CN (1) | CN1039013C (es) |
| AT (1) | ATE184880T1 (es) |
| AU (1) | AU683734B2 (es) |
| BR (1) | BR9502079A (es) |
| CA (1) | CA2149501A1 (es) |
| CO (1) | CO4650137A1 (es) |
| CZ (1) | CZ126295A3 (es) |
| DE (1) | DE69512310T2 (es) |
| DK (1) | DK0683170T3 (es) |
| ES (1) | ES2136799T3 (es) |
| FI (1) | FI952420A (es) |
| GR (1) | GR3032142T3 (es) |
| HU (1) | HU219335B (es) |
| IL (1) | IL113780A (es) |
| NO (1) | NO304694B1 (es) |
| NZ (1) | NZ272131A (es) |
| PE (1) | PE23396A1 (es) |
| PL (1) | PL308635A1 (es) |
| RU (1) | RU95107655A (es) |
| SI (1) | SI0683170T1 (es) |
| TW (1) | TW323285B (es) |
| YU (1) | YU31995A (es) |
| ZA (1) | ZA953975B (es) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN1173819A (zh) * | 1995-02-06 | 1998-02-18 | 伊莱利利公司 | 抑制il－6作用的方法 |
| US20040167080A1 (en) * | 1995-03-15 | 2004-08-26 | Dodge Jeffrey A. | Glucopyranoside benzothiophenes |
| US6458811B1 (en) | 1996-03-26 | 2002-10-01 | Eli Lilly And Company | Benzothiophenes formulations containing same and methods |
| CZ300341B6 (cs) | 1996-03-26 | 2009-04-22 | Eli Lilly And Company | Farmaceutická kompozice obsahující raloxifen |
| DK1175433T3 (da) | 1999-05-04 | 2005-09-19 | Strakan Int Ltd | Androgenglycosider og androgen aktivitet deraf |
| MXPA02002654A (es) * | 1999-09-13 | 2002-07-30 | Wyeth Corp | Glucopiranosidos conjugados de 2-(4-hidroxi -fenil)-1- [4-(2-amin- 1-il-etoxi) -bencil] -1h -indol -5- oles. |
| US6380166B1 (en) | 1999-09-13 | 2002-04-30 | American Home Products Corporation | Glucopyranosides conjugates of 2-(4-hydroxy-phenyl)-3-methyl-1-[4-(2-amin-1-yl-ethoxy)-benzyl]-1H-indol-5-ols |
| WO2001027129A1 (en) * | 1999-10-08 | 2001-04-19 | Strakan Limited | Glycosides and orthoester glycosides of raloxifene and analogues and the use thereof |
| AU7674000A (en) * | 1999-10-08 | 2001-04-23 | Strakan Group Plc | Tamoxifen and tamoxifen analogue glycosides and uses thereof |
| WO2011029088A2 (en) * | 2009-09-07 | 2011-03-10 | Dr. Reddy's Laboratories Ltd. | Preparation of raloxifene and its salts |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4133814A (en) | 1975-10-28 | 1979-01-09 | Eli Lilly And Company | 2-Phenyl-3-aroylbenzothiophenes useful as antifertility agents |
| US4418068A (en) | 1981-04-03 | 1983-11-29 | Eli Lilly And Company | Antiestrogenic and antiandrugenic benzothiophenes |
| TW366342B (en) * | 1992-07-28 | 1999-08-11 | Lilly Co Eli | The use of 2-phenyl-3-aroylbenzothiophenes in inhibiting bone loss |
-
1995
- 1995-03-15 US US08/405,555 patent/US6723739B1/en not_active Expired - Fee Related
- 1995-03-15 US US08/404,701 patent/US5567820A/en not_active Expired - Fee Related
- 1995-05-16 SI SI9530336T patent/SI0683170T1/xx unknown
- 1995-05-16 DE DE69512310T patent/DE69512310T2/de not_active Expired - Fee Related
- 1995-05-16 RU RU95107655/04A patent/RU95107655A/ru unknown
- 1995-05-16 NZ NZ272131A patent/NZ272131A/en unknown
- 1995-05-16 ES ES95303265T patent/ES2136799T3/es not_active Expired - Lifetime
- 1995-05-16 AT AT95303265T patent/ATE184880T1/de not_active IP Right Cessation
- 1995-05-16 CZ CZ951262A patent/CZ126295A3/cs unknown
- 1995-05-16 DK DK95303265T patent/DK0683170T3/da active
- 1995-05-16 CA CA002149501A patent/CA2149501A1/en not_active Abandoned
- 1995-05-16 PE PE1995268768A patent/PE23396A1/es not_active Application Discontinuation
- 1995-05-16 EP EP95303265A patent/EP0683170B1/en not_active Expired - Lifetime
- 1995-05-16 TW TW084104846A patent/TW323285B/zh active
- 1995-05-16 ZA ZA953975A patent/ZA953975B/xx unknown
- 1995-05-17 AU AU20121/95A patent/AU683734B2/en not_active Ceased
- 1995-05-17 JP JP7118338A patent/JPH07316180A/ja not_active Withdrawn
- 1995-05-17 KR KR1019950012173A patent/KR950032183A/ko not_active Application Discontinuation
- 1995-05-17 PL PL95308635A patent/PL308635A1/xx unknown
- 1995-05-18 NO NO951322A patent/NO304694B1/no not_active IP Right Cessation
- 1995-05-18 YU YU31995A patent/YU31995A/sh unknown
- 1995-05-18 IL IL11378095A patent/IL113780A/xx active IP Right Grant
- 1995-05-18 BR BR9502079A patent/BR9502079A/pt not_active Application Discontinuation
- 1995-05-18 FI FI952420A patent/FI952420A/fi unknown
- 1995-05-18 HU HU9501466A patent/HU219335B/hu not_active IP Right Cessation
- 1995-05-18 CO CO95021224A patent/CO4650137A1/es unknown
- 1995-05-18 CN CN95106322A patent/CN1039013C/zh not_active Expired - Fee Related
-
1999
- 1999-12-15 GR GR990403228T patent/GR3032142T3/el unknown
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