PT67352B - PROCESSES FOR THE PREPARATION OF THIAZOLIDINACARBOXIDIC ACIDS AND ACIDS - Google Patents

PROCESSES FOR THE PREPARATION OF THIAZOLIDINACARBOXIDIC ACIDS AND ACIDS

Info

Publication number
PT67352B
PT67352B PT67352A PT6735277A PT67352B PT 67352 B PT67352 B PT 67352B PT 67352 A PT67352 A PT 67352A PT 6735277 A PT6735277 A PT 6735277A PT 67352 B PT67352 B PT 67352B
Authority
PT
Portugal
Prior art keywords
acids
thiazolidinacarboxidic
processes
preparation
thiazolidinacarboxidic acids
Prior art date
Application number
PT67352A
Other languages
French (fr)
Portuguese (pt)
Other versions
PT67352A (en
Inventor
Miguel Angel Ondetti
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of PT67352A publication Critical patent/PT67352A/en
Publication of PT67352B publication Critical patent/PT67352B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/281,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/301,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/04Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D277/06Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D279/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/041,3-Thiazines; Hydrogenated 1,3-thiazines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D279/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/101,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/121,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
PT67352A 1976-12-03 1977-12-02 PROCESSES FOR THE PREPARATION OF THIAZOLIDINACARBOXIDIC ACIDS AND ACIDS PT67352B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US74728176A 1976-12-03 1976-12-03
US83610777A 1977-09-23 1977-09-23

Publications (2)

Publication Number Publication Date
PT67352A PT67352A (en) 1978-01-01
PT67352B true PT67352B (en) 1979-05-15

Family

ID=27114718

Family Applications (1)

Application Number Title Priority Date Filing Date
PT67352A PT67352B (en) 1976-12-03 1977-12-02 PROCESSES FOR THE PREPARATION OF THIAZOLIDINACARBOXIDIC ACIDS AND ACIDS

Country Status (28)

Country Link
JP (1) JPS5382778A (en)
AR (1) AR220689A1 (en)
AT (1) AT363467B (en)
AU (1) AU518147B2 (en)
BG (1) BG32269A3 (en)
CA (1) CA1146940A (en)
CH (1) CH634062A5 (en)
DD (1) DD133798A5 (en)
DE (1) DE2752719C2 (en)
DK (1) DK152494C (en)
EG (1) EG13037A (en)
ES (1) ES464555A1 (en)
FI (1) FI67378C (en)
FR (1) FR2372817A1 (en)
GB (1) GB1578940A (en)
GR (1) GR72453B (en)
HK (1) HK55881A (en)
IE (1) IE46169B1 (en)
IL (1) IL53352A0 (en)
IN (1) IN146945B (en)
IT (1) IT1092179B (en)
NL (3) NL171055C (en)
NO (1) NO148416C (en)
NZ (1) NZ185800A (en)
PT (1) PT67352B (en)
RO (2) RO72596A (en)
SE (1) SE441267B (en)
YU (1) YU41823B (en)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1105731B (en) * 1977-06-29 1985-11-04 Yoshitomi Pharmaceutical THIAZOLIDINE COMPOUNDS
JPS5455565A (en) * 1977-10-06 1979-05-02 Santen Pharmaceut Co Ltd Novel thiazolidine derivative
US4430344A (en) * 1978-04-08 1984-02-07 Santen Pharmaceutical Co., Ltd. Antihypertensive 4-thiazolidinecarboxylic acids
JPS557255A (en) * 1978-07-03 1980-01-19 Santen Pharmaceut Co Ltd Thiazolidine derivative
JPS5531022A (en) * 1978-08-24 1980-03-05 Yoshitomi Pharmaceut Ind Ltd Hydroxamic acid derivative and its preparation
GR73585B (en) * 1978-09-11 1984-03-26 Univ Miami
JPS5540622A (en) * 1978-09-14 1980-03-22 Santen Pharmaceut Co Ltd Hypotensive agent
JPS5829950B2 (en) * 1978-10-05 1983-06-25 ウェルファイド株式会社 Cyclic iminocarboxylic acid derivatives and their salts
JPS5562060A (en) * 1978-10-31 1980-05-10 Santen Pharmaceut Co Ltd Sulfur-containing compound
US4483861A (en) * 1978-10-31 1984-11-20 Santen Pharmaceutical Co., Ltd. Antihypertensive sulfur-containing compounds
JPS565415A (en) * 1979-06-26 1981-01-20 Santen Pharmaceut Co Ltd Ester-type hypotensor
US4347371A (en) * 1978-12-30 1982-08-31 Santen Pharmaceutical Co., Ltd. Disulfide compounds
JPS55124757A (en) * 1979-03-17 1980-09-26 Santen Pharmaceut Co Ltd Sulfur-containing compound
JPS5683483A (en) * 1979-12-13 1981-07-08 Santen Pharmaceut Co Ltd Thiazolidine compound
JPS56139455A (en) * 1980-04-02 1981-10-30 Santen Pharmaceut Co Ltd Sulfur-containing acylaminoacid
DE3152643A1 (en) * 1980-12-29 1982-12-16 Santen Pharmaceutical Co Ltd HETEROCYCLIC 5-MEMBERED RING COMPOUNDS
JPH0662529B2 (en) * 1984-07-13 1994-08-17 三共株式会社 Amino acid derivative
EP0190685B1 (en) * 1985-02-04 1992-07-01 G.D. Searle & Co. Heterocyclic amides

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2446100C3 (en) * 1974-09-26 1982-01-14 Ludwig Merckle Kg Chem. Pharm. Fabrik, 7902 Blaubeuren Phenoxyalkanecarboxamides of thiazolidinecarboxylic acids, process for their preparation and pharmaceuticals
AU509899B2 (en) * 1976-02-13 1980-05-29 E.R. Squibb & Sons, Inc. Proline derivatives and related compounds

Also Published As

Publication number Publication date
YU283777A (en) 1983-01-21
BG32269A3 (en) 1982-06-15
RO72596A (en) 1983-08-03
IL53352A0 (en) 1978-01-31
SE7713722L (en) 1978-06-04
IT1092179B (en) 1985-07-06
NO774126L (en) 1978-06-06
AU518147B2 (en) 1981-09-17
SE441267B (en) 1985-09-23
IE46169B1 (en) 1983-03-09
FR2372817B1 (en) 1981-06-19
EG13037A (en) 1980-12-31
NO148416C (en) 1983-10-12
ES464555A1 (en) 1978-09-01
DE2752719A1 (en) 1978-06-08
GR72453B (en) 1983-11-09
NL171055C (en) 1983-02-01
FR2372817A1 (en) 1978-06-30
HK55881A (en) 1981-11-20
NO148416B (en) 1983-06-27
FI67378C (en) 1985-03-11
FI67378B (en) 1984-11-30
RO72596B (en) 1983-07-30
FI773640A (en) 1978-06-04
AT363467B (en) 1981-08-10
DD133798A5 (en) 1979-01-24
JPS5382778A (en) 1978-07-21
DK152494B (en) 1988-03-07
DE2752719C2 (en) 1982-03-25
DK152494C (en) 1988-07-25
ATA857677A (en) 1981-01-15
NZ185800A (en) 1980-04-28
CA1146940A (en) 1983-05-24
JPS618834B2 (en) 1986-03-18
NL8201146A (en) 1982-07-01
PT67352A (en) 1978-01-01
AU3037977A (en) 1979-05-17
NL7713274A (en) 1978-06-06
NL8201145A (en) 1982-07-01
CH634062A5 (en) 1983-01-14
YU41823B (en) 1988-02-29
GB1578940A (en) 1980-11-12
DK538277A (en) 1978-06-04
IN146945B (en) 1979-10-20
AR220689A1 (en) 1980-11-28
IE46169L (en) 1978-06-03
RO78013A (en) 1981-12-25

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