PA8624401A1 - Procesos para la preparacion de haluros de aril- y heteroaril-alquilsulfonilo - Google Patents
Procesos para la preparacion de haluros de aril- y heteroaril-alquilsulfoniloInfo
- Publication number
- PA8624401A1 PA8624401A1 PA20058624401A PA8624401A PA8624401A1 PA 8624401 A1 PA8624401 A1 PA 8624401A1 PA 20058624401 A PA20058624401 A PA 20058624401A PA 8624401 A PA8624401 A PA 8624401A PA 8624401 A1 PA8624401 A1 PA 8624401A1
- Authority
- PA
- Panama
- Prior art keywords
- halures
- preparation
- processes
- alquilsulfonilo
- heteroaril
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- 239000000825 pharmaceutical preparation Substances 0.000 abstract 1
- 229940127557 pharmaceutical product Drugs 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/32—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of salts of sulfonic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/02—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof
- C07C303/22—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof from sulfonic acids, by reactions not involving the formation of sulfo or halosulfonyl groups; from sulfonic halides by reactions not involving the formation of halosulfonyl groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
LA PRESENTE INVENCION PROVEE PROCESOS PARA LA PREPARACION DE HALUROS DE ARILALQUILSULFONILO Y HALUROS DE HETEROARILALQUILSUFONILO DE FORMULA I: AR-R-SO2-X, LOS CUALES SON UTILES COMO INTERMEDIARIOS EN LA PREPARACION DE PRODUCTOS FARMACEUTICOS.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US54760004P | 2004-02-25 | 2004-02-25 |
Publications (1)
Publication Number | Publication Date |
---|---|
PA8624401A1 true PA8624401A1 (es) | 2006-08-03 |
Family
ID=34910921
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PA20058624401A PA8624401A1 (es) | 2004-02-25 | 2005-02-23 | Procesos para la preparacion de haluros de aril- y heteroaril-alquilsulfonilo |
Country Status (24)
Country | Link |
---|---|
US (1) | US7321061B2 (es) |
EP (1) | EP1718605B1 (es) |
JP (1) | JP2007523954A (es) |
CN (1) | CN1922136A (es) |
AR (1) | AR048239A1 (es) |
AT (1) | ATE433955T1 (es) |
AU (1) | AU2005217619A1 (es) |
BR (1) | BRPI0507979A (es) |
CA (1) | CA2555247A1 (es) |
CO (1) | CO5720992A2 (es) |
CR (1) | CR8550A (es) |
DE (1) | DE602005014942D1 (es) |
EC (1) | ECSP066797A (es) |
ES (1) | ES2326746T3 (es) |
GT (1) | GT200500031A (es) |
IL (1) | IL177432A0 (es) |
NO (1) | NO20063611L (es) |
PA (1) | PA8624401A1 (es) |
PE (1) | PE20060018A1 (es) |
RU (1) | RU2006129650A (es) |
SV (1) | SV2005002015A (es) |
TW (1) | TW200602298A (es) |
WO (1) | WO2005082843A1 (es) |
ZA (1) | ZA200607097B (es) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1907355B1 (en) * | 2005-07-21 | 2015-08-05 | Ziarco Pharma Ltd | Process for the synthesis of sulfonyl halides and sulfonamides from sulfonic acid salts |
JP2010508302A (ja) * | 2006-10-31 | 2010-03-18 | ワイス エルエルシー | ホスホリパーゼ酵素の阻害剤の液剤 |
JP2010508304A (ja) * | 2006-10-31 | 2010-03-18 | ワイス エルエルシー | ホスホリパーゼ酵素阻害剤の半固体製剤 |
US20120116121A1 (en) * | 2009-07-30 | 2012-05-10 | Dow Global Technologies Llc | Process for the sulfochlorination of hydrocarbons |
CN102241613B (zh) * | 2011-05-09 | 2013-06-05 | 南通维立科化工有限公司 | 甲基磺酸钠制备高纯度甲基磺酰氯的生产方法 |
CN102295587A (zh) * | 2011-05-26 | 2011-12-28 | 安徽丰乐农化有限责任公司 | 对甲基苯磺酰氯的制备新工艺 |
CN102976988B (zh) * | 2012-12-24 | 2014-06-18 | 三门峡奥科化工有限公司 | 2-萘硫酚的合成工艺 |
KR102122111B1 (ko) * | 2017-09-01 | 2020-06-11 | 주식회사 엘지화학 | 대체 용매의 선정 방법 |
CN111718286A (zh) * | 2020-07-23 | 2020-09-29 | 邓博天 | 一种带供电基团芳烃磺酰氯的工业化生产方法 |
Family Cites Families (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE48722C (de) | Dr. E. FISCHER in Stuttgart, Schlofsstrafse 29 | Verfahren zur Darstellung von O-Nitrobenzaldehyd aus O-Nitrobenzylchlorid | ||
DE150313C (es) | ||||
US2199568A (en) | 1938-06-11 | 1940-05-07 | Gen Aniline & Film Corp | Manufacture of 1-methyl-4-chloro-5-hydroxynaphthalene-11-sulphonic acid |
US2507408A (en) | 1948-03-05 | 1950-05-09 | Rhone Poulenc Sa | 1-alkylsulfonyl-4-alkyl piperazines |
US2888486A (en) | 1953-11-20 | 1959-05-26 | Du Pont | Process for producing aromatic sulfonyl halides |
DE2545644A1 (de) * | 1975-10-11 | 1977-04-14 | Bayer Ag | Verfahren zur herstellung von sulfonsaeuren |
US4150049A (en) * | 1975-11-05 | 1979-04-17 | The Government Of The United States | Esters of aromatic sulfonic acids |
JPS5277030A (en) * | 1975-12-23 | 1977-06-29 | Toyo Pharma Kk | Production of novel benzyl sulphonic acid derivatives |
JPH09295962A (ja) * | 1996-03-08 | 1997-11-18 | Nagase & Co Ltd | 2,2−ジ置換−エタンスルホン酸誘導体およびその塩 |
DE19838516A1 (de) * | 1998-08-25 | 2000-03-09 | Degussa | Verfahren zur Herstellung von Sulfonylhalogeniden |
JP2000072739A (ja) * | 1998-09-01 | 2000-03-07 | Tanabe Seiyaku Co Ltd | スルホン酸類またはその塩の製法 |
PT1451154E (pt) | 2001-12-03 | 2008-04-21 | Wyeth Corp | Inibidores de fosfolipase a2 citossólica |
EP1907355B1 (en) | 2005-07-21 | 2015-08-05 | Ziarco Pharma Ltd | Process for the synthesis of sulfonyl halides and sulfonamides from sulfonic acid salts |
-
2005
- 2005-02-22 AR ARP050100642A patent/AR048239A1/es not_active Application Discontinuation
- 2005-02-23 PE PE2005000213A patent/PE20060018A1/es not_active Application Discontinuation
- 2005-02-23 AT AT05713940T patent/ATE433955T1/de not_active IP Right Cessation
- 2005-02-23 DE DE602005014942T patent/DE602005014942D1/de active Active
- 2005-02-23 CN CNA2005800058622A patent/CN1922136A/zh active Pending
- 2005-02-23 RU RU2006129650/04A patent/RU2006129650A/ru not_active Application Discontinuation
- 2005-02-23 US US11/064,241 patent/US7321061B2/en not_active Expired - Fee Related
- 2005-02-23 JP JP2007500927A patent/JP2007523954A/ja active Pending
- 2005-02-23 SV SV2005002015A patent/SV2005002015A/es not_active Application Discontinuation
- 2005-02-23 PA PA20058624401A patent/PA8624401A1/es unknown
- 2005-02-23 TW TW094105341A patent/TW200602298A/zh unknown
- 2005-02-23 GT GT200500031A patent/GT200500031A/es unknown
- 2005-02-23 AU AU2005217619A patent/AU2005217619A1/en not_active Abandoned
- 2005-02-23 CA CA002555247A patent/CA2555247A1/en not_active Abandoned
- 2005-02-23 BR BRPI0507979-9A patent/BRPI0507979A/pt not_active IP Right Cessation
- 2005-02-23 ES ES05713940T patent/ES2326746T3/es active Active
- 2005-02-23 WO PCT/US2005/005624 patent/WO2005082843A1/en active Application Filing
- 2005-02-23 EP EP05713940A patent/EP1718605B1/en active Active
-
2006
- 2006-08-08 CR CR8550A patent/CR8550A/es not_active Application Discontinuation
- 2006-08-09 NO NO20063611A patent/NO20063611L/no not_active Application Discontinuation
- 2006-08-10 IL IL177432A patent/IL177432A0/en unknown
- 2006-08-23 CO CO06083312A patent/CO5720992A2/es not_active Application Discontinuation
- 2006-08-24 ZA ZA200607097A patent/ZA200607097B/xx unknown
- 2006-08-25 EC EC2006006797A patent/ECSP066797A/es unknown
Also Published As
Publication number | Publication date |
---|---|
JP2007523954A (ja) | 2007-08-23 |
WO2005082843A1 (en) | 2005-09-09 |
CR8550A (es) | 2007-02-05 |
AU2005217619A1 (en) | 2005-09-09 |
EP1718605B1 (en) | 2009-06-17 |
EP1718605A1 (en) | 2006-11-08 |
BRPI0507979A (pt) | 2007-07-24 |
CN1922136A (zh) | 2007-02-28 |
SV2005002015A (es) | 2005-11-04 |
PE20060018A1 (es) | 2006-02-20 |
ZA200607097B (en) | 2009-08-26 |
CO5720992A2 (es) | 2007-01-31 |
US7321061B2 (en) | 2008-01-22 |
IL177432A0 (en) | 2006-12-10 |
GT200500031A (es) | 2005-09-30 |
TW200602298A (en) | 2006-01-16 |
CA2555247A1 (en) | 2005-09-09 |
ECSP066797A (es) | 2006-11-16 |
AR048239A1 (es) | 2006-04-12 |
ATE433955T1 (de) | 2009-07-15 |
DE602005014942D1 (de) | 2009-07-30 |
ES2326746T3 (es) | 2009-10-19 |
US20050187408A1 (en) | 2005-08-25 |
RU2006129650A (ru) | 2008-03-27 |
NO20063611L (no) | 2006-09-21 |
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