PT88357A - Processo para a preparacao de novos derivados do acido 2-aza-biciclooctano-3-carboxilico - Google Patents

Processo para a preparacao de novos derivados do acido 2-aza-biciclooctano-3-carboxilico

Info

Publication number: PT88357A
Authority: PT; Portugal
Prior art keywords: formula; derivative; see diagramm; iii; compound
Prior art date: 1987-08-28

Application number

PT88357A

Other languages

English (en)

Other versions

PT88357B (pt

Inventor

Michel Vincent

Georges Remond

Michel Laubie

Original Assignee

Obrecht Gary W

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1987-08-28

Filing date

1988-08-26

Publication date

1989-06-30

1988-08-26 Application filed by Obrecht Gary W filed Critical Obrecht Gary W

1989-06-30 Publication of PT88357A publication Critical patent/PT88357A/pt

1995-03-31 Publication of PT88357B publication Critical patent/PT88357B/pt

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
- C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Bioinformatics & Cheminformatics (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Genetics & Genomics (AREA)
Biochemistry (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Molecular Biology (AREA)
Pain & Pain Management (AREA)
Biophysics (AREA)
Neurology (AREA)
Diabetes (AREA)
Rheumatology (AREA)
Ophthalmology & Optometry (AREA)
Gastroenterology & Hepatology (AREA)
Vascular Medicine (AREA)
Biomedical Technology (AREA)
Urology & Nephrology (AREA)
Hematology (AREA)
Neurosurgery (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Indole Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Medicinal Preparation (AREA)

PT88357A 1987-08-28 1988-08-26 Processo para a preparacao de novos derivados do acido 2-aza-biciclooctano-3-carboxilico PT88357B (pt)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR8712013A FR2619813B1 (fr)	1987-08-28	1987-08-28	Nouveaux derives de l'acide aza - 2 bicyclooctane carboxylique - 3, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent

Publications (2)

Publication Number	Publication Date
PT88357A true PT88357A (pt)	1989-06-30
PT88357B PT88357B (pt)	1995-03-31

Family

ID=9354475

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PT88357A PT88357B (pt)	1987-08-28	1988-08-26	Processo para a preparacao de novos derivados do acido 2-aza-biciclooctano-3-carboxilico

Country Status (16)

Country	Link
US (1)	US4959372A (pt)
EP (1)	EP0305297B1 (pt)
JP (1)	JPS6471875A (pt)
AT (1)	ATE52789T1 (pt)
AU (1)	AU612689B2 (pt)
CA (1)	CA1327800C (pt)
DE (1)	DE3860148D1 (pt)
DK (1)	DK170978B1 (pt)
ES (1)	ES2031616T3 (pt)
FR (1)	FR2619813B1 (pt)
GR (1)	GR3000677T3 (pt)
IE (1)	IE60505B1 (pt)
NZ (1)	NZ225943A (pt)
OA (1)	OA08754A (pt)
PT (1)	PT88357B (pt)
ZA (1)	ZA886368B (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2655989B1 (fr) *	1989-12-20	1992-02-28	Adir	Nouveaux derives d'amino-acides substitues, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
US5458883A (en) *	1994-01-12	1995-10-17	Duke University	Method of treating disorders of the eye
JP2004500906A (ja) *	1999-11-12	2004-01-15	ルーベン，　レオ	電気的調節および化学的調節のための心臓デバイス、ならびに心肺障害の処置のための血管作用性腸ペプチド
MXPA03008636A (es)	2001-03-26	2003-12-08	Kotobuki Pharmaceutical Co Ltd	Derivados de isoquinuclidina, metodo para fabricar los mismos y agentes terapeuticos que contienen estos compuestos.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL58849A (en) *	1978-12-11	1983-03-31	Merck & Co Inc	Carboxyalkyl dipeptides and derivatives thereof,their preparation and pharmaceutical compositions containing them
FR2492381A1 (fr) *	1980-10-21	1982-04-23	Science Union & Cie	Nouveaux acides aza bicyclo alcane carboxyliques substitues leurs procedes de preparation et leur emploi comme inhibiteur d'enzyme
DE3227055A1 (de) *	1982-07-20	1984-01-26	Hoechst Ag, 6230 Frankfurt	Neue derivate der 2-aza-bicyclo(2.2.2)octan-3-carbonsaeure, verfahren zu ihrer herstellung, diese enthaltende mittel und deren verwendung sowie 2-aza-bicyclo(2.2.2)octan-3-carbonsaeure als zwischenstufe und verfahren zu deren herstellung

1987
- 1987-08-28 FR FR8712013A patent/FR2619813B1/fr not_active Expired - Lifetime
1988
- 1988-08-11 CA CA000574529A patent/CA1327800C/fr not_active Expired - Fee Related
- 1988-08-24 DK DK472788A patent/DK170978B1/da active
- 1988-08-26 NZ NZ225943A patent/NZ225943A/xx unknown
- 1988-08-26 IE IE259988A patent/IE60505B1/en not_active IP Right Cessation
- 1988-08-26 ES ES198888402165T patent/ES2031616T3/es not_active Expired - Lifetime
- 1988-08-26 JP JP63212329A patent/JPS6471875A/ja active Pending
- 1988-08-26 DE DE8888402165T patent/DE3860148D1/de not_active Expired - Lifetime
- 1988-08-26 US US07/237,497 patent/US4959372A/en not_active Expired - Fee Related
- 1988-08-26 ZA ZA886368A patent/ZA886368B/xx unknown
- 1988-08-26 AT AT88402165T patent/ATE52789T1/de not_active IP Right Cessation
- 1988-08-26 OA OA59416A patent/OA08754A/xx unknown
- 1988-08-26 PT PT88357A patent/PT88357B/pt not_active IP Right Cessation
- 1988-08-26 EP EP88402165A patent/EP0305297B1/fr not_active Expired - Lifetime
- 1988-08-26 AU AU21594/88A patent/AU612689B2/en not_active Ceased
1990
- 1990-07-27 GR GR90400526T patent/GR3000677T3/el unknown

Also Published As

Publication number	Publication date
JPS6471875A (en)	1989-03-16
GR3000677T3 (en)	1991-09-27
EP0305297B1 (fr)	1990-05-16
FR2619813B1 (fr)	1991-05-03
AU612689B2 (en)	1991-07-18
IE882599L (en)	1989-02-28
DK472788A (da)	1989-03-01
PT88357B (pt)	1995-03-31
US4959372A (en)	1990-09-25
DE3860148D1 (de)	1990-06-21
AU2159488A (en)	1989-03-09
CA1327800C (fr)	1994-03-15
ATE52789T1 (de)	1990-06-15
DK170978B1 (da)	1996-04-09
EP0305297A1 (fr)	1989-03-01
IE60505B1 (en)	1994-07-27
ES2031616T3 (es)	1992-12-16
DK472788D0 (da)	1988-08-24
FR2619813A1 (fr)	1989-03-03
ZA886368B (en)	1989-05-30
NZ225943A (en)	1990-06-26
OA08754A (fr)	1989-03-31

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Legal Events

Date

Code

Title

Description

1995-03-31

FG3A

Patent granted, date of granting

Effective date: 19940909

1998-07-31

MM3A

Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 19980331