RU2016146350A - Ингалятор ароматизированного никотинового порошка - Google Patents

Ингалятор ароматизированного никотинового порошка Download PDF

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RU2016146350A
RU2016146350A RU2016146350A RU2016146350A RU2016146350A RU 2016146350 A RU2016146350 A RU 2016146350A RU 2016146350 A RU2016146350 A RU 2016146350A RU 2016146350 A RU2016146350 A RU 2016146350A RU 2016146350 A RU2016146350 A RU 2016146350A
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Prior art keywords
nicotine powder
nicotine
inhaler according
powder inhaler
flavor
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RU2016146350A
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English (en)
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RU2016146350A3 (ru
RU2680422C2 (ru
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Ихар Николаевич ЗИНОВИК
Жерар Зюбер
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Филип Моррис Продактс С.А.
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    • AHUMAN NECESSITIES
    • A24TOBACCO; CIGARS; CIGARETTES; SIMULATED SMOKING DEVICES; SMOKERS' REQUISITES
    • A24FSMOKERS' REQUISITES; MATCH BOXES; SIMULATED SMOKING DEVICES
    • A24F42/00Simulated smoking devices other than electrically operated; Component parts thereof; Manufacture or testing thereof
    • A24F42/60Constructional details
    • AHUMAN NECESSITIES
    • A24TOBACCO; CIGARS; CIGARETTES; SIMULATED SMOKING DEVICES; SMOKERS' REQUISITES
    • A24FSMOKERS' REQUISITES; MATCH BOXES; SIMULATED SMOKING DEVICES
    • A24F47/00Smokers' requisites not otherwise provided for
    • AHUMAN NECESSITIES
    • A24TOBACCO; CIGARS; CIGARETTES; SIMULATED SMOKING DEVICES; SMOKERS' REQUISITES
    • A24BMANUFACTURE OR PREPARATION OF TOBACCO FOR SMOKING OR CHEWING; TOBACCO; SNUFF
    • A24B15/00Chemical features or treatment of tobacco; Tobacco substitutes, e.g. in liquid form
    • A24B15/10Chemical features of tobacco products or tobacco substitutes
    • A24B15/16Chemical features of tobacco products or tobacco substitutes of tobacco substitutes
    • AHUMAN NECESSITIES
    • A24TOBACCO; CIGARS; CIGARETTES; SIMULATED SMOKING DEVICES; SMOKERS' REQUISITES
    • A24FSMOKERS' REQUISITES; MATCH BOXES; SIMULATED SMOKING DEVICES
    • A24F40/00Electrically operated smoking devices; Component parts thereof; Manufacture thereof; Maintenance or testing thereof; Charging means specially adapted therefor
    • A24F40/20Devices using solid inhalable precursors
    • AHUMAN NECESSITIES
    • A24TOBACCO; CIGARS; CIGARETTES; SIMULATED SMOKING DEVICES; SMOKERS' REQUISITES
    • A24FSMOKERS' REQUISITES; MATCH BOXES; SIMULATED SMOKING DEVICES
    • A24F40/00Electrically operated smoking devices; Component parts thereof; Manufacture thereof; Maintenance or testing thereof; Charging means specially adapted therefor
    • A24F40/60Devices with integrated user interfaces
    • AHUMAN NECESSITIES
    • A24TOBACCO; CIGARS; CIGARETTES; SIMULATED SMOKING DEVICES; SMOKERS' REQUISITES
    • A24FSMOKERS' REQUISITES; MATCH BOXES; SIMULATED SMOKING DEVICES
    • A24F42/00Simulated smoking devices other than electrically operated; Component parts thereof; Manufacture or testing thereof
    • A24F42/20Devices without heating means
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/465Nicotine; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/007Pulmonary tract; Aromatherapy
    • A61K9/0073Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0075Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61MDEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY; DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROM THE BODY; DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR
    • A61M15/00Inhalators
    • A61M15/0001Details of inhalators; Constructional features thereof
    • A61M15/0021Mouthpieces therefor
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61MDEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY; DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROM THE BODY; DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR
    • A61M15/00Inhalators
    • A61M15/0028Inhalators using prepacked dosages, one for each application, e.g. capsules to be perforated or broken-up
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61MDEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY; DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROM THE BODY; DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR
    • A61M15/00Inhalators
    • A61M15/0028Inhalators using prepacked dosages, one for each application, e.g. capsules to be perforated or broken-up
    • A61M15/003Inhalators using prepacked dosages, one for each application, e.g. capsules to be perforated or broken-up using capsules, e.g. to be perforated or broken-up
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61MDEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY; DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROM THE BODY; DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR
    • A61M15/00Inhalators
    • A61M15/0028Inhalators using prepacked dosages, one for each application, e.g. capsules to be perforated or broken-up
    • A61M15/003Inhalators using prepacked dosages, one for each application, e.g. capsules to be perforated or broken-up using capsules, e.g. to be perforated or broken-up
    • A61M15/0033Details of the piercing or cutting means
    • A61M15/0035Piercing means
    • A61M15/0036Piercing means hollow piercing means
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61MDEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY; DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROM THE BODY; DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR
    • A61M15/00Inhalators
    • A61M15/06Inhaling appliances shaped like cigars, cigarettes or pipes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61MDEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY; DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROM THE BODY; DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR
    • A61M2202/00Special media to be introduced, removed or treated
    • A61M2202/06Solids
    • A61M2202/064Powder
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61MDEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY; DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROM THE BODY; DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR
    • A61M2206/00Characteristics of a physical parameter; associated device therefor
    • A61M2206/10Flow characteristics
    • A61M2206/16Rotating swirling helical flow, e.g. by tangential inflows

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  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pulmonology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Biomedical Technology (AREA)
  • Anesthesiology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Otolaryngology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Human Computer Interaction (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Cigarettes, Filters, And Manufacturing Of Filters (AREA)

Claims (20)

1. Ингалятор никотинового порошка, содержащий
корпус, проходящий между мундштучным участком и дальним концевым участком;
канал воздушного потока, проходящий между мундштучным участком и дальним концевым участком;
емкость для никотинового порошка, расположенную вдоль канала воздушного потока и содержащую дозу никотинового порошка, содержащего никотиновую соль, и;
элемент доставки аромата, соединенный по текучей среде с каналом воздушного потока;
при этом доза никотинового порошка может вдыхаться в легкие пользователя с производительностью ингаляции, составляющей менее чем примерно 5 л/мин.
2. Ингалятор никотинового порошка по п. 1, в котором элемент доставки аромата расположен раньше по ходу потока относительно емкости для никотинового порошка.
3. Ингалятор никотинового порошка по п. 1, в котором элемент доставки аромата расположен дальше по ходу потока относительно емкости для никотинового порошка.
4. Ингалятор никотинового порошка по п. 1, дополнительно содержащий второй канал воздушного потока, содержащий емкость для ароматизатора, образующую параллельную схему по потоку с емкостью для никотинового порошка.
5. Ингалятор никотинового порошка по любому из пп. 1-4, в котором элемент доставки аромата содержит порошковый ароматизатор.
6. Ингалятор никотинового порошка по любому из пп. 1-4, в котором элемент аромата содержит жидкий ароматизатор.
7. Ингалятор никотинового порошка по любому из пп. 1-4, в котором емкость для никотинового порошка выполнена с возможностью размещения в ней капсулы, содержащей никотиновый порошок, содержащий никотиновую соль.
8. Ингалятор никотинового порошка по п. 7, в котором капсула дополнительно содержит элемент доставки аромата, содержащий порошковый ароматизатор.
9. Ингалятор никотинового порошка по любому из пп. 1-4, 8, в котором элемент доставки аромата содержит разрушаемую капсулу, которая может быть разрушена пользователем для высвобождения ароматизатора.
10. Ингалятор никотинового порошка по любому из пп. 1-4, 8, дополнительно содержащий фильтрующий элемент, расположенный раньше по ходу потока относительно емкости для никотинового порошка, причем элемент доставки аромата расположен внутри фильтрующего элемента.
11. Ингалятор никотинового порошка по п. 10, в котором элемент доставки аромата представляет собой нить, пропитанную ментолом.
12. Ингалятор никотинового порошка по любому из пп. 1-4, 8, 11, дополнительно содержащий дозу второго активного агента.
13. Ингалятор никотинового порошка по любому из пп. 1-4, 8, 11, дополнительно содержащий вихреобразующий элемент, выполненный с возможностью создания вращательного движения в воздушном потоке из канала воздушного потока.
14. Способ ингаляции ароматизированного никотина в легкие пользователя, согласно которому:
вдыхают воздух через ингалятор ароматизированного никотинового порошка по любому из пп. 1-13 с расходом, составляющим менее чем примерно 2 л/мин, для доставки ароматизированного порошкового никотина в легкие пользователя.
RU2016146350A 2014-04-28 2015-04-23 Ингалятор ароматизированного никотинового порошка RU2680422C2 (ru)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201461984968P 2014-04-28 2014-04-28
EP14166210.6 2014-04-28
EP14166210 2014-04-28
US61/984,968 2014-04-28
PCT/IB2015/001283 WO2015166350A2 (en) 2014-04-28 2015-04-23 Flavoured nicotine powder inhaler

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RU2016146350A true RU2016146350A (ru) 2018-05-28
RU2016146350A3 RU2016146350A3 (ru) 2018-08-27
RU2680422C2 RU2680422C2 (ru) 2019-02-21

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US (2) US10912334B2 (ru)
EP (1) EP3136895B1 (ru)
JP (1) JP6712232B2 (ru)
KR (1) KR102428028B1 (ru)
CN (1) CN106170313B (ru)
AU (1) AU2015254999B2 (ru)
CA (1) CA2943746C (ru)
MX (1) MX2016014090A (ru)
PH (1) PH12016501719B1 (ru)
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SG (1) SG11201608985QA (ru)
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CA2943746A1 (en) 2015-11-05
WO2015166350A2 (en) 2015-11-05
TW201544021A (zh) 2015-12-01
PH12016501719A1 (en) 2016-10-24
MX2016014090A (es) 2017-02-09
CA2943746C (en) 2023-08-15
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SG11201608985QA (en) 2016-11-29
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AU2015254999B2 (en) 2019-08-01
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US10912334B2 (en) 2021-02-09
US20170035108A1 (en) 2017-02-09
CN106170313A (zh) 2016-11-30
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US20210153545A1 (en) 2021-05-27

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