OA12801A - Process for preparing acid salts of gemifloxacin. - Google Patents

Process for preparing acid salts of gemifloxacin. Download PDF

Info

Publication number: OA12801A
Authority: OA; OAPI
Prior art keywords: acid; formula; compound; reaction; température
Prior art date: 2002-04-08

Application number

OA1200400271A

Other languages

English (en)

Inventor

Hoon Choi

Sang-Chul Choi

Bo-Seung Choi

Do-Hyun Nam

Original Assignee

Lg Life Sciences Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-04-08

Filing date

2003-04-04

Publication date

2006-07-11

2003-04-04 Application filed by Lg Life Sciences Ltd filed Critical Lg Life Sciences Ltd

2006-07-11 Publication of OA12801A publication Critical patent/OA12801A/en

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)

OA1200400271A 2002-04-08 2003-04-04 Process for preparing acid salts of gemifloxacin. OA12801A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
KR10-2002-0018847A KR100517638B1 (ko)	2002-04-08	2002-04-08	게미플록사신 산염의 새로운 제조방법

Publications (1)

Publication Number	Publication Date
OA12801A true OA12801A (en)	2006-07-11

Family

ID=36241771

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
OA1200400271A OA12801A (en)	2002-04-08	2003-04-04	Process for preparing acid salts of gemifloxacin.

Country Status (32)

Country	Link
US (1)	US7361762B2 (is)
EP (1)	EP1497290B1 (is)
JP (1)	JP4315815B2 (is)
KR (1)	KR100517638B1 (is)
CN (1)	CN1291987C (is)
AP (1)	AP1786A (is)
AT (1)	ATE404559T1 (is)
AU (1)	AU2003219581B2 (is)
BR (1)	BRPI0309037B8 (is)
CA (1)	CA2481217C (is)
CO (1)	CO5611198A2 (is)
CY (1)	CY1108469T1 (is)
DE (1)	DE60322872D1 (is)
DK (1)	DK1497290T3 (is)
EA (1)	EA007222B1 (is)
ES (1)	ES2311694T3 (is)
GE (1)	GEP20074025B (is)
HK (1)	HK1074440A1 (is)
HR (1)	HRP20040929B1 (is)
IL (1)	IL164328A (is)
IS (1)	IS2731B (is)
MA (1)	MA26408A1 (is)
MX (1)	MXPA04009777A (is)
NO (1)	NO330042B1 (is)
NZ (1)	NZ536174A (is)
OA (1)	OA12801A (is)
PL (1)	PL372815A1 (is)
PT (1)	PT1497290E (is)
SI (1)	SI1497290T1 (is)
UA (1)	UA77070C2 (is)
WO (1)	WO2003087100A1 (is)
ZA (1)	ZA200408088B (is)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US7199242B2 (en) *	2001-08-02	2007-04-03	Lg Life Sciences Limited	Processes for the production of amino-protected derivatives of 4-aminomethylene-pyrrolidin-3-one and/or 4-aminomethylene-pyrrolidin-3-alkoxyimino derivatives and/or gemifloxacin or a salt thereof
WO2006134431A1 (en) *	2005-05-03	2006-12-21	Ranbaxy Laboratories Limited	Formate salt of gemifloxacin
EP2161269A1 (en) *	2005-06-15	2010-03-10	Hetero Drugs Limited	Process for the preparation of amorphous gemifloxacin
NZ570865A (en) *	2006-03-07	2010-11-26	Wockhardt Ltd	Alanine and valine prodrugs of nadifloxacin, S-(-)-9-fluoro-6,7-dihydro-8-(4-hydroxypiperidin-1-yl)-5-methyl-1-oxo-1H,5H-benzo[i,j]quinolizine-2-carboxylic acid
US20100076193A1 (en) *	2006-10-31	2010-03-25	Chandrasekaran Ramasubbu	process for the preparation of gemifloxacin

Family Cites Families (27)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS57134482A (en)	1981-02-13	1982-08-19	Dainippon Pharmaceut Co Ltd	1-ethyl-6-fluoro-1,4-dihydro-4-oxo-7-(1-piperazinyl)-1,8- naphthyridine-3-carboxylic acid-3/2 hydrate and its preparation
IN162769B (is)	1984-11-13	1988-07-09	Kyorin Seiyaku Kk
NZ222047A (en)	1986-10-08	1991-01-29	Bristol Myers Co	Quinoline - or naphthyridine - carboxylic acid anti-bacterial agents
JPH01100165A (ja)	1987-10-13	1989-04-18	Shionogi & Co Ltd	オキシムまたはヒドロキシアミン誘導体系抗菌剤
US4920120A (en)	1988-01-25	1990-04-24	Warner-Lambert Company	Antibacterial agents
JPH0356479A (ja)	1989-07-24	1991-03-12	Takeshi Yokota	水溶性キノロン誘導体のｐ‐トルエンスルホン酸塩
PL166381B1 (pl)	1989-08-16	1995-05-31	Pfizer	Sposób wytwarzania nowych podstawionych kwasów 7-azabicyklochinolonokarboksylowych PL PL PL PL
US5137892A (en)	1990-12-12	1992-08-11	Abbott Laboratories	Quinoline, naphthyridine and pyridobenzoxazine derivatives
EP0541086A1 (en)	1991-11-08	1993-05-12	Kaken Pharmaceutical Co., Ltd.	Antibacterial 6-fluoro-quinolones having an oxime group on the substituent in position 7
JPH0673056A (ja)	1992-08-26	1994-03-15	Kaken Pharmaceut Co Ltd	キノリンカルボン酸誘導体およびその塩
EP0688772B1 (en)	1994-06-16	1999-05-06	LG Chemical Limited	Quinoline carboxylic acid derivatives having 7-(4-amino-methyl-3-oxime) pyrrolidine substituents and processes for their preparation
US5776944A (en) *	1994-06-16	1998-07-07	Lg Chemical Ltd.	7-(4-aminomethyl-3-methyloxyiminopyrroplidin-1-yl)-1-cyclopropyl-6-flu oro-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxylic acid and the process for the preparation thereof
JP3449658B2 (ja)	1994-12-21	2003-09-22	杏林製薬株式会社	安定性に優れた８−アルコキシキノロンカルボン酸水和物並びにその製造方法
CA2223404C (en)	1995-06-06	2001-01-16	Thomas A. Morris	Novel crystal form of anhydrous 7-(¬1.alpha., 5.alpha., 6.alpha.\|-6-amino-3-azabicyclo¬3.1.0\|hex-3-yl)-6-fluoro-1-(2,4-difluorophenyl)-1,4-dihydro-4-oxo-1,8-naphthyridine-3-carboxylic acid, methanesulfonic acid salt
UA59341C2 (uk)	1995-08-11	2003-09-15	Пфайзер, Інк.	(1s,2s)-1-(4-гідроксифеніл)-2-(4-гідрокси-4-фенілпіперидин-1-іл)-1-пропанолметансульфонат тригідрат
MA24437A1 (fr)	1996-03-29	1998-10-01	Smithkline Beecham Corp	Procede de la preparation et de la formulation de dihydrate d'eprosartan
MA24500A1 (fr)	1997-03-21	1998-10-01	Lg Life Sciences Ltd	Derive du sel d'acide carboxylique de naphthyridine .
KR100286874B1 (ko) *	1998-03-04	2001-04-16	성재갑	보호된 4-아미노메틸-피롤리딘-3-온의 제조방법
ATE249432T1 (de)	1998-05-29	2003-09-15	Upjohn Co	3-((1'-n-methylamino)ethyl-n-benzyl)pyrrolidin- monomethanesulfonat
GB9820405D0 (en)	1998-09-18	1998-11-11	Smithkline Beecham Plc	Process
DK1223935T3 (da)	1999-06-29	2008-02-04	Lg Life Sciences Ltd	Anvendelse af gemifloxacinforbindelser mod bakterier
AU6947900A (en)	1999-09-01	2001-03-26	Smithkline Beecham Corporation	Methods of use of fluoroquinolone compounds against bacteria
GB9920919D0 (en)	1999-09-03	1999-11-10	Sb Pharmco Inc	Novel compound
GB9920917D0 (en)	1999-09-03	1999-11-10	Sb Pharmco Inc	Novel process
AU7709400A (en)	1999-09-22	2001-04-24	Smithkline Beecham Corporation	Methods of use of fluoroquinolone compounds against bacteria
KR20010091379A (ko)	2000-03-15	2001-10-23	성재갑	7-(4-아미노메틸-3-옥심)피롤리딘 치환체를 갖는 퀴놀린카르복실산 유도체의 신규 제조방법
KR20020018560A (ko)	2000-09-01	2002-03-08	성재갑	3-아미노메틸-4-ｚ-메톡시이미노피롤리딘의 신규 제조방법

2002
- 2002-04-08 KR KR10-2002-0018847A patent/KR100517638B1/ko active IP Right Grant
2003
- 2003-04-04 CA CA2481217A patent/CA2481217C/en not_active Expired - Lifetime
- 2003-04-04 PL PL03372815A patent/PL372815A1/xx not_active Application Discontinuation
- 2003-04-04 US US10/510,514 patent/US7361762B2/en not_active Expired - Lifetime
- 2003-04-04 AP APAP/P/2004/003148A patent/AP1786A/en active
- 2003-04-04 MX MXPA04009777A patent/MXPA04009777A/es active IP Right Grant
- 2003-04-04 AU AU2003219581A patent/AU2003219581B2/en not_active Ceased
- 2003-04-04 EA EA200401328A patent/EA007222B1/ru not_active IP Right Cessation
- 2003-04-04 ES ES03715805T patent/ES2311694T3/es not_active Expired - Lifetime
- 2003-04-04 UA UA20041008144A patent/UA77070C2/uk unknown
- 2003-04-04 JP JP2003584056A patent/JP4315815B2/ja not_active Expired - Fee Related
- 2003-04-04 WO PCT/KR2003/000683 patent/WO2003087100A1/en active Application Filing
- 2003-04-04 OA OA1200400271A patent/OA12801A/en unknown
- 2003-04-04 DE DE60322872T patent/DE60322872D1/de not_active Expired - Lifetime
- 2003-04-04 CN CNB038095483A patent/CN1291987C/zh not_active Expired - Lifetime
- 2003-04-04 BR BRPI0309037A patent/BRPI0309037B8/pt not_active IP Right Cessation
- 2003-04-04 DK DK03715805T patent/DK1497290T3/da active
- 2003-04-04 GE GEAP8436A patent/GEP20074025B/en unknown
- 2003-04-04 PT PT03715805T patent/PT1497290E/pt unknown
- 2003-04-04 SI SI200331341T patent/SI1497290T1/sl unknown
- 2003-04-04 NZ NZ536174A patent/NZ536174A/en not_active IP Right Cessation
- 2003-04-04 EP EP03715805A patent/EP1497290B1/en not_active Expired - Lifetime
- 2003-04-04 AT AT03715805T patent/ATE404559T1/de active
2004
- 2004-09-30 IS IS7477A patent/IS2731B/is unknown
- 2004-10-05 CO CO04099283A patent/CO5611198A2/es active IP Right Grant
- 2004-10-07 ZA ZA200408088A patent/ZA200408088B/xx unknown
- 2004-10-07 MA MA27894A patent/MA26408A1/fr unknown
- 2004-10-07 HR HRP20040929AA patent/HRP20040929B1/hr not_active IP Right Cessation
- 2004-10-21 IL IL164328A patent/IL164328A/en unknown
- 2004-10-27 NO NO20044629A patent/NO330042B1/no not_active IP Right Cessation
2005
- 2005-06-29 HK HK05105460.5A patent/HK1074440A1/xx not_active IP Right Cessation
2008
- 2008-10-31 CY CY20081101234T patent/CY1108469T1/el unknown

Also Published As

Publication number	Publication date
SI1497290T1 (sl)	2008-12-31
IS7477A (is)	2004-09-30
ATE404559T1 (de)	2008-08-15
BR0309037A (pt)	2005-02-01
DK1497290T3 (da)	2008-12-15
EP1497290A1 (en)	2005-01-19
US7361762B2 (en)	2008-04-22
WO2003087100A1 (en)	2003-10-23
NO330042B1 (no)	2011-02-07
ZA200408088B (en)	2006-05-31
CA2481217A1 (en)	2003-10-23
CN1291987C (zh)	2006-12-27
ES2311694T3 (es)	2009-02-16
AP1786A (en)	2007-10-04
IL164328A (en)	2009-08-03
CY1108469T1 (el)	2014-04-09
CA2481217C (en)	2010-06-01
JP4315815B2 (ja)	2009-08-19
NZ536174A (en)	2006-09-29
MXPA04009777A (es)	2004-12-13
EA200401328A1 (ru)	2005-06-30
EA007222B1 (ru)	2006-08-25
AU2003219581A1 (en)	2003-10-27
JP2005529112A (ja)	2005-09-29
PL372815A1 (en)	2005-08-08
HK1074440A1 (en)	2005-11-11
KR20030080292A (ko)	2003-10-17
CO5611198A2 (es)	2006-02-28
UA77070C2 (uk)	2006-10-16
BRPI0309037B1 (pt)	2018-07-31
CN1649868A (zh)	2005-08-03
AU2003219581B2 (en)	2006-08-24
US20050148622A1 (en)	2005-07-07
AP2004003148A0 (en)	2004-12-31
PT1497290E (pt)	2008-11-14
MA26408A1 (fr)	2004-12-01
IS2731B (is)	2011-04-15
HRP20040929A2 (en)	2005-02-28
EP1497290A4 (en)	2006-05-10
DE60322872D1 (de)	2008-09-25
GEP20074025B (en)	2007-01-25
KR100517638B1 (ko)	2005-09-28
IL164328A0 (en)	2005-12-18
BRPI0309037B8 (pt)	2021-05-25
HRP20040929B1 (hr)	2013-12-06
EP1497290B1 (en)	2008-08-13
NO20044629L (no)	2004-10-27

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CZ311292A3 (en)	1993-12-15	Substituted tetrahydrothiophenes
KR20070090937A (ko)	2007-09-06	2-(피라졸-1-일)피리딘 유도체
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DE4446337A1 (de)	1996-06-27	Verfahren zur Herstellung von 3-Cyanobenzaldehyden