PT934321E - Tienopirimidinas com accao inibidora da fosfodiesterase v - Google Patents

Tienopirimidinas com accao inibidora da fosfodiesterase v

Info

Publication number
PT934321E
PT934321E PT97912139T PT97912139T PT934321E PT 934321 E PT934321 E PT 934321E PT 97912139 T PT97912139 T PT 97912139T PT 97912139 T PT97912139 T PT 97912139T PT 934321 E PT934321 E PT 934321E
Authority
PT
Portugal
Prior art keywords
tienopyrimidines
phosphodiesterase
inhibitor action
inhibitor
action
Prior art date
Application number
PT97912139T
Other languages
English (en)
Inventor
Schelling Dr Pierre
Rochus Jonas
Franz-Werner Kluxen
Maria Christadler
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of PT934321E publication Critical patent/PT934321E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Gynecology & Obstetrics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT97912139T 1996-10-24 1997-10-08 Tienopirimidinas com accao inibidora da fosfodiesterase v PT934321E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19644228A DE19644228A1 (de) 1996-10-24 1996-10-24 Thienopyrimidine

Publications (1)

Publication Number Publication Date
PT934321E true PT934321E (pt) 2003-12-31

Family

ID=7809880

Family Applications (1)

Application Number Title Priority Date Filing Date
PT97912139T PT934321E (pt) 1996-10-24 1997-10-08 Tienopirimidinas com accao inibidora da fosfodiesterase v

Country Status (24)

Country Link
US (1) US6130223A (pt)
EP (1) EP0934321B1 (pt)
JP (1) JP2001502342A (pt)
KR (1) KR100488429B1 (pt)
CN (1) CN1105116C (pt)
AR (1) AR008504A1 (pt)
AT (1) ATE246689T1 (pt)
AU (1) AU726639B2 (pt)
BR (1) BR9712652A (pt)
CA (1) CA2269815C (pt)
CZ (1) CZ294027B6 (pt)
DE (2) DE19644228A1 (pt)
DK (1) DK0934321T3 (pt)
ES (1) ES2201275T3 (pt)
HK (1) HK1024484A1 (pt)
HU (1) HUP9904680A3 (pt)
NO (1) NO991951L (pt)
PL (1) PL192163B1 (pt)
PT (1) PT934321E (pt)
RU (1) RU2197492C2 (pt)
SK (1) SK284979B6 (pt)
TW (1) TW457242B (pt)
WO (1) WO1998017668A1 (pt)
ZA (1) ZA979516B (pt)

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CN106061504B (zh) 2014-01-21 2019-09-06 詹森药业有限公司 包括代谢型谷氨酸能受体亚型2的正别构调节物或正位激动剂的组合及其用途
KR20200126026A (ko) 2014-01-21 2020-11-05 얀센 파마슈티카 엔.브이. 대사 조절형 글루탐산 작동성 수용체 제2아형의 양성 알로스테릭 조절제 또는 오르토스테릭 작동제를 포함하는 조합 및 그 용도
CN106233141B (zh) 2014-02-18 2018-08-21 罗伯特·I·汉金 用于诊断和治疗味觉或嗅觉的损失和/或失真的方法和组合物
JP6687550B2 (ja) 2014-06-23 2020-04-22 セルジーン コーポレイション 肝疾患又は肝機能異常を治療するためのアプレミラスト
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Also Published As

Publication number Publication date
AR008504A1 (es) 2000-01-19
KR20000052772A (ko) 2000-08-25
JP2001502342A (ja) 2001-02-20
WO1998017668A1 (de) 1998-04-30
DE19644228A1 (de) 1998-04-30
ATE246689T1 (de) 2003-08-15
NO991951D0 (no) 1999-04-23
SK50299A3 (en) 2000-03-13
CA2269815A1 (en) 1998-04-30
AU726639B2 (en) 2000-11-16
TW457242B (en) 2001-10-01
PL332970A1 (en) 1999-10-25
RU2197492C2 (ru) 2003-01-27
EP0934321B1 (de) 2003-08-06
US6130223A (en) 2000-10-10
CA2269815C (en) 2007-09-25
HUP9904680A2 (hu) 2000-05-28
ZA979516B (en) 1998-05-12
CZ142299A3 (cs) 1999-07-14
DE59710547D1 (de) 2003-09-11
CZ294027B6 (cs) 2004-09-15
EP0934321A1 (de) 1999-08-11
KR100488429B1 (ko) 2005-05-10
CN1105116C (zh) 2003-04-09
NO991951L (no) 1999-06-17
PL192163B1 (pl) 2006-09-29
AU4945097A (en) 1998-05-15
HUP9904680A3 (en) 2001-11-28
CN1240450A (zh) 2000-01-05
BR9712652A (pt) 1999-10-26
DK0934321T3 (da) 2003-11-03
HK1024484A1 (en) 2000-10-13
SK284979B6 (sk) 2006-03-02
ES2201275T3 (es) 2004-03-16

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