PA8653801A1 - DERIVATIVES OF OCTAHIDROPIRROLO [3,4-C] PIRROL - Google Patents
DERIVATIVES OF OCTAHIDROPIRROLO [3,4-C] PIRROLInfo
- Publication number
- PA8653801A1 PA8653801A1 PA20058653801A PA8653801A PA8653801A1 PA 8653801 A1 PA8653801 A1 PA 8653801A1 PA 20058653801 A PA20058653801 A PA 20058653801A PA 8653801 A PA8653801 A PA 8653801A PA 8653801 A1 PA8653801 A1 PA 8653801A1
- Authority
- PA
- Panama
- Prior art keywords
- pirrol
- derivatives
- octahidropirrolo
- octahydropirrolo
- procedures
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Abstract
LA PRESENTE INVENCION SE REFIERE A DERIVADOS DE OCTAHIDROPIRROLO [3,4-C]PIRROL DE FORMULA (I): Y A PROCEDIMIENTOS PARA SU PREPARACION, A COMPOSICIONES QUE LOS CONTIENEN Y A SUS USOS.THIS INVENTION REFERS TO OCTAHYDROPIRROLO DERIVATIVES [3,4-C] FORMULA PIRROL (I): AND TO PROCEDURES FOR THEIR PREPARATION, TO COMPOSITIONS THAT CONTAIN THEM AND THEIR USES.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP04106044A EP1671972A1 (en) | 2004-11-24 | 2004-11-24 | Octahydropyrrolo[3,4-c]pyrrole derivatives |
EP05100474 | 2005-01-26 |
Publications (1)
Publication Number | Publication Date |
---|---|
PA8653801A1 true PA8653801A1 (en) | 2006-06-02 |
Family
ID=35985757
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PA20058653801A PA8653801A1 (en) | 2004-11-24 | 2005-11-24 | DERIVATIVES OF OCTAHIDROPIRROLO [3,4-C] PIRROL |
Country Status (12)
Country | Link |
---|---|
EP (1) | EP1846409A1 (en) |
JP (1) | JP2008520644A (en) |
AR (1) | AR054707A1 (en) |
CA (1) | CA2587141A1 (en) |
GT (1) | GT200500340A (en) |
NL (1) | NL1030503C2 (en) |
PA (1) | PA8653801A1 (en) |
PE (1) | PE20061055A1 (en) |
SV (1) | SV2007002315A (en) |
TW (1) | TW200626600A (en) |
UY (1) | UY29221A1 (en) |
WO (1) | WO2006056848A1 (en) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2008083124A1 (en) | 2006-12-28 | 2008-07-10 | Rigel Pharmaceuticals, Inc. | N-substituted-heterocycloalkyloxybenzamide compounds and methods of use |
EP2201982A1 (en) | 2008-12-24 | 2010-06-30 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Histamine H4 receptor antagonists for the treatment of vestibular disorders |
JPWO2011013752A1 (en) * | 2009-07-31 | 2013-01-10 | 塩野義製薬株式会社 | Pharmaceutical composition containing a fused heterocyclic derivative |
WO2011050202A1 (en) | 2009-10-23 | 2011-04-28 | Janssen Pharmaceutica Nv | Fused heterocyclic compounds as orexin receptor modulators |
CN102781942B (en) | 2009-10-23 | 2015-09-23 | 詹森药业有限公司 | Octahydro pyrrolo-[3,4-c] pyrroles is replaced as two of orexin receptor modulators |
EP2491034B1 (en) | 2009-10-23 | 2013-12-18 | Janssen Pharmaceutica, N.V. | Fused heterocyclic compounds as orexin receptor modulators |
WO2012145581A1 (en) | 2011-04-20 | 2012-10-26 | Janssen Pharmaceutica Nv | Disubstituted octahy-dropyrrolo [3,4-c] pyrroles as orexin receptor modulators |
SI2858647T1 (en) | 2012-06-08 | 2018-11-30 | Sensorion | H4 receptor inhibitors for treating tinnitus |
CN108883110B (en) | 2016-03-10 | 2022-05-27 | 詹森药业有限公司 | Methods of treating depression using orexin-2 receptor antagonists |
WO2019152883A1 (en) * | 2018-02-02 | 2019-08-08 | Padforward Llc | Inhibitors of protein arginine deiminases |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2620341A (en) * | 1949-03-24 | 1952-12-02 | Burroughs Wellcome Co | N,n-dialkyl-quinoline-4-carboxamidines |
ES2162047T3 (en) * | 1995-05-11 | 2001-12-16 | Upjohn Co | OXAZOLIDINONES WITH REST DIAZINYL AND CARBAZINYL SPIROCICLICAL AND BICYCLE. |
GB9902453D0 (en) * | 1999-02-05 | 1999-03-24 | Zeneca Ltd | Chemical compounds |
CA2440803A1 (en) * | 2001-03-07 | 2002-09-12 | Pfizer Products Inc. | Modulators of chemokine receptor activity |
WO2002072548A2 (en) * | 2001-03-09 | 2002-09-19 | Ortho-Mcneil Pharmaceutical, Inc. | Heterocyclic compounds and their use as histamine h4 ligands. |
CA2497788A1 (en) * | 2002-09-06 | 2004-03-18 | Janssen Pharmaceutica, N.V. | Use of histamine h4 receptor modulators for the treatment of allergy and asthma |
EP1543011B1 (en) * | 2002-09-06 | 2006-05-03 | Janssen Pharmaceutica N.V. | Thienopyrrolyl and furanopyrrolyl compounds and their use as histamine h4 receptor ligands |
RU2005106274A (en) * | 2002-09-06 | 2005-11-10 | Янссен Фармацевтика, Н.В. (Be) | HETEROCYCLIC COMPOUNDS |
-
2005
- 2005-11-10 EP EP05824102A patent/EP1846409A1/en not_active Withdrawn
- 2005-11-10 JP JP2007542155A patent/JP2008520644A/en active Pending
- 2005-11-10 WO PCT/IB2005/003478 patent/WO2006056848A1/en active Application Filing
- 2005-11-10 CA CA002587141A patent/CA2587141A1/en not_active Abandoned
- 2005-11-21 UY UY29221A patent/UY29221A1/en not_active Application Discontinuation
- 2005-11-21 PE PE2005001360A patent/PE20061055A1/en not_active Application Discontinuation
- 2005-11-22 AR ARP050104891A patent/AR054707A1/en unknown
- 2005-11-23 NL NL1030503A patent/NL1030503C2/en not_active IP Right Cessation
- 2005-11-23 TW TW094141134A patent/TW200626600A/en unknown
- 2005-11-23 GT GT200500340A patent/GT200500340A/en unknown
- 2005-11-24 SV SV2005002315A patent/SV2007002315A/en not_active Application Discontinuation
- 2005-11-24 PA PA20058653801A patent/PA8653801A1/en unknown
Also Published As
Publication number | Publication date |
---|---|
AR054707A1 (en) | 2007-07-11 |
SV2007002315A (en) | 2007-02-16 |
PE20061055A1 (en) | 2006-11-09 |
WO2006056848A1 (en) | 2006-06-01 |
GT200500340A (en) | 2006-07-13 |
NL1030503A1 (en) | 2006-05-29 |
EP1846409A1 (en) | 2007-10-24 |
UY29221A1 (en) | 2006-06-30 |
TW200626600A (en) | 2006-08-01 |
NL1030503C2 (en) | 2006-11-28 |
CA2587141A1 (en) | 2006-06-01 |
JP2008520644A (en) | 2008-06-19 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
PA8653801A1 (en) | DERIVATIVES OF OCTAHIDROPIRROLO [3,4-C] PIRROL | |
UY29886A1 (en) | NEW PIRAZOL DERIVATIVES, PHARMACCUTIC COMPOSITIONS CONTAINING THEM, PROCEDURES FOR THE PREPARATION OF THE SAME AND APPLICATIONS | |
HN1999000106A (en) | HETERO-CYCLE COMPOUNDS AS ROTAMASE ENZYME INHIBITORS. | |
PA8570901A1 (en) | DERIVATIVES OF ACIL-4-CARBOXIFENILUREA, PROCEDURES FOR PREPARATION AND USE | |
CR9954A (en) | PIRAZINE DERIVATIVES | |
CR11106A (en) | KINASE INHIBITORS P710 S6 | |
CR8649A (en) | FORMAMIDINE DERIVATIVES FOR THE TREATMENT OF DISEASES | |
UY29360A1 (en) | NEW DERIVATIVES OF PIRAZOL, PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM, PREPARATION PROCEDURES AND APPLICATIONS. | |
UY31481A1 (en) | NEW PIRIMIDINE DERIVATIVES, PREPARATION PROCESSES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND APPLICATIONS | |
HN2003000064A (en) | USEFUL NICOTINAMIDE DERIVATIVES AS PDE4 INHIBITORS | |
UY30195A1 (en) | DERIVATIVES OF PHENETANOLAMINE, PREPARATION PROCEDURE, COMPOSITIONS CONTAINING THEM AND APPLICATIONS | |
CR10149A (en) | CYTOTOXIC AGENTS UNDERSTANDING NEW TOMAIMYCIN DERIVATIVES AND THERAPEUTIC USE | |
CU20090072A7 (en) | L-GLUTAMIC ACID MARKED WITH [F-18], L-GLUTAMINE MARKED WITH [F-18], ITS DERIVATIVES AND ITS USE, AS WELL AS PROCEDURES FOR PREPARATION | |
CR11661A (en) | FUSIONED HETEROCICLIC DERIVATIVE AND ITS USE | |
HN2003000062A (en) | USEFUL NICOTINAMIDE DERIVATIVES AS PDE4 INHIBITORS | |
HN2008001393A (en) | DERIVATIVES OF 1,2,4,5- TETRAHIDRO -3H- BENZAZEPINAS, ITS PREPARATION PROCEDURE AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM | |
GT200600117A (en) | NEW PHARMACEUTICAL COMPOUNDS | |
UY31048A1 (en) | NEW PIRIMIDINE COMPOUNDS AND USES OF THE SAME | |
PA8660401A1 (en) | TRIAZOL DERIVATIVES REPLACED AS AN OXITOCINE ANTAGONISTS | |
GT200600144A (en) | 1H-QUINAZOLIN-2,4-DIONAS | |
CU23415B7 (en) | DERIVATIVES OF 2,6- QUINOLINILO AND 2,6- NAFTILO, PROCESSES FOR THEIR PREPARATION AND ITS USES | |
CR8205A (en) | USEFUL NICOTINAMIDE DERIVATIVES AS PDE4 INHIBITORS | |
CR7956A (en) | INTERMEDIATE ANTIBACTERIAL INDOLONA OXAZOLIDINONES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME | |
SV2006002319A (en) | REPLACED INDOLES, COMPOSITIONS THAT CONTAIN THEM, MANUFACTURING PROCEDURE AND USE | |
PA8614201A1 (en) | DERIVATIVES OF DISULFIDE, SULFIDE, SULFOXIDE AND SULPHONE OF CYCLING SUGARS AND THEIR USES |