PL377608A1 - Sposób wytwarzania proleków 3'-nukleozydowych - Google Patents

Sposób wytwarzania proleków 3'-nukleozydowych

Info

Publication number
PL377608A1
PL377608A1 PL377608A PL37760803A PL377608A1 PL 377608 A1 PL377608 A1 PL 377608A1 PL 377608 A PL377608 A PL 377608A PL 37760803 A PL37760803 A PL 37760803A PL 377608 A1 PL377608 A1 PL 377608A1
Authority
PL
Poland
Prior art keywords
production
nucleoside prodrugs
nucleoside
prodrugs
Prior art date
Application number
PL377608A
Other languages
English (en)
Inventor
Richard Storer
Adel Moussa
Steven Mathieu
Original Assignee
Idenix (Cayman) Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Idenix (Cayman) Limited filed Critical Idenix (Cayman) Limited
Publication of PL377608A1 publication Critical patent/PL377608A1/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
PL377608A 2002-12-23 2003-12-23 Sposób wytwarzania proleków 3'-nukleozydowych PL377608A1 (pl)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US43615002P 2002-12-23 2002-12-23

Publications (1)

Publication Number Publication Date
PL377608A1 true PL377608A1 (pl) 2006-02-06

Family

ID=32682350

Family Applications (1)

Application Number Title Priority Date Filing Date
PL377608A PL377608A1 (pl) 2002-12-23 2003-12-23 Sposób wytwarzania proleków 3'-nukleozydowych

Country Status (16)

Country Link
US (1) US20040181051A1 (pl)
EP (1) EP1575971A4 (pl)
JP (1) JP2006514038A (pl)
KR (1) KR20050110611A (pl)
CN (1) CN100335492C (pl)
AU (1) AU2003300434A1 (pl)
BR (1) BR0316868A (pl)
CA (1) CA2511616A1 (pl)
IL (1) IL169314A0 (pl)
MX (1) MXPA05006865A (pl)
NO (1) NO20053557L (pl)
NZ (1) NZ540913A (pl)
PL (1) PL377608A1 (pl)
RU (1) RU2005123395A (pl)
WO (1) WO2004058792A1 (pl)
ZA (1) ZA200505040B (pl)

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KR20070087624A (ko) * 2004-12-23 2007-08-28 노파르티스 아게 Ｈｃｖ 치료용 조성물
AU2006222563A1 (en) 2005-03-08 2006-09-14 Biota Scientific Management Pty Ltd. Bicyclic nucleosides and nucleotides as therapeutic agents
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WO2007113159A1 (en) 2006-04-04 2007-10-11 F. Hoffmann-La Roche Ag 3',5'-di-o-acylated nucleosides for hcv treatment
WO2010015637A1 (en) * 2008-08-06 2010-02-11 Novartis Ag New antiviral modified nucleosides
SG172359A1 (en) 2008-12-23 2011-07-28 Pharmasset Inc Nucleoside phosphoramidates
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BRPI0922508A8 (pt) 2008-12-23 2016-01-19 Pharmasset Inc Análogos de nucleosídeo
EP2385951A4 (en) * 2009-01-09 2013-05-29 Univ Cardiff PHOSPHORAMIDATE DERIVATIVES OF GUANOSINE NUCLEOSIDE COMPOUNDS FOR THE TREATMENT OF VIRAL INFECTIONS
PT2752422T (pt) 2010-03-31 2017-11-07 Gilead Pharmasset Llc Síntese estereosseletiva de princípios ativos contendo fósforo
CN116036114A (zh) 2016-09-07 2023-05-02 阿堤亚制药公司 用于rna病毒治疗的2’-取代的-n6-取代的嘌呤核苷酸
AU2019384826A1 (en) * 2018-11-25 2021-07-15 Tnt Medical Corporation Orally active prodrug of gemcitabine

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Also Published As

Publication number Publication date
CA2511616A1 (en) 2004-07-15
CN1751058A (zh) 2006-03-22
AU2003300434A1 (en) 2004-07-22
KR20050110611A (ko) 2005-11-23
JP2006514038A (ja) 2006-04-27
BR0316868A (pt) 2005-10-25
EP1575971A1 (en) 2005-09-21
MXPA05006865A (es) 2005-12-12
EP1575971A4 (en) 2008-03-05
US20040181051A1 (en) 2004-09-16
CN100335492C (zh) 2007-09-05
RU2005123395A (ru) 2006-01-27
NO20053557L (no) 2005-09-08
IL169314A0 (en) 2007-07-04
WO2004058792A1 (en) 2004-07-15
ZA200505040B (en) 2006-04-26
NZ540913A (en) 2008-02-29

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