NO921449L - Karbamater av rapamycin - Google Patents

Karbamater av rapamycin

Info

Publication number: NO921449L
Authority: NO; Norway
Prior art keywords: rapamycin; carbamates
Prior art date: 1991-04-17

Application number

NO92921449A

Other languages

English (en)

Other versions

NO921449D0 (no

Inventor

Wenling Kao

Robert Lewis Vogel

John Henry Musser

Original Assignee

American Home Prod

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1991-04-17

Filing date

1992-04-10

Publication date

1992-10-19

1991-04-17 Priority claimed from US07/686,728 external-priority patent/US5118678A/en

1992-02-18 Priority claimed from US07/837,048 external-priority patent/US5194447A/en

1992-04-10 Application filed by American Home Prod filed Critical American Home Prod

1992-04-10 Publication of NO921449D0 publication Critical patent/NO921449D0/no

1992-10-19 Publication of NO921449L publication Critical patent/NO921449L/no

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/18—Bridged systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/08—Plasma substitutes; Perfusion solutions; Dialytics or haemodialytics; Drugs for electrolytic or acid-base disorders, e.g. hypovolemic shock
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives

NO92921449A 1991-04-17 1992-04-10 Karbamater av rapamycin NO921449L (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US07/686,728 US5118678A (en)	1991-04-17	1991-04-17	Carbamates of rapamycin
US07/837,048 US5194447A (en)	1992-02-18	1992-02-18	Sulfonylcarbamates of rapamycin

Publications (2)

Publication Number	Publication Date
NO921449D0 NO921449D0 (no)	1992-04-10
NO921449L true NO921449L (no)	1992-10-19

Family

ID=27103855

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO92921449A NO921449L (no)	1991-04-17	1992-04-10	Karbamater av rapamycin

Country Status (12)

Country	Link
EP (1)	EP0509795A2 (no)
JP (1)	JPH05112573A (no)
KR (1)	KR920019798A (no)
AU (1)	AU642592B2 (no)
CZ (1)	CZ117392A3 (no)
FI (1)	FI921595A (no)
HU (1)	HU9201254D0 (no)
IE (1)	IE921249A1 (no)
MX (1)	MX9201710A (no)
NO (1)	NO921449L (no)
NZ (1)	NZ242367A (no)
SK (1)	SK117392A3 (no)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5776943A (en) *	1991-05-14	1998-07-07	American Home Products Corporation	Rapamycin metabolites
US5118677A (en) *	1991-05-20	1992-06-02	American Home Products Corporation	Amide esters of rapamycin
WO1993018043A1 (en) *	1992-03-05	1993-09-16	American Home Products Corporation	Novel rapamycin 42-sulfonates and 42-(n-carboalkoxy)sulfamates useful as immunosuppressive agents
GB9307491D0 (en) *	1993-04-08	1993-06-02	Sandoz Ltd	Organic compounds
CH686761A5 (de)	1993-05-27	1996-06-28	Sandoz Ag	Galenische Formulierungen.
CA2175215C (en) *	1993-11-19	2008-06-03	Yat Sun Or	Semisynthetic analogs of rapamycin (macrolides) being immunomodulators
US5527907A (en) *	1993-11-19	1996-06-18	Abbott Laboratories	Macrolide immunomodulators
US5362718A (en)	1994-04-18	1994-11-08	American Home Products Corporation	Rapamycin hydroxyesters
JP2002534468A (ja)	1999-01-13	2002-10-15	バイエルコーポレイション	ｐ３８キナーゼ阻害剤としてのω−カルボキシアリール置換ジフェニル尿素
US8124630B2 (en)	1999-01-13	2012-02-28	Bayer Healthcare Llc	ω-carboxyaryl substituted diphenyl ureas as raf kinase inhibitors
WO2001012633A1 (en) *	1999-08-18	2001-02-22	American Home Products Corporation	Water soluble sdz-rad esters
EP2324825A1 (en)	2002-02-11	2011-05-25	Bayer Healthcare LLC	Aryl ureas with angiogenesis inhibiting activity
US7557129B2 (en)	2003-02-28	2009-07-07	Bayer Healthcare Llc	Cyanopyridine derivatives useful in the treatment of cancer and other disorders
ATE366108T1 (de)	2003-05-20	2007-07-15	Bayer Pharmaceuticals Corp	Diaryl-harnstoffe für durch pdgfr vermittelte krankheiten
NZ580384A (en)	2003-07-23	2011-03-31	Bayer Pharmaceuticals Corp	4{4-[3-(4-chloro-3-trifluoromethylphenyl)-ureido]-3-fluorophenoxy}-pyridine-2-carboxylic acid methylamide and metabolites for the treatment and prevention of diseases and conditions
WO2005042567A1 (en) *	2003-11-03	2005-05-12	Altachem Pharma Ltd.	Rapamycin peptides conjugates: synthesis and uses thereof
US8021849B2 (en)	2004-11-05	2011-09-20	Siemens Healthcare Diagnostics Inc.	Methods and kits for the determination of sirolimus in a sample
CA2602010A1 (en)	2005-03-07	2006-09-14	Wyeth	Oxepane isomer of 42-o-(2-hydroxy)ethyl-rapamycin
US7189582B2 (en)	2005-04-27	2007-03-13	Dade Behring Inc.	Compositions and methods for detection of sirolimus
CA3126495A1 (en) *	2019-01-25	2020-07-30	NodThera Limited	Carbamate derivatives and uses thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4885171A (en) *	1978-11-03	1989-12-05	American Home Products Corporation	Use of rapamycin in treatment of certain tumors
US4316885A (en) *	1980-08-25	1982-02-23	Ayerst, Mckenna And Harrison, Inc.	Acyl derivatives of rapamycin
US4650803A (en) *	1985-12-06	1987-03-17	University Of Kansas	Prodrugs of rapamycin
AU6286690A (en) *	1989-08-18	1991-04-03	Fisons Plc	Macrocyclic compounds
PT98990A (pt) *	1990-09-19	1992-08-31	American Home Prod	Processo para a preparacao de esteres de acidos carboxilicos de rapamicina
US5118677A (en) *	1991-05-20	1992-06-02	American Home Products Corporation	Amide esters of rapamycin

1992
- 1992-04-10 FI FI921595A patent/FI921595A/fi unknown
- 1992-04-10 JP JP4090825A patent/JPH05112573A/ja active Pending
- 1992-04-10 NO NO92921449A patent/NO921449L/no unknown
- 1992-04-11 KR KR1019920006033A patent/KR920019798A/ko not_active Application Discontinuation
- 1992-04-13 HU HU9201254A patent/HU9201254D0/hu unknown
- 1992-04-13 MX MX9201710A patent/MX9201710A/es unknown
- 1992-04-14 AU AU14880/92A patent/AU642592B2/en not_active Ceased
- 1992-04-15 NZ NZ24236792A patent/NZ242367A/en unknown
- 1992-04-15 EP EP19920303401 patent/EP0509795A2/en not_active Withdrawn
- 1992-04-16 IE IE124992A patent/IE921249A1/en not_active Application Discontinuation
- 1992-04-16 CZ CS921173A patent/CZ117392A3/cs unknown
- 1992-04-16 SK SK1173-92A patent/SK117392A3/sk unknown

Also Published As

Publication number	Publication date
FI921595A0 (fi)	1992-04-10
KR920019798A (ko)	1992-11-20
NO921449D0 (no)	1992-04-10
SK117392A3 (en)	1995-04-12
JPH05112573A (ja)	1993-05-07
CZ117392A3 (en)	1993-09-15
EP0509795A3 (no)	1994-03-23
HU9201254D0 (en)	1992-07-28
IE921249A1 (en)	1992-10-21
AU1488092A (en)	1992-10-22
MX9201710A (es)	1993-01-01
FI921595A (fi)	1992-10-18
EP0509795A2 (en)	1992-10-21
NZ242367A (en)	1994-07-26
AU642592B2 (en)	1993-10-21

Publication	Publication Date	Title
NO921217D0 (no)	1992-03-27	Silyletere av rapamycin
NO921976D0 (no)	1992-05-19	Amidestere av rapamycin
ZA922738B (en)	1993-10-14	Carbamates of rapamycin
FI931203A0 (fi)	1993-03-18	Karboxylsyraestrar av rapamycin
NO921449L (no)	1992-10-19	Karbamater av rapamycin
DE69332540D1 (de)	2003-01-16	Rapamycinderivate
DE69332484D1 (de)	2002-12-19	Rapamycinderivate
FI935223A (fi)	1993-11-24	Rake-mottagare med selektiv kombinering av straolar
PH31253A (en)	1998-06-18	Carbamates of rapamycin.
FI935016A (fi)	1993-11-12	Kalibrering av effektmaetare
FI931627A (fi)	1993-04-08	Foerfarande foer producering av tecken pao diamanter
NO914666L (no)	1992-05-29	Fjerning av trialkylarsiner
FI930376A (fi)	1993-11-30	Tillslutningsanordning av gaengtyp med saekringsorgan
DE69332582T2 (de)	2003-11-20	Rapamycinderivate
FI915242A (fi)	1993-05-07	Rf-skaermning av kretskort
FI931773A0 (fi)	1993-04-20	Pao en masspektrometer baserat kontinuerligt utslaeppsoevervakningssystemfoer maetning av roekgaser fraon farligt avfall
NO940190D0 (no)	1994-01-19	Anvendelse av x-ketoglutarat
FI935756A (fi)	1993-12-20	Paoskyndande av laekningen av en skada
FI932055A (fi)	1993-05-06	Foerfarande foer betahaerdning av skyddshoeljet pao kaernbraensle
NO931399D0 (no)	1993-04-16	Anvendelse av naturstein
FI923360A (fi)	1993-01-25	Foerfarande foer framstaellning av dimetylacetoacetamid
FI933214A (fi)	1994-01-23	Foerfarande foer framstaellning av mannitol
FI932658A0 (fi)	1993-06-10	Foerfarande foer framstaellning av viskosfibrer med bandformade tvaersnitt
FI925493A0 (fi)	1992-12-03	Rumselementsystem foer ersaettning av vaotutrymmen med tillfaelligutrymmeni samband med byggnadsarbeten
ZA937515B (en)	1995-04-11	Carbamates of rapamycin