PT2764008T - Processo para a produção de estetrol - Google Patents

Processo para a produção de estetrol

Info

Publication number: PT2764008T
Authority: PT; Portugal
Prior art keywords: estetrol; production
Prior art date: 2011-10-07

Application number

PT127786648T

Other languages

English (en)

Inventor

Pascal Jean-Claude

Original Assignee

Estetra Sprl

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2011-10-07

Filing date

2012-10-05

Publication date

2016-11-10

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48043195&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT2764008(T) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2012-10-05 Application filed by Estetra Sprl filed Critical Estetra Sprl

2016-11-10 Publication of PT2764008T publication Critical patent/PT2764008T/pt

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0066—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J75/00—Processes for the preparation of steroids in general
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Steroid Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

PT127786648T 2011-10-07 2012-10-05 Processo para a produção de estetrol PT2764008T (pt)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US201161544591P	2011-10-07	2011-10-07
EP11184278		2011-10-07

Publications (1)

Publication Number	Publication Date
PT2764008T true PT2764008T (pt)	2016-11-10

Family

ID=48043195

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PT127786648T PT2764008T (pt)	2011-10-07	2012-10-05	Processo para a produção de estetrol

Country Status (27)

Country	Link
US (1)	US8987484B2 (pt)
EP (1)	EP2764008B1 (pt)
JP (1)	JP6196625B2 (pt)
KR (1)	KR102007874B1 (pt)
CN (1)	CN103890001B (pt)
AU (1)	AU2012320423C1 (pt)
BR (1)	BR112014008196B8 (pt)
CA (1)	CA2847813C (pt)
CL (1)	CL2014000802A1 (pt)
CY (1)	CY1118674T1 (pt)
DK (1)	DK2764008T3 (pt)
EA (1)	EA024003B1 (pt)
ES (1)	ES2593316T3 (pt)
HK (1)	HK1199882A1 (pt)
HR (1)	HRP20161282T1 (pt)
HU (1)	HUE028963T2 (pt)
IN (1)	IN2014MN00841A (pt)
LT (1)	LT2764008T (pt)
ME (1)	ME02527B (pt)
MX (1)	MX348917B (pt)
PL (1)	PL2764008T3 (pt)
PT (1)	PT2764008T (pt)
RS (1)	RS55231B1 (pt)
SG (1)	SG11201401282PA (pt)
SI (1)	SI2764008T1 (pt)
SM (1)	SMT201600375B (pt)
WO (1)	WO2013050553A1 (pt)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
PL2714710T3 (pl)	2011-06-01	2017-03-31	Estetra S.P.R.L.	Sposób wytwarzania estetrolowych związków pośrednich
KR101957937B1 (ko)	2011-06-01	2019-03-14	에스테트라 에스.피.알.엘.	에스테트롤 중간체의 제조 방법
EP2383279A1 (en)	2011-07-19	2011-11-02	Pantarhei Bioscience B.V.	Process for the preparation of estetrol
WO2013034780A2 (en) *	2012-12-20	2013-03-14	Crystal Pharma, S.A.U.	Process for the preparation of estetrol and related compounds
CA2924255C (en)	2013-09-18	2022-11-22	Crystal Pharma, S.A.U.	Process for the preparation of estetrol
RS62844B1 (sr)	2015-06-18	2022-02-28	Estetra Srl	Orodisperzibilna dozna jedinica koja sadrži komponentu estetrola
CA2988498C (en)	2015-06-18	2022-02-08	Mithra Pharmaceuticals S.A.	Orodispersible dosage unit containing an estetrol component
JP6866561B2 (ja)	2015-06-18	2021-04-28	エステトラソシエテプリーヴアレスポンサビリテリミテ	エステトロールを含有する口腔内崩壊錠
SI3310346T1 (sl) *	2015-06-18	2021-07-30	Estetra Sprl	Orodisperzibilna tableta, ki vsebuje estetrol
KR20220144885A (ko)	2016-08-05	2022-10-27	에스테트라, 소시에떼 아 레스폰서빌리떼 리미떼	월경통 및 생리통의 관리방법
JOP20200260A1 (ar)	2018-04-19	2019-10-19	Estetra Sprl	مركبات واستخداماتها للتخفيف من الأعراض المصاحبة لانقطاع الطمث
TWI801561B (zh)	2018-04-19	2023-05-11	比利時商依思特拉私人有限責任公司	化合物及其用於緩解絕經相關症狀的用途
HU231240B1 (hu) *	2019-09-03	2022-04-28	Richter Gedeon Nyrt.	Ipari eljárás nagytisztaságú ösztetrol hatóanyag előállítására
IT201900017414A1 (it)	2019-09-27	2021-03-27	Ind Chimica Srl	Processo per la preparazione di (15α,16α,17β)-estra-1,3,5(10)-triene-3,15,16,17-tetrolo (Estetrolo) ed intermedi di detto processo
IT201900021879A1 (it)	2019-11-22	2021-05-22	Ind Chimica Srl	PROCESSO PER LA PREPARAZIONE DI (15α,16α,17β)-ESTRA-1,3,5(10)-TRIENE-3,15,16,17-TETROLO (ESTETROLO) ED INTERMEDI DI DETTO PROCESSO
BR112022005359A2 (pt) *	2019-09-27	2022-07-19	Ind Chimica Srl	Processo de preparação de (15a,16a,17ss)-estra-1,3,5(10)-trieno-3,15,16,17-tetrol(estetrol) e intermediários do referido processo
IT202100019631A1 (it)	2021-07-23	2023-01-23	Newchem S P A	Metodo per produrre estetrolo e i suoi intermedi
WO2023021026A1 (en)	2021-08-17	2023-02-23	Aspen Oss B.V.	A synthetic pathway to estra-1,3,5(10)-triene-3,15a,16a,17b-tetrol
GB202405864D0 (en)	2021-10-01	2024-06-12	Ind Chimica S R L	Process for preparing (15alpha,16alpha,17eta)-estra-1,3,5-(10)-triene-3,15,16,17-tetrol(estetrol) monohydrate

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
TW548277B (en) *	1999-07-16	2003-08-21	Akzo Nobel Nv	Orally active androgens
ATE317396T1 (de) *	1999-12-02	2006-02-15	Akzo Nobel Nv	14,15-beta-methylen substituierte androgene
AU2003279624A1 (en) *	2002-11-08	2004-06-07	Pantarhei Bioscience B.V.	Synthesis of estetrol via estrone derived steroids
UA89964C2 (ru) *	2004-09-08	2010-03-25	Н.В. Органон	15β-ЗАМЕЩЕННЫЕ СТЕРОИДЫ, КОТОРЫЕ ИМЕЮТ СЕЛЕКТИВНУЮ ЭСТРОГЕННУЮ АКТИВНОСТЬ
PL2714710T3 (pl)	2011-06-01	2017-03-31	Estetra S.P.R.L.	Sposób wytwarzania estetrolowych związków pośrednich
KR101957937B1 (ko)	2011-06-01	2019-03-14	에스테트라 에스.피.알.엘.	에스테트롤 중간체의 제조 방법
EP2383279A1 (en) *	2011-07-19	2011-11-02	Pantarhei Bioscience B.V.	Process for the preparation of estetrol

2012
- 2012-10-05 SG SG11201401282PA patent/SG11201401282PA/en unknown
- 2012-10-05 WO PCT/EP2012/069761 patent/WO2013050553A1/en active Application Filing
- 2012-10-05 KR KR1020147007408A patent/KR102007874B1/ko active IP Right Grant
- 2012-10-05 US US14/349,940 patent/US8987484B2/en active Active
- 2012-10-05 AU AU2012320423A patent/AU2012320423C1/en active Active
- 2012-10-05 LT LTEP12778664.8T patent/LT2764008T/lt unknown
- 2012-10-05 RS RS20160859A patent/RS55231B1/sr unknown
- 2012-10-05 PT PT127786648T patent/PT2764008T/pt unknown
- 2012-10-05 ME MEP-2016-229A patent/ME02527B/me unknown
- 2012-10-05 EP EP12778664.8A patent/EP2764008B1/en active Active
- 2012-10-05 DK DK12778664.8T patent/DK2764008T3/en active
- 2012-10-05 JP JP2014533925A patent/JP6196625B2/ja active Active
- 2012-10-05 BR BR112014008196A patent/BR112014008196B8/pt active IP Right Grant
- 2012-10-05 CA CA2847813A patent/CA2847813C/en active Active
- 2012-10-05 ES ES12778664.8T patent/ES2593316T3/es active Active
- 2012-10-05 CN CN201280049319.2A patent/CN103890001B/zh active Active
- 2012-10-05 EA EA201490713A patent/EA024003B1/ru unknown
- 2012-10-05 MX MX2014003723A patent/MX348917B/es active IP Right Grant
- 2012-10-05 HU HUE12778664A patent/HUE028963T2/en unknown
- 2012-10-05 SI SI201230705A patent/SI2764008T1/sl unknown
- 2012-10-05 PL PL12778664T patent/PL2764008T3/pl unknown
2014
- 2014-04-02 CL CL2014000802A patent/CL2014000802A1/es unknown
- 2014-05-05 IN IN841MUN2014 patent/IN2014MN00841A/en unknown
2015
- 2015-01-13 HK HK15100344.6A patent/HK1199882A1/zh unknown
2016
- 2016-10-05 HR HRP20161282TT patent/HRP20161282T1/hr unknown
- 2016-10-10 CY CY20161101001T patent/CY1118674T1/el unknown
- 2016-10-17 SM SM201600375T patent/SMT201600375B/it unknown

Also Published As

Publication number	Publication date
CY1118674T1 (el)	2017-07-12
CN103890001B (zh)	2016-05-04
SMT201600375B (it)	2017-01-10
NZ621973A (en)	2015-08-28
AU2012320423A1 (en)	2014-03-20
ME02527B (me)	2017-02-20
MX348917B (es)	2017-07-04
AU2012320423B2 (en)	2017-02-09
EP2764008B1 (en)	2016-08-17
KR20140083994A (ko)	2014-07-04
CA2847813C (en)	2018-12-11
BR112014008196B1 (pt)	2020-10-20
CL2014000802A1 (es)	2014-11-14
ES2593316T3 (es)	2016-12-07
WO2013050553A1 (en)	2013-04-11
JP2014528438A (ja)	2014-10-27
SG11201401282PA (en)	2014-05-29
PL2764008T3 (pl)	2017-04-28
CN103890001A (zh)	2014-06-25
DK2764008T3 (en)	2016-11-07
LT2764008T (lt)	2016-11-10
EA201490713A1 (ru)	2014-07-30
KR102007874B1 (ko)	2019-08-06
CA2847813A1 (en)	2013-04-11
BR112014008196B8 (pt)	2020-12-15
BR112014008196A2 (pt)	2017-04-18
US8987484B2 (en)	2015-03-24
US20140243539A1 (en)	2014-08-28
RS55231B1 (sr)	2017-02-28
MX2014003723A (es)	2014-10-13
IN2014MN00841A (pt)	2015-07-03
HRP20161282T1 (hr)	2016-11-18
JP6196625B2 (ja)	2017-09-13
AU2012320423C1 (en)	2018-01-25
HK1199882A1 (zh)	2015-07-24
EP2764008A1 (en)	2014-08-13
EA024003B1 (ru)	2016-08-31
SI2764008T1 (sl)	2016-10-28
HUE028963T2 (en)	2017-01-30

Publication	Publication Date	Title
HK1199882A1 (zh)	2015-07-24	用於製備雌四醇的方法
HRP20160692T1 (hr)	2016-08-12	Postupak za proizvodnju intermedijera estetrola
PL2744768T3 (pl)	2016-10-31	Sposób wytwarzania klinkieru zawierającego ternezyt
EP2699534A4 (en)	2015-01-14	PROCESS FOR PRODUCING TRANS-1233zd
PL2734536T3 (pl)	2017-03-31	Sposób wytwarzania estetrolu
ZA201308445B (en)	2015-07-29	Process for the production of estetrol intermediates
SG11201400939YA (en)	2014-07-30	Process for the preparation of methoxymelonal
EP2797868A4 (en)	2015-08-12	PROCESS FOR PRODUCING HEXANEDIOLS
HK1205097A1 (en)	2015-12-11	Process for the production of methylbutinol
ZA201205844B (en)	2014-01-29	Process for the production of anhydrides
EP2740719A4 (en)	2015-03-11	PROCESS FOR THE PREPARATION OF A-FLUOROALDEHYDE
IL231645A (en)	2016-09-29	Process for making isoxazolyl - methoxy - nicotinic acids
HUE044066T2 (hu)	2019-09-30	Eljárás metilén-difenil-diizocianát elõállítására
PL2681199T3 (pl)	2019-03-29	Sposób wytwarzania (-)-hupercyny A
ZA201403104B (en)	2016-07-27	Process for the preparation of higher alcohols
SG11201403392UA (en)	2014-10-30	Process for the production of alcohols
PL2689069T3 (pl)	2017-04-28	Proces produkcji podsypki (balastu)
SG11201403380UA (en)	2014-09-26	Process for the production of alcohols
EP2700716A4 (en)	2015-04-29	PROCESS FOR THE PREPARATION OF L-CYSTONE
PL394420A1 (pl)	2012-10-08	Sposób wytwarzania dilauroilofluoresceiny
PL394378A1 (pl)	2012-10-08	Sposób otrzymywania E-2-amino-4-nitrostilbenów