PT66779A - PROCESS FOR THE PREPARATION OF 5- (2-FUROIL) -, 5- (2-TENOIL) -, 5- (3-FUROIL) -, AND 5- (3TENOIL) -1,2-DIHYDRO-ACID DERIVATIVES 3H-PIRROLE (1,2-ALPHA) PIRROLE-1-CARBOXILIQUE - Google Patents

PROCESS FOR THE PREPARATION OF 5- (2-FUROIL) -, 5- (2-TENOIL) -, 5- (3-FUROIL) -, AND 5- (3TENOIL) -1,2-DIHYDRO-ACID DERIVATIVES 3H-PIRROLE (1,2-ALPHA) PIRROLE-1-CARBOXILIQUE

Info

Publication number: PT66779A
Authority: PT; Portugal
Prior art keywords: furoil; pirrole; carboxilique; 3tenoil; tenoil
Prior art date: 1976-07-14

Application number

PT66779A

Other languages

French (fr)

Portuguese (pt)

Other versions

PT66779B (en

Original Assignee

Syntex Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-07-14

Filing date

1977-07-08

Publication date

1977-08-01

1977-02-23 Priority claimed from US05/771,283 external-priority patent/US4087539A/en

1977-07-08 Application filed by Syntex Inc filed Critical Syntex Inc

1977-08-01 Publication of PT66779A publication Critical patent/PT66779A/en

1978-12-18 Publication of PT66779B publication Critical patent/PT66779B/en

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pain & Pain Management (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Rheumatology (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Urology & Nephrology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)

PT66779A 1976-07-14 1977-07-08 PROCESS FOR THE PREPARATION OF 5- (2-FUROIL) -, 5- (2-TENOIL) -, 5- (3-FUROIL) -ET 5- (3TENOIL) -1,2-DIHYDRO-3H-ACID DERIVATIVES -PIRROLE / 1,2-ALPHA / PIRROLE-1-CARBOXILIC PT66779B (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US70485776A	1976-07-14	1976-07-14
US05/771,283 US4087539A (en)	1976-07-14	1977-02-23	5-(2-Furoyl)-, 5-(2-thenoyl)-, 5-(3-furoyl)- and 5-(3-thenoyl)-1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid derivatives and process for the production thereof

Publications (2)

Publication Number	Publication Date
PT66779A true PT66779A (en)	1977-08-01
PT66779B PT66779B (en)	1978-12-18

Family

ID=27107392

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PT66779A PT66779B (en)	1976-07-14	1977-07-08	PROCESS FOR THE PREPARATION OF 5- (2-FUROIL) -, 5- (2-TENOIL) -, 5- (3-FUROIL) -ET 5- (3TENOIL) -1,2-DIHYDRO-3H-ACID DERIVATIVES -PIRROLE / 1,2-ALPHA / PIRROLE-1-CARBOXILIC

Country Status (26)

Country	Link
JP (1)	JPS539789A (en)
AR (1)	AR218631A1 (en)
AU (1)	AU513385B2 (en)
CA (1)	CA1100140A (en)
CH (2)	CH651045A5 (en)
CS (1)	CS208724B2 (en)
DE (1)	DE2731662A1 (en)
DK (1)	DK152652C (en)
ES (2)	ES460705A1 (en)
FI (1)	FI63407C (en)
FR (1)	FR2361396A1 (en)
GB (1)	GB1554076A (en)
GR (1)	GR61607B (en)
HK (1)	HK17581A (en)
IE (1)	IE45302B1 (en)
IL (1)	IL52492A (en)
IT (1)	IT1117314B (en)
MY (1)	MY8100371A (en)
NL (1)	NL7707652A (en)
NO (1)	NO147563C (en)
NZ (1)	NZ184611A (en)
PL (1)	PL111408B1 (en)
PT (1)	PT66779B (en)
SE (1)	SE434644B (en)
SU (2)	SU664566A3 (en)
YU (2)	YU43157B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4097579A (en) *	1977-03-31	1978-06-27	Syntex (U.S.A.) Inc.	5-(2-Pyrroyl)-1,2-dihydro-3H-pyrrolo 1,2-a!pyrrole-1-carboxylic acid derivatives and process for the production thereof
US4140698A (en) *	1977-07-25	1979-02-20	Syntex (Usa) Inc.	1,2-Dihydro-3H-pyrrolo[1,2-a]pyrrole-1-nitriles
US4353829A (en) *	1980-11-21	1982-10-12	Syntex (U.S.A.) Inc.	Process for 5-aroylation of 1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic esters
JPS5910589A (en) *	1982-06-10	1984-01-20	メルク　エンド　カムパニー　インコーポレーテツド	Antiinflammatory and analgesic novel 5-(pyrrol-2-oyl)-1,2-dihydro-3h-pyrrolo(1,2-a) pyrrole derivative
US4511724A (en) *	1982-06-10	1985-04-16	Merck & Co., Inc.	5-(Pyrrol-2-oyl)-1,2-dihydro-3H-pyrrolo [1,2-a]pyrrole derivatives as anti-inflammatory and analgesic agents
HU198927B (en) *	1987-01-14	1989-12-28	Richter Gedeon Vegyeszet	Process for producing 1-/substituted aminomethyl/-octa-hydroindolo-(2,3-a)quinolizine derivatives, pharmaceutically applicable acid addition salts thereof, as well as pharmaceutical compositions comprising same
US4874871A (en) *	1987-03-25	1989-10-17	Syntex (U.S.A.) Inc.	Process for preparing (+)-2,3-Dihydro-1H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid and related compounds

1977
- 1977-05-17 JP JP5697877A patent/JPS539789A/en active Granted
- 1977-07-07 GR GR53906A patent/GR61607B/en unknown
- 1977-07-07 DK DK307677A patent/DK152652C/en not_active IP Right Cessation
- 1977-07-07 AR AR268357A patent/AR218631A1/en active
- 1977-07-08 PT PT66779A patent/PT66779B/en unknown
- 1977-07-08 IE IE1422/77A patent/IE45302B1/en unknown
- 1977-07-08 NL NL7707652A patent/NL7707652A/en not_active Application Discontinuation
- 1977-07-08 IL IL52492A patent/IL52492A/en unknown
- 1977-07-08 CH CH4005/84A patent/CH651045A5/en not_active IP Right Cessation
- 1977-07-08 CH CH848877A patent/CH644861A5/en not_active IP Right Cessation
- 1977-07-11 FI FI772154A patent/FI63407C/en not_active IP Right Cessation
- 1977-07-11 GB GB28923/77A patent/GB1554076A/en not_active Expired
- 1977-07-11 NZ NZ184611A patent/NZ184611A/en unknown
- 1977-07-12 FR FR7721559A patent/FR2361396A1/en active Granted
- 1977-07-12 CA CA282,600A patent/CA1100140A/en not_active Expired
- 1977-07-12 CS CS774647A patent/CS208724B2/en unknown
- 1977-07-13 SE SE7708142A patent/SE434644B/en not_active IP Right Cessation
- 1977-07-13 NO NO772493A patent/NO147563C/en unknown
- 1977-07-13 IT IT68631/77A patent/IT1117314B/en active
- 1977-07-13 ES ES460705A patent/ES460705A1/en not_active Expired
- 1977-07-13 PL PL1977199602A patent/PL111408B1/en unknown
- 1977-07-13 SU SU772504151A patent/SU664566A3/en active
- 1977-07-13 AU AU26976/77A patent/AU513385B2/en not_active Expired
- 1977-07-13 DE DE19772731662 patent/DE2731662A1/en active Granted
- 1977-12-29 SU SU772558960A patent/SU793400A3/en active
1978
- 1978-05-24 ES ES470213A patent/ES470213A1/en not_active Expired
1981
- 1981-04-30 HK HK175/81A patent/HK17581A/en unknown
- 1981-12-30 MY MY371/81A patent/MY8100371A/en unknown
1983
- 1983-02-28 YU YU476/83A patent/YU43157B/en unknown
- 1983-02-28 YU YU475/83A patent/YU43156B/en unknown

Also Published As

Publication number	Publication date
YU43156B (en)	1989-04-30
YU47583A (en)	1984-06-30
FI63407C (en)	1983-06-10
DK152652B (en)	1988-04-05
AU513385B2 (en)	1980-11-27
HK17581A (en)	1981-05-08
SE434644B (en)	1984-08-06
AU2697677A (en)	1979-01-18
MY8100371A (en)	1981-12-31
CH651045A5 (en)	1985-08-30
FR2361396B1 (en)	1981-11-27
FI63407B (en)	1983-02-28
IT1117314B (en)	1986-02-17
NL7707652A (en)	1978-01-17
CA1100140A (en)	1981-04-28
ES470213A1 (en)	1979-09-16
NO772493L (en)	1978-01-17
CH644861A5 (en)	1984-08-31
CS208724B2 (en)	1981-09-15
GB1554076A (en)	1979-10-17
SU793400A3 (en)	1980-12-30
NZ184611A (en)	1979-03-28
IL52492A0 (en)	1977-10-31
JPS6254110B2 (en)	1987-11-13
IE45302L (en)	1978-01-14
ES460705A1 (en)	1979-10-01
DK152652C (en)	1988-09-12
PT66779B (en)	1978-12-18
DK307677A (en)	1978-01-15
PL199602A1 (en)	1979-01-29
SU664566A3 (en)	1979-05-25
NO147563B (en)	1983-01-24
IE45302B1 (en)	1982-07-28
DE2731662A1 (en)	1978-01-19
DE2731662C2 (en)	1989-11-09
JPS539789A (en)	1978-01-28
IL52492A (en)	1981-06-29
AR218631A1 (en)	1980-06-30
PL111408B1 (en)	1980-08-30
SE7708142L (en)	1978-01-15
FR2361396A1 (en)	1978-03-10
NO147563C (en)	1983-05-18
YU43157B (en)	1989-04-30
GR61607B (en)	1978-12-02
FI772154A (en)	1978-01-15
YU47683A (en)	1984-04-30

Publication	Publication Date	Title
FR2342981A1 (en)	1977-09-30	HYDROGENOSILANES PREPARATION PROCESS
FR2309041A1 (en)	1976-11-19	NETWORK FOR THE DETECTION OF INFRA-RED IMAGES AND ITS MANUFACTURING PROCESS
BE861172A (en)	1978-05-24	PROCESS FOR THE PREPARATION OF ALPHA-AMINO-AMIDES
PT66174A (en)	1977-03-01	PROCESS FOR THE PREPARATION OF 1,2-DIIROL DERIVATIVES AND COMPOSITIONS CONTAINED THEREOF
PT66780A (en)	1977-08-01	PROCESS FOR THE PREPARATION OF 5-AROIL-1,2-DIHYDRO-3H-PIRROLE (1,2-ALPHA) PIRROLE-1-CARBOXILIC ACID DERIVATIVES
MA19294A1 (en)	1982-04-01	PROCESS FOR THE PREPARATION OF SUBSTITUTED IMINO-DIACIDES.
FR2353589A1 (en)	1977-12-30	PROCESS FOR THE PREPARATION OF ORGANOPOLYSILOXANES
PT67004B (en)	1979-02-12	PROCESS FOR THE PREPARATION OF 7-ACILAMINE-8-OXO-3-OXA-1-AZABICICLE- / 4,2,0 / -OCTANE-2-CARBOXIC ACID DERIVATIVES
BE859325A (en)	1978-04-03	PROCESS FOR THE DIRECTED CHLORINATION OF ALCOYLBENZENES
PT66779A (en)	1977-08-01	PROCESS FOR THE PREPARATION OF 5- (2-FUROIL) -, 5- (2-TENOIL) -, 5- (3-FUROIL) -, AND 5- (3TENOIL) -1,2-DIHYDRO-ACID DERIVATIVES 3H-PIRROLE (1,2-ALPHA) PIRROLE-1-CARBOXILIQUE
BE855236A (en)	1977-11-30	OMEGA-NOR-AROMATIC 13,14-DEHYDRO-PROSTAGLANDIN DERIVATIVES AND PROCESS FOR THEIR PREPARATION
RO76587A (en)	1981-04-20	PROCESS FOR THE PREPARATION OF 1,3,4 TRIADIAZOLE DERIVATIVES
BE858806A (en)	1978-03-16	PROCESS FOR THE PREPARATION OF GLYCOL-ALDEHYDE AND ETHYLENE-GLYCOL
BE856723A (en)	1978-01-12	PROCESS FOR THE PREPARATION OF VINCAMINE AND RELATED ALKALOIDS
FR2339588A1 (en)	1977-08-26	PROCESS FOR THE PREPARATION OF ALDEHYDES AND AROMATIC KETONES
PT66029B (en)	1978-06-19	PROCESS FOR THE PREPARATION OF NEW HYDRAZINE DERIVATIVES
BE880031A (en)	1980-05-14	PROCESS FOR THE PREPARATION OF 1 ALPHA, 3 BETA-DIHYDROXY-DELTA 5-STEROIDES
BE867414A (en)	1978-09-18	PROCESS FOR THE PREPARATION OF HYDROXY-ALPHA-AMINOBENZYLPENICILLINS
BE867228A (en)	1978-11-20	PROCESS FOR THE PREPARATION OF HYDROXYPHENYLGLYCOCOLLES
BE854815A (en)	1977-09-16	MALEIC ANHYDRIDE PREPARATION PROCESS
BE852700R (en)	1977-09-21	PROCESS FOR PREPARATION OF OXAPHOSPHOLANES-1,2
PT66064B (en)	1978-06-23	PROCESS FOR THE PREPARATION OF ALKALOID DERIVATIVES
BE874547A (en)	1979-09-03	PERFECTED PROCESS FOR THE PREPARATION OF ORGANO-THIOALDOXIMES
AR224378A1 (en)	1981-11-30	PROCEDURE FOR THE PREPARATION OF 1,2,4,5-TETRAHYDRO-7-ALCOXI- (AND 7,8-DIALCOXI) -3H, 3-BENZAZEPINES AND 3-SUBSTITUTED DERIVATIVES OF THE SAME FROM THE CORRESPONDING FENETILAMINES
FR2323674A1 (en)	1977-04-08	PROCESS FOR THE PREPARATION OF SUBSTITUTE 1-PHENYL-2,2,2-TRIHALOGENO-ETHANOLS ESTERS