NO325454B1 - Anvendelse av N-{5-[4-(4-metyl-piperazino-metyl)-benzoylamido]-2-metylfenyl}-4-(3-pyridyl)-2-pyrimidin-amin. - Google Patents

Anvendelse av N-{5-[4-(4-metyl-piperazino-metyl)-benzoylamido]-2-metylfenyl}-4-(3-pyridyl)-2-pyrimidin-amin. Download PDF

Info

Publication number: NO325454B1
Authority: NO; Norway
Prior art keywords: cells; methyl; compound; acid; kit
Prior art date: 2001-04-05

Application number

NO20034414A

Other languages

English (en)

Norwegian (no)

Other versions

NO20034414D0 (no

NO20034414L (no

Inventor

Kenichi Koike

Atsushi Komiyama

Kovichi Takeuchi

Original Assignee

Novartis Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-04-05

Filing date

2003-10-02

Publication date

2008-05-05

2003-10-02 Application filed by Novartis Ag filed Critical Novartis Ag

2003-10-02 Publication of NO20034414D0 publication Critical patent/NO20034414D0/no

2003-12-04 Publication of NO20034414L publication Critical patent/NO20034414L/no

2008-05-05 Publication of NO325454B1 publication Critical patent/NO325454B1/no

Links

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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents

NO20034414A 2001-04-05 2003-10-02 Anvendelse av N-{5-[4-(4-metyl-piperazino-metyl)-benzoylamido]-2-metylfenyl}-4-(3-pyridyl)-2-pyrimidin-amin. NO325454B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GBGB0108606.5A GB0108606D0 (en)	2001-04-05	2001-04-05	Organic compounds
PCT/US2002/010742 WO2002080925A1 (en)	2001-04-05	2002-04-05	Use of n-phenyl-2-pyrimidineamine derivativea against mast cell-based diseases like allergic disorders

Publications (3)

Publication Number	Publication Date
NO20034414D0 NO20034414D0 (no)	2003-10-02
NO20034414L NO20034414L (no)	2003-12-04
NO325454B1 true NO325454B1 (no)	2008-05-05

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ID=9912339

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Application Number	Title	Priority Date	Filing Date
NO20034414A NO325454B1 (no)	2001-04-05	2003-10-02	Anvendelse av N-{5-[4-(4-metyl-piperazino-metyl)-benzoylamido]-2-metylfenyl}-4-(3-pyridyl)-2-pyrimidin-amin.

Country Status (18)

Country	Link
EP (1)	EP1389113A1 (ko)
KR (2)	KR20040007485A (ko)
CN (1)	CN1529602A (ko)
AU (1)	AU2002307140B2 (ko)
BR (1)	BR0208663A (ko)
CA (1)	CA2443092A1 (ko)
CZ (1)	CZ20032705A3 (ko)
GB (1)	GB0108606D0 (ko)
HU (1)	HUP0303751A3 (ko)
IL (1)	IL158061A0 (ko)
MX (1)	MXPA03009058A (ko)
NO (1)	NO325454B1 (ko)
NZ (1)	NZ528934A (ko)
PL (1)	PL363080A1 (ko)
RU (1)	RU2304436C2 (ko)
SK (1)	SK12312003A3 (ko)
WO (1)	WO2002080925A1 (ko)
ZA (1)	ZA200307563B (ko)

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US7678805B2 (en)	2001-06-29	2010-03-16	Ab Science	Use of tyrosine kinase inhibitors for treating inflammatory bowel diseases (IBD)
JP2004537537A (ja)	2001-06-29	2004-12-16	アブサイエンス	炎症性疾患を治療するためのチロシンキナーゼ阻害剤の使用法
ATE376182T1 (de)	2001-06-29	2007-11-15	Ab Science	C-kit inhibitoren
US7700610B2 (en)	2001-06-29	2010-04-20	Ab Science	Use of tyrosine kinase inhibitors for treating allergic diseases
GB0201882D0 (en) *	2002-01-28	2002-03-13	Novartis Ag	Organic compounds
CA2479257A1 (en) *	2002-03-21	2003-10-02	Dana-Farber Cancer Institute, Inc.	Inhibition of cell death responses induced by oxidative stress
US8450302B2 (en)	2002-08-02	2013-05-28	Ab Science	2-(3-aminoaryl) amino-4-aryl-thiazoles and their use as c-kit inhibitors
ES2294344T3 (es)	2002-08-02	2008-04-01	Ab Science	2-(3-aminoaril)amino-4-aril-tiazoles y su utilizacion como inhibidores de c-kit.
JP2006519220A (ja) *	2003-02-27	2006-08-24	アブサイエンス	異なる型の肥満細胞症に適合可能なテイラーメイド治療方法
AU2003232650A1 (en) *	2003-05-06	2004-11-26	Il Yang Pharm Co., Ltd.	N-phenyl-2-pyrimidine-amine derivatives and process for the preparation thereof
TWI324604B (en) *	2003-06-18	2010-05-11	Novartis Ag	New use of staurosporine derivatives
WO2005115385A1 (en) *	2004-05-24	2005-12-08	Ab Science	Use of c-kit inhibitors for treating acne
JP2008510766A (ja) *	2004-08-27	2008-04-10	ゲーペーツェービオテックアーゲー	ピリミジン誘導体
CA2606716C (en) *	2005-05-02	2013-07-23	Novartis Ag	Use of pyrimidylaminobenzamide derivatives for the treatment of systematic mastocytosis
KR100845278B1 (ko) *	2006-08-04	2008-07-09	포항공과대학교 산학협력단	비만 세포의 활성을 유도하는 펩타이드 및 이를 포함하는면역조절제
ES2633691T3 (es) *	2009-04-06	2017-09-22	Neurotech Pharmaceuticals Co., Ltd.	Composición farmacéutica para tratar o prevenir lesiones por quemaduras
CN103058935B (zh) *	2013-01-15	2015-05-06	四川大学	一种嘧啶类化合物及其制备方法和用途

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CO4940418A1 (es) *	1997-07-18	2000-07-24	Novartis Ag	Modificacion de cristal de un derivado de n-fenil-2- pirimidinamina, procesos para su fabricacion y su uso

2001
- 2001-04-05 GB GBGB0108606.5A patent/GB0108606D0/en not_active Ceased
2002
- 2002-04-05 CZ CZ20032705A patent/CZ20032705A3/cs unknown
- 2002-04-05 IL IL15806102A patent/IL158061A0/xx unknown
- 2002-04-05 AU AU2002307140A patent/AU2002307140B2/en not_active Expired
- 2002-04-05 EP EP02763956A patent/EP1389113A1/en not_active Ceased
- 2002-04-05 CA CA002443092A patent/CA2443092A1/en not_active Abandoned
- 2002-04-05 CN CNA028089707A patent/CN1529602A/zh active Pending
- 2002-04-05 PL PL02363080A patent/PL363080A1/xx unknown
- 2002-04-05 BR BR0208663-8A patent/BR0208663A/pt not_active IP Right Cessation
- 2002-04-05 KR KR10-2003-7012939A patent/KR20040007485A/ko not_active Application Discontinuation
- 2002-04-05 RU RU2003130635/15A patent/RU2304436C2/ru not_active IP Right Cessation
- 2002-04-05 HU HU0303751A patent/HUP0303751A3/hu unknown
- 2002-04-05 KR KR1020097003644A patent/KR20090034998A/ko not_active Application Discontinuation
- 2002-04-05 MX MXPA03009058A patent/MXPA03009058A/es not_active Application Discontinuation
- 2002-04-05 NZ NZ528934A patent/NZ528934A/en not_active IP Right Cessation
- 2002-04-05 SK SK1231-2003A patent/SK12312003A3/sk not_active Application Discontinuation
- 2002-04-05 WO PCT/US2002/010742 patent/WO2002080925A1/en active Application Filing
2003
- 2003-09-29 ZA ZA200307563A patent/ZA200307563B/en unknown
- 2003-10-02 NO NO20034414A patent/NO325454B1/no not_active IP Right Cessation

Also Published As

Publication number	Publication date
KR20090034998A (ko)	2009-04-08
PL363080A1 (en)	2004-11-15
NO20034414D0 (no)	2003-10-02
CZ20032705A3 (en)	2004-06-16
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Publication	Publication Date	Title
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