NO922842L - BENZOTIAZOLD DERIVATIVES, THE PROCEDURE FOR THEIR PREPARATION AND THEIR USE AS A THERAPEUTICS - Google Patents

BENZOTIAZOLD DERIVATIVES, THE PROCEDURE FOR THEIR PREPARATION AND THEIR USE AS A THERAPEUTICS

Info

Publication number
NO922842L
NO922842L NO92922842A NO922842A NO922842L NO 922842 L NO922842 L NO 922842L NO 92922842 A NO92922842 A NO 92922842A NO 922842 A NO922842 A NO 922842A NO 922842 L NO922842 L NO 922842L
Authority
NO
Norway
Prior art keywords
benzotiazold
therapeutics
derivatives
procedure
preparation
Prior art date
Application number
NO92922842A
Other languages
Norwegian (no)
Other versions
NO922842D0 (en
Inventor
Pascal George
Danielle De Peretti
Jean-Francois Gibert
Michel Mangane
Odette Le Galloudec
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9109137A external-priority patent/FR2679232B1/en
Priority claimed from FR9109139A external-priority patent/FR2679136A1/en
Priority claimed from FR9109138A external-priority patent/FR2679233B1/en
Priority claimed from FR9109136A external-priority patent/FR2679231B1/en
Application filed by Synthelabo filed Critical Synthelabo
Publication of NO922842D0 publication Critical patent/NO922842D0/en
Publication of NO922842L publication Critical patent/NO922842L/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
NO92922842A 1991-07-19 1992-07-17 BENZOTIAZOLD DERIVATIVES, THE PROCEDURE FOR THEIR PREPARATION AND THEIR USE AS A THERAPEUTICS NO922842L (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
FR9109137A FR2679232B1 (en) 1991-07-19 1991-07-19 ALPHA-HYDROXYIMIDAZO [2,1-B] BENZOTHIAZOLE-3-ACETAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION.
FR9109139A FR2679136A1 (en) 1991-07-19 1991-07-19 Medicaments and pharmaceutical compositions based on imidazo[2,1-b]benzothiazol-3-acetamide derivatives
FR9109138A FR2679233B1 (en) 1991-07-19 1991-07-19 IMIDAZO [2,1-B] BENZOTHIAZOLE-3-ACETAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION.
FR9109136A FR2679231B1 (en) 1991-07-19 1991-07-19 IMIDAZO [2,1-B] BENZOTHIAZOLE-3-ACETAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION, IN THERAPEUTICS.

Publications (2)

Publication Number Publication Date
NO922842D0 NO922842D0 (en) 1992-07-17
NO922842L true NO922842L (en) 1993-01-20

Family

ID=27446813

Family Applications (1)

Application Number Title Priority Date Filing Date
NO92922842A NO922842L (en) 1991-07-19 1992-07-17 BENZOTIAZOLD DERIVATIVES, THE PROCEDURE FOR THEIR PREPARATION AND THEIR USE AS A THERAPEUTICS

Country Status (15)

Country Link
EP (1) EP0524055A1 (en)
JP (1) JPH05202063A (en)
KR (1) KR930002358A (en)
CN (1) CN1068826A (en)
AU (1) AU646582B2 (en)
CA (1) CA2074112A1 (en)
CZ (1) CZ224492A3 (en)
FI (1) FI923290A (en)
HU (1) HU9202358D0 (en)
IE (1) IE922342A1 (en)
IL (1) IL102536A0 (en)
MX (1) MX9204179A (en)
NO (1) NO922842L (en)
NZ (1) NZ243595A (en)
PL (1) PL295306A1 (en)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2699921B1 (en) * 1992-12-30 1995-02-10 Synthelabo 2- (Thien-2-yl) imidazo [2,1-b] benzothiazole-3-acetic acid derivatives, their preparation and their therapeutic use.
WO1996028454A1 (en) * 1995-03-13 1996-09-19 Nikken Chemicals Co., Ltd. Imidazothiazole compounds
WO1998006724A1 (en) * 1996-08-09 1998-02-19 Yamanouchi Pharmaceutical Co., Ltd. Metabotropic glutamate receptor agonists
FR2759698B1 (en) * 1997-02-20 1999-03-19 Synthelabo 1,4-DIPHENYLIMIDAZOLE-5-ACETAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
DK0891978T3 (en) * 1997-07-18 2002-07-01 Hoffmann La Roche 5H-thiazole (3,2-a) pyrimidinderivativer
EP1357124B1 (en) * 2001-01-30 2005-08-03 Zenyaku Kogyo Kabushiki Kaisha Heterocyclic compounds and cerebral function improvers containing the same as the active ingredient
AU2002344951A1 (en) * 2001-07-02 2003-01-21 Boehringer Ingelheim International Gmbh Substituted piperazine and diazepanes as histamine h3 receptor agonists
ATE423116T1 (en) * 2002-12-18 2009-03-15 Mallinckrodt Inc SYNTHESIS OF HETEROARYL ACETAMIDS
WO2004089356A2 (en) * 2003-04-03 2004-10-21 Semafore Pharmaceuticals Inc. Targeted bone marrow protection agents
JP4610668B2 (en) 2006-03-17 2011-01-12 アムビト ビオスシエンセス コルポラチオン Imidazolothiazole compounds for treating diseases
DK2201018T3 (en) 2007-09-19 2016-05-17 Ambit Biosciences Corp SOLID FORMS COMPRISING N- (5-TERT-BUTYL-ISOXAZOL-3-YL) -N '- {4- [7- (2-morpholin-4-yl-ethoxy) imidazo [2,1-b] [1, 3] benzothiazole-2-YL] PHENYL} UREA, COMPOSITIONS THEREOF AND USES THEREFORE
US20190292204A1 (en) * 2018-03-26 2019-09-26 University of Sharjah C/o Dr. Mohamed Al Hemairy [email protected] Novel heterocyclic systems and pharmaceutical compositions thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4464384A (en) * 1981-12-23 1984-08-07 Yamanouchi Pharmaceutical Co., Ltd. 2-Phenylimidazo[2,1-b]benzothiazole compounds, salts thereof, process of producing them, and pharmaceutical compositions containing them
GB8724566D0 (en) * 1987-10-20 1987-11-25 Roussel Lab Ltd Chemical compounds
JP2726999B2 (en) * 1988-06-22 1998-03-11 日研化学株式会社 Imidazo [2,1-b] benzothiazole derivatives and anti-ulcer agents containing the compounds as active ingredients
GB8908845D0 (en) * 1989-04-19 1989-06-07 Roussel Lab Ltd Chemical compounds
CA2028756A1 (en) * 1989-11-24 1991-05-25 Alfons H. M. Raeymaekers Immunostimulating 6-aryl-5,6-dihydro-imidazo[2,1-b]thiazole derivatives

Also Published As

Publication number Publication date
AU646582B2 (en) 1994-02-24
IE922342A1 (en) 1993-01-27
EP0524055A1 (en) 1993-01-20
KR930002358A (en) 1993-02-23
NO922842D0 (en) 1992-07-17
FI923290A0 (en) 1992-07-17
FI923290A (en) 1993-01-20
PL295306A1 (en) 1993-03-08
MX9204179A (en) 1993-08-01
CZ224492A3 (en) 1993-02-17
NZ243595A (en) 1994-08-26
CN1068826A (en) 1993-02-10
CA2074112A1 (en) 1993-01-20
AU2038092A (en) 1993-01-21
JPH05202063A (en) 1993-08-10
IL102536A0 (en) 1993-01-14
HU9202358D0 (en) 1992-10-28

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