SE7803195L - Forfarande for framstellning av 1,2,4-triazinderivat med farmakologisk verkan - Google Patents

Forfarande for framstellning av 1,2,4-triazinderivat med farmakologisk verkan

Info

Publication number
SE7803195L
SE7803195L SE7803195A SE7803195A SE7803195L SE 7803195 L SE7803195 L SE 7803195L SE 7803195 A SE7803195 A SE 7803195A SE 7803195 A SE7803195 A SE 7803195A SE 7803195 L SE7803195 L SE 7803195L
Authority
SE
Sweden
Prior art keywords
procedure
preparation
pharmacological effect
triazine derivatives
triazine
Prior art date
Application number
SE7803195A
Other languages
English (en)
Inventor
Delmar
Original Assignee
Allen & Hanburys Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB12598/77A external-priority patent/GB1584461A/en
Application filed by Allen & Hanburys Ltd filed Critical Allen & Hanburys Ltd
Publication of SE7803195L publication Critical patent/SE7803195L/sv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D253/00Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00
    • C07D253/02Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00 not condensed with other rings
    • C07D253/061,2,4-Triazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D253/00Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00
    • C07D253/02Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00 not condensed with other rings
    • C07D253/061,2,4-Triazines
    • C07D253/0651,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members
    • C07D253/071,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members with hetero atoms, or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pulmonology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SE7803195A 1977-03-25 1978-03-20 Forfarande for framstellning av 1,2,4-triazinderivat med farmakologisk verkan SE7803195L (sv)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB12598/77A GB1584461A (en) 1977-03-25 1977-03-25 Imidazotriazines imidazotriazinones and pharmaceutical compositions containing them
GB4725077 1977-11-14

Publications (1)

Publication Number Publication Date
SE7803195L true SE7803195L (sv) 1978-09-26

Family

ID=26249130

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7803195A SE7803195L (sv) 1977-03-25 1978-03-20 Forfarande for framstellning av 1,2,4-triazinderivat med farmakologisk verkan

Country Status (14)

Country Link
US (1) US4278673A (sv)
JP (1) JPS53119891A (sv)
AT (1) AT363952B (sv)
AU (1) AU516179B2 (sv)
DE (1) DE2811780A1 (sv)
DK (1) DK109578A (sv)
ES (1) ES468119A1 (sv)
FI (1) FI780828A (sv)
FR (1) FR2384773A1 (sv)
IE (1) IE46653B1 (sv)
IT (1) IT1105177B (sv)
NL (1) NL7803195A (sv)
NZ (1) NZ186699A (sv)
SE (1) SE7803195L (sv)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5496927A (en) * 1985-02-04 1996-03-05 Merrell Pharmaceuticals Inc. Peptidase inhibitors
US4687776A (en) * 1986-10-24 1987-08-18 Warner-Lambert Company Drug stabilization
US4788064A (en) * 1987-07-31 1988-11-29 Warner-Lambert Company Transdermal delivery system
US5208226A (en) * 1989-09-08 1993-05-04 Glaxo Group Limited Medicaments
US5270305A (en) * 1989-09-08 1993-12-14 Glaxo Group Limited Medicaments
HU230154B1 (hu) * 1997-11-12 2015-09-28 Bayer Intellectual Property Gmbh Eljárás 2-es helyzetben fenil-szubszituenst hordozó imidazo-triazinon-származékok előállítására
DE19827640A1 (de) 1998-06-20 1999-12-23 Bayer Ag 7-Alkyl- und Cycloalkyl-substituierte Imidazotriazinone
DE10063106A1 (de) * 2000-12-18 2002-06-20 Bayer Ag Verfahren zur Herstellung von 2-(2-Ethoxyphenyl)-substituierten Imidazotriazinonen
DE10064105A1 (de) 2000-12-21 2002-06-27 Bayer Ag Neue Substituierte Imidazotriazinone
JP4540295B2 (ja) * 2001-05-09 2010-09-08 バイエル・シェーリング・ファルマ・アクチェンゲゼルシャフト 2−フェニル置換イミダゾトリアジノンの新しい用途
GB0113343D0 (en) * 2001-06-01 2001-07-25 Bayer Ag Novel Heterocycles 2
US7087605B2 (en) * 2001-06-01 2006-08-08 Bayer Aktiengesellschaft 5-Ethyl-imidazotriazinones
GB0113344D0 (en) 2001-06-01 2001-07-25 Bayer Ag Novel heterocycles 3
DE10130167A1 (de) 2001-06-22 2003-01-02 Bayer Ag Imidazotriazine
DE10135815A1 (de) 2001-07-23 2003-02-06 Bayer Ag Verwendung von 2-Alkoxyphenyl-substituierten Imidazotriazinonen
GB0209988D0 (en) * 2002-05-01 2002-06-12 Bayer Ag Novel Heterocycles
GB2388111A (en) * 2002-05-01 2003-11-05 Bayer Ag Novel imidazotriazinone compounds
GB2388594A (en) * 2002-05-16 2003-11-19 Bayer Ag Imidazo-triazine PDE 4 inhibitors
DE10232113A1 (de) 2002-07-16 2004-01-29 Bayer Ag Vardenafil Hydrochlorid Trihydrat enthaltende Arzneimittel
WO2004087652A2 (en) * 2003-04-01 2004-10-14 Smithkline Beecham Corporation Imidazotriazine compounds
JP2008501617A (ja) * 2004-06-11 2008-01-24 アスビオファーマ株式会社 Pde7阻害作用を有するイミダゾトリアジノン誘導体
JP2008516071A (ja) * 2004-10-13 2008-05-15 クナーフ インシュレーション ゲーエムベーハー ポリエステル結合性組成物
DE102005001989A1 (de) * 2005-01-15 2006-07-20 Bayer Healthcare Ag Intravenöse Formulierungen von PDE-Inhibitoren
DE102005009240A1 (de) * 2005-03-01 2006-09-07 Bayer Healthcare Ag Arzneiformen mit verbesserten pharmakokinetischen Eigenschaften
DE102005009241A1 (de) * 2005-03-01 2006-09-07 Bayer Healthcare Ag Arzneiformen mit kontrollierter Bioverfügbarkeit
SG166106A1 (en) * 2005-09-29 2010-11-29 Bayer Schering Pharma Ag Pde inhibitors and combinations thereof for the treatment of urological disorders
DE102006048693A1 (de) * 2006-10-14 2008-04-17 Bayer Healthcare Ag Inhibition der PDE2A
WO2008151734A1 (en) * 2007-06-13 2008-12-18 Bayer Schering Pharma Aktiengesellschaft Pde inhibitors for the treatment of hearing impairment

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE791025A (fr) * 1971-11-19 1973-05-07 Allen & Hanburys Ltd Composes heterocycliques
GB1457873A (en) * 1973-01-04 1976-12-08 Allen & Hanburys Ltd Imidazotriazines

Also Published As

Publication number Publication date
IE780625L (en) 1978-09-25
FR2384773B1 (sv) 1980-07-04
AU516179B2 (en) 1981-05-21
FI780828A (fi) 1978-09-26
NZ186699A (en) 1980-12-19
AU3431478A (en) 1979-09-27
NL7803195A (nl) 1978-09-27
IE46653B1 (en) 1983-08-10
IT1105177B (it) 1985-10-28
US4278673A (en) 1981-07-14
FR2384773A1 (fr) 1978-10-20
ATA196378A (de) 1981-02-15
JPS53119891A (en) 1978-10-19
DE2811780A1 (de) 1978-09-28
ES468119A1 (es) 1979-09-01
IT7848546A0 (it) 1978-03-22
DK109578A (da) 1978-09-26
AT363952B (de) 1981-09-10

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