PT915874E - Processo de preparacao de valaciclovir e intermediarios relevantes - Google Patents

Processo de preparacao de valaciclovir e intermediarios relevantes

Info

Publication number
PT915874E
PT915874E PT97937496T PT97937496T PT915874E PT 915874 E PT915874 E PT 915874E PT 97937496 T PT97937496 T PT 97937496T PT 97937496 T PT97937496 T PT 97937496T PT 915874 E PT915874 E PT 915874E
Authority
PT
Portugal
Prior art keywords
valaciclovir
intermediaries
relevant
preparation process
preparation
Prior art date
Application number
PT97937496T
Other languages
English (en)
Inventor
Silvio Pirovano
Maurizio Montoro
Original Assignee
Ind Chimica Srl
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ind Chimica Srl filed Critical Ind Chimica Srl
Publication of PT915874E publication Critical patent/PT915874E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/18Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one oxygen and one nitrogen atom, e.g. guanine

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Catalysts (AREA)
PT97937496T 1996-07-18 1997-07-17 Processo de preparacao de valaciclovir e intermediarios relevantes PT915874E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT96MI001491A IT1283447B1 (it) 1996-07-18 1996-07-18 Processo di preparazione del valaciclovir e relativi intermedi

Publications (1)

Publication Number Publication Date
PT915874E true PT915874E (pt) 2004-04-30

Family

ID=11374611

Family Applications (1)

Application Number Title Priority Date Filing Date
PT97937496T PT915874E (pt) 1996-07-18 1997-07-17 Processo de preparacao de valaciclovir e intermediarios relevantes

Country Status (8)

Country Link
EP (1) EP0915874B1 (pt)
AU (1) AU4010797A (pt)
BG (1) BG63721B1 (pt)
CA (1) CA2261050A1 (pt)
ES (1) ES2212122T3 (pt)
IT (1) IT1283447B1 (pt)
PT (1) PT915874E (pt)
WO (1) WO1998003553A1 (pt)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1436295A4 (en) * 2001-09-07 2007-07-11 Teva Pharma CRISTALLINE FORMS OF VALACYCLOVIR HYDROCHLORIDE
KR20050044449A (ko) * 2001-11-14 2005-05-12 테바 파마슈티컬 인더스트리즈 리미티드 발라시클로비르의 합성 및 정제 방법
US20050043329A1 (en) * 2002-09-06 2005-02-24 Shlomit Wizel Crystalline forms of valacyclovir hydrochloride
AU2003232719A1 (en) * 2003-05-30 2005-01-21 Eos Eczacibasi Ozgun Kimyasal Urunler Sanayi Ve Ticaret A.S. Novel crystalline forms of valacyclovir hydrochloride
EP2014660A3 (en) * 2003-06-02 2009-07-15 Teva Pharmaceutical Industries Ltd Novel crystalline forms of valacyclovir hydrochloride
KR20060117355A (ko) * 2004-01-21 2006-11-16 테바 파마슈티컬 인더스트리즈 리미티드 발라시클로버 염산염의 제조 방법
WO2006029253A2 (en) * 2004-09-04 2006-03-16 Teva Pharmaceutical Industries Ltd. A valacyclovir impurity, process for the preparation of valacyclovir impurity and use as a reference standard
US20060178512A1 (en) * 2005-02-04 2006-08-10 Cheruthur Govindan Method for preparing amino acid esters of nucleoside analogues
ES2291101B1 (es) * 2005-12-23 2009-02-16 Quimica Sintetica, S.A. Procedimiento para la preparacion de valaciclovir.
JP5152180B2 (ja) * 2007-04-27 2013-02-27 味の素株式会社 バラシクロビルの製造方法
CN101456859B (zh) * 2009-01-06 2011-07-20 华南理工大学 抗病毒药物缬昔洛韦的制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AP55A (en) * 1987-08-15 1989-09-26 The Wellcome Foundation Ltd Therapeutic Acyclic Nucleosides
ATE199719T1 (de) * 1993-06-10 2001-03-15 Rolabo Sl Verfahren zur herstellung von aminosäureester von nukleosid analogen
GB9501178D0 (en) * 1995-01-20 1995-03-08 Wellcome Found Guanine derivative

Also Published As

Publication number Publication date
ITMI961491A0 (pt) 1996-07-18
ES2212122T3 (es) 2004-07-16
BG103082A (en) 1999-09-30
IT1283447B1 (it) 1998-04-21
EP0915874B1 (en) 2003-12-10
ITMI961491A1 (it) 1998-01-18
WO1998003553A1 (en) 1998-01-29
AU4010797A (en) 1998-02-10
CA2261050A1 (en) 1998-01-29
BG63721B1 (bg) 2002-10-31
EP0915874A2 (en) 1999-05-19

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