PT912536E - Processo de monoacilacao de hidroxi-taxanos - Google Patents

Processo de monoacilacao de hidroxi-taxanos

Info

Publication number
PT912536E
PT912536E PT97931868T PT97931868T PT912536E PT 912536 E PT912536 E PT 912536E PT 97931868 T PT97931868 T PT 97931868T PT 97931868 T PT97931868 T PT 97931868T PT 912536 E PT912536 E PT 912536E
Authority
PT
Portugal
Prior art keywords
monoacylation
taxane
hydroxy
taxane monoacylation
monoacylation process
Prior art date
Application number
PT97931868T
Other languages
English (en)
Inventor
Eric Didier
Pascal Pecquet
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of PT912536E publication Critical patent/PT912536E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D305/00Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
PT97931868T 1996-07-09 1997-07-04 Processo de monoacilacao de hidroxi-taxanos PT912536E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9608505A FR2750989B1 (fr) 1996-07-09 1996-07-09 Procede de monoacylation d'hydroxy taxanes

Publications (1)

Publication Number Publication Date
PT912536E true PT912536E (pt) 2002-11-29

Family

ID=9493827

Family Applications (1)

Application Number Title Priority Date Filing Date
PT97931868T PT912536E (pt) 1996-07-09 1997-07-04 Processo de monoacilacao de hidroxi-taxanos

Country Status (20)

Country Link
US (1) US6127555A (pt)
EP (1) EP0912536B1 (pt)
JP (1) JP2000514082A (pt)
AR (1) AR007834A1 (pt)
AT (1) ATE218559T1 (pt)
AU (1) AU3546997A (pt)
CA (1) CA2259278A1 (pt)
CO (1) CO4890872A1 (pt)
DE (1) DE69713098T2 (pt)
DK (1) DK0912536T3 (pt)
ES (1) ES2177988T3 (pt)
FR (1) FR2750989B1 (pt)
IN (1) IN188980B (pt)
MA (1) MA24258A1 (pt)
PE (1) PE69499A1 (pt)
PT (1) PT912536E (pt)
TN (1) TNSN97118A1 (pt)
UY (1) UY24609A1 (pt)
WO (1) WO1998001435A1 (pt)
ZA (1) ZA976071B (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5973160A (en) 1992-12-23 1999-10-26 Poss; Michael A. Methods for the preparation of novel sidechain-bearing taxanes
US5750736A (en) * 1996-07-11 1998-05-12 Napro Biotherapeutics, Inc. Method for acylating 10-deacetylbaccatin III selectively at the c-10 position
US7288665B1 (en) 1997-08-18 2007-10-30 Florida State University Process for selective derivatization of taxanes

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2698871B1 (fr) * 1992-12-09 1995-02-24 Rhone Poulenc Rorer Sa Nouveau taxoïdes, leur préparation et les compositions pharmaceutiques qui les contiennent.
FR2702212B1 (fr) * 1993-03-02 1995-04-07 Rhone Poulenc Rorer Sa Nouveaux taxoïdes, leur préparation et les compositions pharmaceutiques qui les contiennent.
FR2718135B1 (fr) * 1994-04-05 1996-04-26 Rhone Poulenc Rorer Sa Procédé de préparation d'hydroxy-7 taxanes.
FR2721023B1 (fr) * 1994-06-09 1996-07-12 Rhone Poulenc Rorer Sa Nouveaux Taxoïdes, leur préparation et les compositions pharmaceutiques qui les contiennent.

Also Published As

Publication number Publication date
PE69499A1 (es) 1999-10-15
IN188980B (pt) 2002-11-30
UY24609A1 (es) 2001-08-27
EP0912536A1 (fr) 1999-05-06
EP0912536B1 (fr) 2002-06-05
ATE218559T1 (de) 2002-06-15
JP2000514082A (ja) 2000-10-24
ES2177988T3 (es) 2002-12-16
DE69713098T2 (de) 2002-11-28
FR2750989B1 (fr) 1998-09-25
US6127555A (en) 2000-10-03
DE69713098D1 (de) 2002-07-11
CO4890872A1 (es) 2000-02-28
AU3546997A (en) 1998-02-02
FR2750989A1 (fr) 1998-01-16
DK0912536T3 (da) 2002-09-16
WO1998001435A1 (fr) 1998-01-15
TNSN97118A1 (fr) 2005-03-15
MA24258A1 (fr) 1998-04-01
ZA976071B (en) 1998-02-02
AR007834A1 (es) 1999-11-24
CA2259278A1 (fr) 1998-01-15

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