PA8484301A1 - Formulaciones farmaceuticas de liberacion controlada - Google Patents

Formulaciones farmaceuticas de liberacion controlada

Info

Publication number
PA8484301A1
PA8484301A1 PA19998484301A PA8484301A PA8484301A1 PA 8484301 A1 PA8484301 A1 PA 8484301A1 PA 19998484301 A PA19998484301 A PA 19998484301A PA 8484301 A PA8484301 A PA 8484301A PA 8484301 A1 PA8484301 A1 PA 8484301A1
Authority
PA
Panama
Prior art keywords
pharmaceutical formulations
controlled liberation
liberation
controlled
formulations
Prior art date
Application number
PA19998484301A
Other languages
English (en)
Inventor
Elizabeth King
Ross James Macrae
Original Assignee
Warner Lambert Exp Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27269526&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PA8484301(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB9823192.1A external-priority patent/GB9823192D0/en
Priority claimed from GBGB9825117.6A external-priority patent/GB9825117D0/en
Priority claimed from GBGB9826392.4A external-priority patent/GB9826392D0/en
Application filed by Warner Lambert Exp Ltd filed Critical Warner Lambert Exp Ltd
Publication of PA8484301A1 publication Critical patent/PA8484301A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846Poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Gynecology & Obstetrics (AREA)
  • Neurology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

LA INVENCION PROPORCIONA FORMULACIONES FARMACEUTICAS DE LIBERACION CONTROLADA PARA ADMINISTRACION ORAL QUE CONTIENEN UN INHIBIDOR GMPC PDE-5. LAS FORMULACIONES SON UTILES, ENTRE OTROS, EN EL TRATAMIENTO O PREVENCION DE LA DISFUNCION SEXUAL.
PA19998484301A 1998-10-23 1999-10-18 Formulaciones farmaceuticas de liberacion controlada PA8484301A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9823192.1A GB9823192D0 (en) 1998-10-23 1998-10-23 Pharmaceutical formulations
GBGB9825117.6A GB9825117D0 (en) 1998-11-16 1998-11-16 Pharmaceutical formulations
GBGB9826392.4A GB9826392D0 (en) 1998-11-27 1998-11-27 Pharmaceutical formulations

Publications (1)

Publication Number Publication Date
PA8484301A1 true PA8484301A1 (es) 2000-09-29

Family

ID=27269526

Family Applications (1)

Application Number Title Priority Date Filing Date
PA19998484301A PA8484301A1 (es) 1998-10-23 1999-10-18 Formulaciones farmaceuticas de liberacion controlada

Country Status (44)

Country Link
US (1) US6964780B1 (es)
EP (1) EP1123088B1 (es)
JP (1) JP2002528408A (es)
KR (1) KR20010075659A (es)
CN (1) CN1324233A (es)
AP (1) AP2001002125A0 (es)
AT (1) ATE340562T1 (es)
AU (1) AU756509B2 (es)
BG (1) BG65323B1 (es)
BR (1) BR9914718A (es)
CA (1) CA2348086C (es)
CO (1) CO5160262A1 (es)
CR (1) CR6326A (es)
CY (1) CY1106239T1 (es)
CZ (1) CZ20011427A3 (es)
DE (1) DE69933383T2 (es)
DK (1) DK1123088T3 (es)
DZ (1) DZ2923A1 (es)
EA (1) EA004068B1 (es)
EE (1) EE200100235A (es)
ES (1) ES2272082T3 (es)
GT (1) GT199900184A (es)
HK (1) HK1041818A1 (es)
HR (1) HRP20010285A2 (es)
HU (1) HUP0104318A3 (es)
ID (1) ID28232A (es)
IL (1) IL141764A (es)
IS (1) IS5865A (es)
MA (1) MA26700A1 (es)
MX (1) MXPA01004011A (es)
MY (1) MY130727A (es)
NO (1) NO20011933L (es)
NZ (1) NZ510275A (es)
OA (1) OA11664A (es)
PA (1) PA8484301A1 (es)
PE (1) PE20001286A1 (es)
PL (1) PL195789B1 (es)
PT (1) PT1123088E (es)
SK (1) SK286473B6 (es)
TR (1) TR200101103T2 (es)
TW (1) TW577756B (es)
UA (1) UA67802C2 (es)
UY (1) UY25765A1 (es)
WO (1) WO2000024383A1 (es)

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WO2000025752A1 (en) 1998-11-02 2000-05-11 Church, Marla, J. Multiparticulate modified release composition
US10179130B2 (en) 1999-10-29 2019-01-15 Purdue Pharma L.P. Controlled release hydrocodone formulations
BRPI0015284B8 (pt) 1999-10-29 2021-05-25 Euro Celtique S/A formulações de hidrocodona de liberação controlada
KR100610131B1 (ko) * 2000-09-06 2006-08-09 다나베 세이야꾸 가부시키가이샤 경구 투여용 제제
KR101045144B1 (ko) 2000-10-30 2011-06-30 유로-셀티크 소시에떼 아노뉨 서방성 하이드로코돈 제형
US7927623B2 (en) 2001-02-15 2011-04-19 Mitsubishi Tanabe Pharma Corporation Tablets quickly disintegrated in oral cavity
UA78974C2 (en) 2001-10-20 2007-05-10 Boehringer Ingelheim Pharma Use of flibanserin for treating disorders of sexual desire
US10675280B2 (en) 2001-10-20 2020-06-09 Sprout Pharmaceuticals, Inc. Treating sexual desire disorders with flibanserin
ITMI20020515A1 (it) * 2002-03-12 2003-09-12 Jagotec Ag Sistema per il rilasco controllato di uno o piu' principi attivi
GB0318824D0 (en) * 2003-08-11 2003-09-10 Glaxo Group Ltd Novel composition
MXPA06013133A (es) 2004-05-11 2007-05-23 Emotional Brain Bv Formulaciones farmaceuticas y usos de las mismas en el tratamiento de la disfuncion sexual femenina.
DE102004023069A1 (de) * 2004-05-11 2005-12-08 Bayer Healthcare Ag Neue Darreichungsformen des PDE 5-Inhibitors Vardenafil
GB0421121D0 (en) * 2004-09-22 2004-10-27 Natrocell Technologies Ltd Composite rodenticide
DE102005001989A1 (de) * 2005-01-15 2006-07-20 Bayer Healthcare Ag Intravenöse Formulierungen von PDE-Inhibitoren
DE102005009240A1 (de) 2005-03-01 2006-09-07 Bayer Healthcare Ag Arzneiformen mit verbesserten pharmakokinetischen Eigenschaften
DE102005009241A1 (de) * 2005-03-01 2006-09-07 Bayer Healthcare Ag Arzneiformen mit kontrollierter Bioverfügbarkeit
CA2613617A1 (en) * 2005-06-27 2007-01-04 Daniel Drai Compositions and methods for enhancement of sexual function
PL1912650T3 (pl) 2005-08-03 2018-01-31 Sprout Pharmaceuticals Inc Zastosowanie flibanseryny w leczeniu otyłości
BRPI0616633A2 (pt) * 2005-09-29 2011-06-28 Bayer Healthcare Ag inibidores de pde e combinações dos mesmos para o tratamento de transtornos urológicos
WO2007048803A1 (en) 2005-10-29 2007-05-03 Boehringer Ingelheim International Gmbh Benzimidazolone derivatives for the treatment of premenstrual and other female sexual disorders
EP1790343A1 (en) 2005-11-11 2007-05-30 Emotional Brain B.V. Pharmaceuticals formulations and uses thereof in the treatment of female sexual dysfunction
US20090312242A1 (en) 2006-06-30 2009-12-17 Ramiro Castro Flibanserin for the treatment of urinary incontinence and related diseases
AR062320A1 (es) 2006-08-14 2008-10-29 Boehringer Ingelheim Int Formulaciones de flibanserina y metodo para fabricarlas
CN104721168A (zh) 2006-08-25 2015-06-24 贝林格尔·英格海姆国际有限公司 控制释放***及其制造方法
EP1925307A1 (en) * 2006-11-03 2008-05-28 Emotional Brain B.V. Use of 3-alpha-androstanediol in the treatment of sexual dysfunction
US20080226715A1 (en) * 2007-03-16 2008-09-18 Albert Cha Therapeutic compositions and methods
JP2010532319A (ja) * 2007-06-13 2010-10-07 バイエル・シェーリング・ファルマ・アクチェンゲゼルシャフト 聴覚障害の処置用のpde阻害剤
UY31335A1 (es) 2007-09-12 2009-04-30 Tratamiento de sintomas vasomotores
WO2009098697A1 (en) * 2008-02-08 2009-08-13 Dexxon Ltd. Modafinil and sildenafil dosage forms
WO2010067140A1 (es) * 2008-12-12 2010-06-17 Siegfried Rhein S.A. De C.V. Composicion de liberacion pulsatil de sildenafil y proceso para prepararla
KR101004205B1 (ko) * 2008-12-17 2010-12-24 동아제약주식회사 유데나필 함유 서방성 제제를 제조하기 위한 제어방출 조성물
EA015250B9 (ru) * 2010-11-19 2013-10-30 Тева Фармасьютикал Индастриз, Лтд. Таблетка силденафила, обеспечивающая модифицированную фармакокинетику, и способ ее изготовления
BR112013029199B1 (pt) 2011-05-13 2022-02-08 Eb Ip Hybritabs B.V. Dispositivo de distribuição de dois fármacos
US20140328911A1 (en) * 2011-07-22 2014-11-06 Pom Wonderful. Llc Compositions comprising pomegranate polyphenols in combination with erectile dysfunction-treating compounds, and methods of treating erectile dysfunction therewith
WO2017168174A1 (en) * 2016-04-02 2017-10-05 N4 Pharma Uk Limited New pharmaceutical forms of sildenafil
CN113995727B (zh) * 2021-11-08 2023-04-07 山东鲁抗医药股份有限公司 一种5型磷酸二酯酶抑制剂片剂及其制备方法

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Also Published As

Publication number Publication date
NO20011933L (no) 2001-06-25
CZ20011427A3 (cs) 2001-10-17
GT199900184A (es) 2001-04-14
SK286473B6 (sk) 2008-11-06
CA2348086C (en) 2007-01-23
HRP20010285A2 (en) 2002-06-30
HK1041818A1 (zh) 2002-07-26
ID28232A (id) 2001-05-10
UY25765A1 (es) 2001-08-27
UA67802C2 (uk) 2004-07-15
DE69933383T2 (de) 2007-02-01
EA200100298A1 (ru) 2001-08-27
IL141764A (en) 2008-06-05
MXPA01004011A (es) 2003-03-10
CN1324233A (zh) 2001-11-28
PL195789B1 (pl) 2007-10-31
KR20010075659A (ko) 2001-08-09
WO2000024383A1 (en) 2000-05-04
NZ510275A (en) 2003-07-25
MA26700A1 (fr) 2004-12-20
CY1106239T1 (el) 2011-06-08
ES2272082T3 (es) 2007-04-16
BG65323B1 (bg) 2008-02-29
BR9914718A (pt) 2001-07-10
TR200101103T2 (tr) 2001-09-21
US6964780B1 (en) 2005-11-15
SK5192001A3 (en) 2002-09-10
PE20001286A1 (es) 2000-11-22
IL141764A0 (en) 2002-03-10
AU5878799A (en) 2000-05-15
OA11664A (en) 2005-01-07
HUP0104318A3 (en) 2003-12-29
JP2002528408A (ja) 2002-09-03
CA2348086A1 (en) 2000-05-04
DZ2923A1 (fr) 2004-03-01
NO20011933D0 (no) 2001-04-19
CO5160262A1 (es) 2002-05-30
DE69933383D1 (de) 2006-11-09
EP1123088B1 (en) 2006-09-27
ATE340562T1 (de) 2006-10-15
DK1123088T3 (da) 2007-01-02
AP2001002125A0 (en) 2001-04-04
EA004068B1 (ru) 2003-12-25
MY130727A (en) 2007-07-31
PT1123088E (pt) 2007-01-31
AU756509B2 (en) 2003-01-16
EE200100235A (et) 2002-08-15
TW577756B (en) 2004-03-01
PL347476A1 (en) 2002-04-08
IS5865A (is) 2001-02-27
BG105465A (bg) 2001-12-29
CR6326A (es) 2004-02-23
EP1123088A1 (en) 2001-08-16
HUP0104318A2 (hu) 2002-03-28

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