SE416645B - Forfarande for framstellning av 6-deoxitetracykliner genom katalytisk hydrogenering av eventuellt 11a-halogenerade 6-demetyl-6-deoxi-6-metylentetracykliner - Google Patents

Forfarande for framstellning av 6-deoxitetracykliner genom katalytisk hydrogenering av eventuellt 11a-halogenerade 6-demetyl-6-deoxi-6-metylentetracykliner

Info

Publication number: SE416645B
Authority: SE; Sweden
Prior art keywords: metylentetracyclines; halogenered; deoxi; deoxytetracyclines; demethyl
Prior art date: 1973-04-20

Application number

SE7403949A

Other languages

English (en)

Inventor

Jr T A Morris

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1973-04-20

Filing date

1974-03-22

Publication date

1981-01-26

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26997777&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SE416645(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1974-03-22 Application filed by Pfizer filed Critical Pfizer

1981-01-26 Publication of SE416645B publication Critical patent/SE416645B/sv

Links

230000003197 catalytic effect Effects 0.000 title 1
238000000034 method Methods 0.000 title 1
238000002360 preparation method Methods 0.000 title 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/65—Tetracyclines
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C231/00—Preparation of carboxylic acid amides
- C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
- C07C237/24—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring of the carbon skeleton
- C07C237/26—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring of the carbon skeleton of a ring being part of a condensed ring system formed by at least four rings, e.g. tetracycline
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2603/00—Systems containing at least three condensed rings
- C07C2603/02—Ortho- or ortho- and peri-condensed systems
- C07C2603/40—Ortho- or ortho- and peri-condensed systems containing four condensed rings
- C07C2603/42—Ortho- or ortho- and peri-condensed systems containing four condensed rings containing only six-membered rings
- C07C2603/44—Naphthacenes; Hydrogenated naphthacenes
- C07C2603/46—1,4,4a,5,5a,6,11,12a- Octahydronaphthacenes, e.g. tetracyclines

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Epidemiology (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Catalysts (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Plural Heterocyclic Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

SE7403949A 1973-04-20 1974-03-22 Forfarande for framstellning av 6-deoxitetracykliner genom katalytisk hydrogenering av eventuellt 11a-halogenerade 6-demetyl-6-deoxi-6-metylentetracykliner SE416645B (sv)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US35308473A	1973-04-20	1973-04-20
US05/421,206 US3954862A (en)	1973-04-20	1973-12-03	Process for producing α-6-deoxytetracyclines

Publications (1)

Publication Number	Publication Date
SE416645B true SE416645B (sv)	1981-01-26

Family

ID=26997777

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SE7403949A SE416645B (sv)	1973-04-20	1974-03-22	Forfarande for framstellning av 6-deoxitetracykliner genom katalytisk hydrogenering av eventuellt 11a-halogenerade 6-demetyl-6-deoxi-6-metylentetracykliner

Country Status (30)

Country	Link
US (1)	US3954862A (sv)
JP (1)	JPS5710863B2 (sv)
AR (1)	AR200521A1 (sv)
AT (1)	AT333954B (sv)
AU (1)	AU461511B2 (sv)
BG (1)	BG25070A3 (sv)
CA (1)	CA1011736A (sv)
CH (1)	CH589044A5 (sv)
CS (2)	CS235053B2 (sv)
DD (1)	DD114404A5 (sv)
DE (1)	DE2418499C2 (sv)
DK (1)	DK155662C (sv)
EG (1)	EG11172A (sv)
ES (1)	ES425221A1 (sv)
FI (1)	FI60196C (sv)
FR (1)	FR2226389B1 (sv)
GB (1)	GB1458744A (sv)
HK (1)	HK28279A (sv)
IE (1)	IE40048B1 (sv)
IL (1)	IL44492A (sv)
IN (1)	IN138740B (sv)
KE (1)	KE2937A (sv)
LU (1)	LU69856A1 (sv)
MY (1)	MY7900242A (sv)
NL (1)	NL157893B (sv)
NO (1)	NO146596C (sv)
PH (1)	PH10555A (sv)
RO (2)	RO80170A (sv)
SE (1)	SE416645B (sv)
YU (1)	YU39303B (sv)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4743699A (en) *	1982-01-19	1988-05-10	Plurichemie Anstalt	Homogeneous catalytic system and a process for the preparation of same
US4500458A (en) *	1982-01-19	1985-02-19	Plurichemie Anstalt	Process for the preparation of α-6-deoxytetracyclines
USRE32535E (en) *	1982-01-19	1987-10-27	Plurichemie Anstalt	Process for the preparation of α-6-deoxytetracyclines
DK386784A (da) *	1983-08-17	1985-02-18	Hovione Int Ltd	Fremgangsmaade til fremstilling af alfa-6-desoxy-tetracykliner
JPS6343554U (sv) *	1986-09-05	1988-03-23
US4987242A (en) *	1988-10-28	1991-01-22	Jagmohan Khanna	Hydrogenation catalyst useful in the production of alpha-6-deoxytetracyclines
US4973719A (en) *	1988-10-28	1990-11-27	Ranbaxy Laboratories Limited	Process for the production of alpha-6-deoxytetracyclines
EP0452412A4 (en) *	1989-01-04	1992-06-03	Houba, Inc.	Process for the production of alpha-6-deoxytetracyclines
US5049683A (en) *	1989-01-04	1991-09-17	Houba, Inc.	Process for the production of alpha-6-deoxytetracyclines
DE68900339D1 (de) *	1989-04-03	1991-11-21	Ranbaxy Lab Ltd	Verfahren zur herstellung von alpha-6-deoxytetracyclinen.
DE102007003434A1 (de)	2007-01-23	2008-07-24	Jäger, Anton	Reinigungsvorrichtung
CN105152961B (zh) *	2015-08-31	2017-07-11	河南师范大学	一种强力霉素中间体6‑次甲基土霉素的合成方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR1430859A (sv) *	1960-05-23	1966-05-25
CH579531A5 (sv) *	1972-02-24	1976-09-15	Ankerfarm Spa

1973
- 1973-12-03 US US05/421,206 patent/US3954862A/en not_active Expired - Lifetime
1974
- 1974-03-22 CA CA195,764A patent/CA1011736A/en not_active Expired
- 1974-03-22 SE SE7403949A patent/SE416645B/sv not_active IP Right Cessation
- 1974-03-25 IL IL44492A patent/IL44492A/en unknown
- 1974-03-25 IN IN645/CAL/74A patent/IN138740B/en unknown
- 1974-03-26 AU AU67143/74A patent/AU461511B2/en not_active Expired
- 1974-03-26 GB GB1347974A patent/GB1458744A/en not_active Expired
- 1974-03-27 IE IE668/74A patent/IE40048B1/xx unknown
- 1974-03-28 PH PH15670A patent/PH10555A/en unknown
- 1974-04-01 YU YU895/74A patent/YU39303B/xx unknown
- 1974-04-03 NO NO741223A patent/NO146596C/no unknown
- 1974-04-05 NL NL7404666.A patent/NL157893B/xx not_active IP Right Cessation
- 1974-04-05 FI FI1045/74A patent/FI60196C/fi active
- 1974-04-08 EG EG105/74A patent/EG11172A/xx active
- 1974-04-08 DK DK193874A patent/DK155662C/da not_active IP Right Cessation
- 1974-04-08 JP JP3894774A patent/JPS5710863B2/ja not_active Expired
- 1974-04-08 AT AT292274A patent/AT333954B/de not_active IP Right Cessation
- 1974-04-10 ES ES425221A patent/ES425221A1/es not_active Expired
- 1974-04-10 AR AR253236A patent/AR200521A1/es active
- 1974-04-11 CH CH510574A patent/CH589044A5/xx not_active IP Right Cessation
- 1974-04-11 DE DE2418499A patent/DE2418499C2/de not_active Expired
- 1974-04-12 LU LU69856A patent/LU69856A1/xx unknown
- 1974-04-12 FR FR7413094A patent/FR2226389B1/fr not_active Expired
- 1974-04-18 DD DD177985A patent/DD114404A5/xx unknown
- 1974-04-19 RO RO74102560A patent/RO80170A/ro unknown
- 1974-04-19 BG BG7400026460A patent/BG25070A3/xx unknown
- 1974-04-19 CS CS742822A patent/CS235053B2/cs unknown
- 1974-04-19 RO RO7478493A patent/RO78908A/ro unknown
- 1974-04-19 CS CS741920A patent/CS235092B2/cs unknown
1979
- 1979-03-16 KE KE2937A patent/KE2937A/xx unknown
- 1979-05-03 HK HK282/79A patent/HK28279A/xx unknown
- 1979-12-30 MY MY242/79A patent/MY7900242A/xx unknown

Also Published As

Publication number	Publication date
AU6714374A (en)	1975-05-29
GB1458744A (en)	1976-12-15
HK28279A (en)	1979-05-11
NO146596C (no)	1982-11-03
KE2937A (en)	1979-03-30
IE40048B1 (en)	1979-02-28
RO78908A (ro)	1982-08-17
MY7900242A (en)	1979-12-31
ATA292274A (de)	1976-04-15
FI60196B (fi)	1981-08-31
FR2226389A1 (sv)	1974-11-15
CH589044A5 (sv)	1977-06-30
RO80170A (ro)	1982-10-26
IN138740B (sv)	1976-03-27
DD114404A5 (sv)	1975-08-05
IL44492A0 (en)	1974-06-30
DE2418499A1 (de)	1974-11-07
CS235053B2 (en)	1985-04-16
NO146596B (no)	1982-07-26
FR2226389B1 (sv)	1976-12-17
YU39303B (en)	1984-10-31
DK155662C (da)	1989-10-09
AR200521A1 (es)	1974-11-15
IE40048L (en)	1975-06-03
DE2418499C2 (de)	1982-12-23
NL157893B (nl)	1978-09-15
PH10555A (en)	1977-06-08
YU85974A (en)	1982-05-31
CS235092B2 (en)	1985-04-16
IL44492A (en)	1977-01-31
EG11172A (en)	1977-01-31
FI60196C (fi)	1981-12-10
AT333954B (de)	1976-12-27
DK155662B (da)	1989-05-01
BG25070A3 (en)	1978-07-12
NO741223L (no)	1974-10-22
ES425221A1 (es)	1976-05-16
LU69856A1 (sv)	1974-11-21
CA1011736A (en)	1977-06-07
JPS5710863B2 (sv)	1982-03-01
AU461511B2 (en)	1975-05-29
JPS49135961A (sv)	1974-12-27
NL7404666A (sv)	1974-10-22
US3954862A (en)	1976-05-04

Legal Events

Date

Code

Title

Description

1995-01-31

NUG

Patent has lapsed

Ref document number: 7403949-6

Effective date: 19940410

Format of ref document f/p: F

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SE7710599L (sv)	1977-09-21	Forfarande for framstellning av bensisoxazoler
SE411212B (sv)	1979-12-10	Forfarande for framstellning av 3-halogen-cefalosporiner
SE416645B (sv)	1981-01-26	Forfarande for framstellning av 6-deoxitetracykliner genom katalytisk hydrogenering av eventuellt 11a-halogenerade 6-demetyl-6-deoxi-6-metylentetracykliner
RO70474A (ro)	1982-04-12	PROCEDEU PENTRU PREPARAREA PARAXILENULёI
NO143531C (no)	1981-03-11	Fremgangsmaate for fremstilling av acylerte benzoksazolinon-derivater.
NO790627L (no)	1975-01-14	Fremgangsmaate for fremstilling av hydroksyalkylxantiner
SE417601B (sv)	1981-03-30	Forfarande for framstellning av amidinokarbamider
NO153806C (no)	1986-05-28	Fremgangsmaate for fremstilling av 6-deoksytetracyklin.
SE387341B (sv)	1976-09-06	Forfarande for framstellning av 1-aryl-n-dialkyl-aminoalkyl-3,4-dihydro2(h)-isokinolinkarboxamider
TR17584A (tr)	1975-07-23	Herbisid triazinlerinin hazirlanmasina mahsus usul
SE421129B (sv)	1981-11-30	Forfarande for framstellning av poly-n-alkyl-iminoalaner
SE409994B (sv)	1979-09-17	Forfarande for framstellning av amidinokarbamider
SE411211B (sv)	1979-12-10	Forfarande for framstellning av 3-halogencefalosporiner
RO69264A (ro)	1982-04-12	Procedeu pentru prepararea alfa-amino-alcoolilor
SE401835B (sv)	1978-05-29	Forfarande for framstellning av 17beta-hydroxi-16,16-dimetylest-4-en-3-on
SE407219B (sv)	1979-03-19	Forfarande for framstellning av metyl-3-(2--kinoxalinylmetylen)-karbazat-n1,n4-dioxid
NO139479C (no)	1979-03-21	Fremgangsmaate for fremstilling av 4-amino-3,5-dihalogen-fenyl-etanolaminer
SE406086B (sv)	1979-01-22	Forfarande for framstellning av cyklisk-dikarboximido-substituerade fosfonotioater
NO146597C (no)	1982-11-03	Fremgangsmaate for fremstilling av 6-metylentetracykliner
SE386144B (sv)	1976-08-02	Forfarande for framstellning av en alkaliamid.
RO70980A (ro)	1981-08-17	Procedeu pentru prepararea oxamidei