PT1467724E - Composicao farmaceutica orodispersavel de agomelatina - Google Patents

Composicao farmaceutica orodispersavel de agomelatina

Info

Publication number
PT1467724E
PT1467724E PT03731733T PT03731733T PT1467724E PT 1467724 E PT1467724 E PT 1467724E PT 03731733 T PT03731733 T PT 03731733T PT 03731733 T PT03731733 T PT 03731733T PT 1467724 E PT1467724 E PT 1467724E
Authority
PT
Portugal
Prior art keywords
orodispersavel
agomelatin
pharmaceutical composition
pharmaceutical
composition
Prior art date
Application number
PT03731733T
Other languages
English (en)
Inventor
Patrick Wuthrich
Rolland Herve
Julien Marc
Tharrault Francois
Original Assignee
Servier Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Servier Lab filed Critical Servier Lab
Publication of PT1467724E publication Critical patent/PT1467724E/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
PT03731733T 2002-01-23 2003-01-22 Composicao farmaceutica orodispersavel de agomelatina PT1467724E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0200792A FR2834890B1 (fr) 2002-01-23 2002-01-23 Composition pharmaceutique orodispersible d'agomelatine

Publications (1)

Publication Number Publication Date
PT1467724E true PT1467724E (pt) 2006-08-31

Family

ID=27589556

Family Applications (1)

Application Number Title Priority Date Filing Date
PT03731733T PT1467724E (pt) 2002-01-23 2003-01-22 Composicao farmaceutica orodispersavel de agomelatina

Country Status (28)

Country Link
US (2) US20050131071A1 (pt)
EP (1) EP1467724B1 (pt)
JP (2) JP4335011B2 (pt)
KR (1) KR100605798B1 (pt)
CN (1) CN1287780C (pt)
AR (1) AR038207A1 (pt)
AT (1) ATE324882T1 (pt)
AU (1) AU2003220786B2 (pt)
BR (1) BRPI0307072B1 (pt)
CA (1) CA2473201C (pt)
CY (1) CY1105415T1 (pt)
DE (1) DE60304993T2 (pt)
DK (1) DK1467724T3 (pt)
EA (1) EA007299B1 (pt)
ES (1) ES2262999T3 (pt)
FR (1) FR2834890B1 (pt)
GE (1) GEP20063818B (pt)
HK (1) HK1076742A1 (pt)
MA (1) MA27101A1 (pt)
MX (1) MXPA04007198A (pt)
NO (1) NO333712B1 (pt)
NZ (1) NZ533843A (pt)
PL (1) PL204937B1 (pt)
PT (1) PT1467724E (pt)
SI (1) SI1467724T1 (pt)
UA (1) UA77752C2 (pt)
WO (1) WO2003061644A1 (pt)
ZA (1) ZA200405153B (pt)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2834889B1 (fr) * 2002-01-18 2004-04-02 Roquette Freres Forme pharmaceutique solide orodispersible
US20030228370A1 (en) * 2002-06-11 2003-12-11 Michel Serpelloni Orodispersible solid pharmaceutical form
AR047553A1 (es) * 2003-07-04 2006-01-25 Lundbeck & Co As H La combinacion de un inhibidor de reabsorcion de serotonina y agomelatina
FR2884714B1 (fr) * 2005-04-20 2011-05-06 Servier Lab Utilisation de l'agomelatine pour l'obtention de medicaments destines au traitement des troubles bipolaires
FR2890562B1 (fr) * 2005-09-09 2012-10-12 Servier Lab Utilisation de l'agomelatine pour l'obtention de medicaments destines au traitement des troubles du sommeil chez le patient deprime
FR2890564B1 (fr) * 2005-09-09 2007-10-19 Servier Lab Nouvelle association entre l'agomelatine et un inhibiteur de la recapture de la noradrenaline et les compositions pharmaceutiques qui la contiennent
FR2894475B1 (fr) 2005-12-14 2008-05-16 Servier Lab Composition pharmaceutique orodispersible pour administra- -tion oromucosale ou sublinguale d'agomelatine
US20070275075A1 (en) * 2006-03-06 2007-11-29 Ilan Zalit Ezetimibe compositions
CN101206200B (zh) * 2006-12-19 2011-12-28 北京德众万全药物技术开发有限公司 一种分离分析阿戈美拉汀中间体及其终产品的hplc方法
EP2150525A1 (en) * 2007-05-01 2010-02-10 Concert Pharmaceuticals Inc. Naphthyl(ethyl) acetamides
EP2359813A1 (en) * 2010-02-04 2011-08-24 Ratiopharm GmbH Pharmaceutical composition comprising N-(2-chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyethyl)-1-piperazinyl]-2-methyl-4-pyrimidinyl]amino]-5-thiazolecarboxamid
CN101836966A (zh) * 2010-05-27 2010-09-22 北京万全阳光医药科技有限公司 一种含有阿戈美拉汀的口腔崩解片
CN102579415B (zh) * 2011-01-14 2014-11-05 成都康弘药业集团股份有限公司 一种含有阿戈美拉汀的口腔粘膜或舌下给药的药物组合物
AR084865A1 (es) 2011-01-17 2013-07-10 Takeda Pharmaceutical Preparacion de desintegracion rapida, comprimido dispersable por via oral
US8426461B2 (en) 2011-01-17 2013-04-23 Takeda Pharmaceutical Company Limited Orally dispersible tablet
WO2012130837A1 (en) * 2011-03-28 2012-10-04 Ratiopharm Gmbh Solid agomelatine in non-crystalline form
FR2978916B1 (fr) * 2011-08-10 2013-07-26 Servier Lab Composition pharmaceutique solide pour administration buccale d'agomelatine
EP2562151A1 (en) * 2011-08-25 2013-02-27 Dr. Reddy's Laboratories Ltd. Processes for the preparation of agomelatine and its intermediates
JP6061924B2 (ja) 2011-10-14 2017-01-18 武田薬品工業株式会社 口腔内分散性製剤
CN103169669B (zh) * 2011-12-26 2015-06-17 中国人民解放军军事医学科学院毒物药物研究所 阿戈美拉汀包衣微丸以及可在口中分散的药物组合物
EP2872129B1 (en) 2012-07-16 2017-03-08 ratiopharm GmbH Complex of agomelatine and cyclodextrin
CN102988315B (zh) * 2012-09-28 2017-11-17 浙江华海药业股份有限公司 阿戈美拉汀固体制剂的制备方法
FR3001894A1 (fr) * 2013-02-08 2014-08-15 Servier Lab Composition pharmaceutique solide pour administration buccale d'agomelatine
PT2810656T (pt) 2013-06-06 2017-11-13 Zentiva As Formulações de agomelatina compreendendo agomelatina na forma de cocristais
EP2810647A1 (en) 2013-06-06 2014-12-10 Zentiva, a.s. Pharmaceutical formulations comprising agomelatine in the form of agomelatine co-crystal with an organic acid
CN103816129B (zh) * 2014-02-27 2020-04-28 浙江华海药业股份有限公司 阿戈美拉汀口崩片
CN104586797A (zh) * 2015-01-05 2015-05-06 万特制药(海南)有限公司 阿戈美拉汀分散片及其制备方法
CN106333929A (zh) * 2016-09-24 2017-01-18 万特制药(海南)有限公司 一种含有阿戈美拉汀的分散片及其制备方法

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3505433A1 (de) * 1985-02-16 1986-08-21 Basf Ag, 6700 Ludwigshafen Direkttablettierhilfsmittel
DE3506276C1 (de) * 1985-02-22 1986-04-24 Meggle Milchindustrie Gmbh & Co Kg, 8094 Reitmehring Direkttablettiermittel
FR2658818B1 (fr) * 1990-02-27 1993-12-31 Adir Cie Nouveaux derives a structure naphtalenique, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
FR2710265B1 (fr) * 1993-09-22 1995-10-20 Adir Composition pharmaceutique bioadhésive pour la libération contrôlée de principes actifs.
CA2179382C (en) * 1994-01-31 2009-11-10 Takao Mizumoto Intrabuccally dissolving compressed moldings and production process thereof
PL187242B1 (pl) * 1996-05-13 2004-06-30 Novartis Consumer Health Sa Policzkowy układ dostarczający
US6024981A (en) * 1997-04-16 2000-02-15 Cima Labs Inc. Rapidly dissolving robust dosage form
EP1058538B9 (en) * 1998-03-06 2013-01-02 Aptalis Pharma S.r.l. Fast disintegrating tablets
JP2000273039A (ja) * 1999-01-20 2000-10-03 Taisho Pharmaceut Co Ltd 口腔内崩壊性組成物
DE60036205T2 (de) * 2000-07-27 2008-05-21 Roquette Frères Granulat bestehend aus Stärke und Laktose
UA80393C2 (uk) * 2000-12-07 2007-09-25 Алтана Фарма Аг Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
FR2834889B1 (fr) * 2002-01-18 2004-04-02 Roquette Freres Forme pharmaceutique solide orodispersible

Also Published As

Publication number Publication date
UA77752C2 (uk) 2007-01-15
AR038207A1 (es) 2005-01-05
JP2009137994A (ja) 2009-06-25
JP4335011B2 (ja) 2009-09-30
FR2834890B1 (fr) 2004-02-27
HK1076742A1 (en) 2006-01-27
CA2473201C (fr) 2010-08-17
NO20043441L (no) 2004-08-18
EA007299B1 (ru) 2006-08-25
GEP20063818B (en) 2006-05-10
CY1105415T1 (el) 2010-04-28
WO2003061644A1 (fr) 2003-07-31
SI1467724T1 (sl) 2006-08-31
US20050131071A1 (en) 2005-06-16
KR20040075102A (ko) 2004-08-26
AU2003220786B2 (en) 2007-08-02
CN1622804A (zh) 2005-06-01
KR100605798B1 (ko) 2006-08-01
NZ533843A (en) 2005-08-26
JP2005523253A (ja) 2005-08-04
NO333712B1 (no) 2013-09-02
CN1287780C (zh) 2006-12-06
BR0307072A (pt) 2004-12-28
MXPA04007198A (es) 2004-10-29
MA27101A1 (fr) 2004-12-20
EP1467724A1 (fr) 2004-10-20
ATE324882T1 (de) 2006-06-15
DK1467724T3 (da) 2006-08-28
PL204937B1 (pl) 2010-02-26
ES2262999T3 (es) 2006-12-01
EA200400928A1 (ru) 2004-12-30
ZA200405153B (en) 2005-08-31
EP1467724B1 (fr) 2006-05-03
FR2834890A1 (fr) 2003-07-25
US20100260840A1 (en) 2010-10-14
DE60304993T2 (de) 2007-01-18
CA2473201A1 (fr) 2003-07-31
DE60304993D1 (de) 2006-06-08
BRPI0307072B1 (pt) 2017-05-02
PL370160A1 (en) 2005-05-16

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