PE20171305A1 - Formulaciones inyectables de paracetamol - Google Patents

Formulaciones inyectables de paracetamol

Info

Publication number
PE20171305A1
PE20171305A1 PE2017001066A PE2017001066A PE20171305A1 PE 20171305 A1 PE20171305 A1 PE 20171305A1 PE 2017001066 A PE2017001066 A PE 2017001066A PE 2017001066 A PE2017001066 A PE 2017001066A PE 20171305 A1 PE20171305 A1 PE 20171305A1
Authority
PE
Peru
Prior art keywords
paracetamol
formulation
alcohol
injectable formulations
flebitis
Prior art date
Application number
PE2017001066A
Other languages
English (en)
Inventor
Ketan R Patel
Milan R Patel
Asheel K Patel
Prakashchandra J Shah
Original Assignee
Troikaa Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=55022620&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PE20171305(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Troikaa Pharmaceuticals Ltd filed Critical Troikaa Pharmaceuticals Ltd
Publication of PE20171305A1 publication Critical patent/PE20171305A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/22Heterocyclic compounds, e.g. ascorbic acid, tocopherol or pyrrolidones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Dermatology (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Inorganic Chemistry (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

SE REFIERE A UNA FORMULACION INYECTABLE DE PARACETAMOL QUE COMPRENDE: A) 250 mg/ml DE PARACETAMOL O SUS SALES FARMACEUTICAMENTE ACEPTABLES; Y B) UN SISTEMA DE SOLVENTES QUE COMPRENDE i) 0-40% P/V DE GLICOFUROL, ii) 0-30% P/V DE UN ALCOHOL DE CADENA CORTA TAL COMO ALCOHOL ETILICO, ALCOHOL ISOPROPILICO O MEZCLAS DE LOS MISMOS, iii) 0-5% P/V DE UN ESTABILIZADOR, iv) 0-55% P/V DE OTRO SOLVENTE TAL COMO AGENTES TENSOACTIVOS, CICLODEXTRINAS, N-METIL-PIRROLIDONA, ENTRE OTROS, Y v) AGUA PARA COMPLETAR EL VOLUMEN DE LA FORMULACION. ADICIONALMENTE DICHA FORMULACION COMPRENDE INGREDIENTES AUXILIARES TAL COMO ANTIOXIDANTES, MODIFICADORES DE pH, ENTRE OTROS, Y SON APTAS PARA SU ADMINISTRACION POR VIA INTRAVENOSA LENTA CON EFECTOS SECUNDARIOS MINIMIZADOS TALES COMO FLEBITIS Y DOLOR
PE2017001066A 2014-12-20 2015-11-17 Formulaciones inyectables de paracetamol PE20171305A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IN4102MU2014 2014-12-20

Publications (1)

Publication Number Publication Date
PE20171305A1 true PE20171305A1 (es) 2017-09-05

Family

ID=55022620

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2017001066A PE20171305A1 (es) 2014-12-20 2015-11-17 Formulaciones inyectables de paracetamol

Country Status (28)

Country Link
US (1) US20180000940A1 (es)
EP (1) EP3233055A1 (es)
JP (1) JP2017538762A (es)
KR (1) KR20170099911A (es)
CN (1) CN107205924A (es)
AR (1) AR103188A1 (es)
AU (1) AU2015365533A1 (es)
BR (1) BR112017012975B1 (es)
CA (1) CA2969303A1 (es)
CL (1) CL2017001629A1 (es)
CO (1) CO2017006268A2 (es)
CU (1) CU20170088A7 (es)
DO (1) DOP2017000134A (es)
EA (1) EA201791409A1 (es)
EC (1) ECSP17038668A (es)
IL (1) IL252729A0 (es)
JO (1) JO3689B1 (es)
MA (1) MA40599A1 (es)
MD (1) MD20170071A2 (es)
MX (1) MX2017008264A (es)
PE (1) PE20171305A1 (es)
PH (1) PH12017501005A1 (es)
SG (1) SG11201704435PA (es)
TN (1) TN2017000232A1 (es)
TW (1) TWI649097B (es)
UA (1) UA122136C2 (es)
UY (1) UY36466A (es)
WO (1) WO2016097899A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN107229455B (zh) 2016-03-24 2019-09-17 阿里巴巴集团控股有限公司 一种业务处理方法、装置及***

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2751875B1 (fr) * 1996-08-05 1998-12-24 Scr Newpharm Nouvelles formulations liquides stables a base de paracetamol et leur mode de preparation
IT1301976B1 (it) * 1998-07-31 2000-07-20 Angelini Ricerche Spa Composizione farmaceutica iniettabile a base di paracetamolo
IT1313579B1 (it) 1999-07-30 2002-09-09 Acraf Composizione farmaceutica liquida a base di paracetamolo.
ITMI20012135A1 (it) 2001-10-16 2003-04-16 Bioren S A Soluzioni iniettabili pronte all'uso di paracetamolo
MX2007014862A (es) * 2005-05-27 2008-02-21 Panacea Biotec Ltd Composiciones inyectables y procedimiento para la preparacion de dichas composiciones.
PT1973527E (pt) * 2005-12-15 2010-01-04 Acusphere Inc Processos de produção de formulações farmacêuticas à base de partículas destinadas a administração parentérica
EP2170313A2 (en) 2007-06-18 2010-04-07 Combino Pharm, S.L. Aqueous formulations of acetaminophen for injection
WO2009098716A2 (en) 2008-01-17 2009-08-13 Aptuit Laurus Private Limited Stable pharmaceutical aqueous compositions
WO2010040652A1 (en) * 2008-10-09 2010-04-15 Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F. S.P.A. Liquid pharmaceutical formulation containing paracetamol
JP5872551B2 (ja) * 2010-06-30 2016-03-01 トロイカ ファーマスーティカルズ リミテッド パラセタモールを含む医薬組成物およびその製造法
TWI577377B (zh) * 2010-09-16 2017-04-11 Viiv醫療保健公司 醫藥組合物
CN102258485A (zh) * 2011-01-11 2011-11-30 北京润德康医药技术有限公司 一种含对乙酰氨基酚的注射用制剂及其应用
CN102600068A (zh) * 2011-01-24 2012-07-25 联康药业克雷恩特塞提斯制药实验室有限责任公司 稳定即用的可注射扑热息痛制剂

Also Published As

Publication number Publication date
CO2017006268A2 (es) 2017-10-20
IL252729A0 (en) 2017-08-31
MD20170071A2 (ro) 2017-09-30
EP3233055A1 (en) 2017-10-25
TN2017000232A1 (en) 2018-10-19
UY36466A (es) 2016-07-29
AU2015365533A1 (en) 2017-07-06
CL2017001629A1 (es) 2018-03-16
BR112017012975A2 (pt) 2018-02-27
DOP2017000134A (es) 2017-09-15
CN107205924A (zh) 2017-09-26
TWI649097B (zh) 2019-02-01
TW201622703A (zh) 2016-07-01
CA2969303A1 (en) 2016-06-23
MX2017008264A (es) 2017-10-02
UA122136C2 (uk) 2020-09-25
JO3689B1 (ar) 2020-08-27
BR112017012975B1 (pt) 2023-09-26
SG11201704435PA (en) 2017-06-29
AR103188A1 (es) 2017-04-19
EA201791409A1 (ru) 2017-10-31
MA40599A1 (fr) 2017-11-30
WO2016097899A1 (en) 2016-06-23
PH12017501005A1 (en) 2017-12-11
KR20170099911A (ko) 2017-09-01
US20180000940A1 (en) 2018-01-04
ECSP17038668A (es) 2017-12-01
JP2017538762A (ja) 2017-12-28
CU20170088A7 (es) 2018-03-13

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