NO305839B1 - FremgangsmÕte for fremstilling av 7-trialkylsilyl-baccatin-III - Google Patents

FremgangsmÕte for fremstilling av 7-trialkylsilyl-baccatin-III

Info

Publication number: NO305839B1
Authority: NO; Norway
Prior art keywords: pct; symbols; iii; preparation; date oct
Prior art date: 1994-04-05

Application number

NO964103A

Other languages

English (en)

Norwegian (no)

Other versions

NO964103D0 (no

NO964103L (no

Inventor

Jean-Pierre Bastart

Jean-Pierre Leconte

Original Assignee

Rh Ne Poulenc Rorer Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1994-04-05

Filing date

1996-09-27

Publication date

1999-08-02

1996-09-27 Application filed by Rh Ne Poulenc Rorer Sa filed Critical Rh Ne Poulenc Rorer Sa

1996-09-27 Publication of NO964103D0 publication Critical patent/NO964103D0/no

1996-09-27 Publication of NO964103L publication Critical patent/NO964103L/no

1999-08-02 Publication of NO305839B1 publication Critical patent/NO305839B1/no

Links

YWLXLRUDGLRYDR-ZHPRIASZSA-N 5beta,20-epoxy-1,7beta,10beta,13alpha-tetrahydroxy-9-oxotax-11-ene-2alpha,4alpha-diyl 4-acetate 2-benzoate Chemical compound O([C@H]1[C@H]2[C@@](C([C@H](O)C3=C(C)[C@@H](O)C[C@]1(O)C3(C)C)=O)(C)[C@@H](O)C[C@H]1OC[C@]12OC(=O)C)C(=O)C1=CC=CC=C1 YWLXLRUDGLRYDR-ZHPRIASZSA-N 0.000 abstract 2
-1 alkyl radicals Chemical class 0.000 abstract 2
125000004432 carbon atom Chemical group C* 0.000 abstract 2
CIUQDSCDWFSTQR-UHFFFAOYSA-N [C]1=CC=CC=C1 Chemical compound [C]1=CC=CC=C1 CIUQDSCDWFSTQR-UHFFFAOYSA-N 0.000 abstract 1
QUPDWYMUPZLYJZ-UHFFFAOYSA-N ethyl Chemical compound C[CH2] QUPDWYMUPZLYJZ-UHFFFAOYSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
- C07F7/1804—Compounds having Si-O-C linkages
- C07F7/1872—Preparation; Treatments not provided for in C07F7/20
- C07F7/1892—Preparation; Treatments not provided for in C07F7/20 by reactions not provided for in C07F7/1876 - C07F7/1888
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
- C07F7/1804—Compounds having Si-O-C linkages
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
- C07F7/1804—Compounds having Si-O-C linkages
- C07F7/1872—Preparation; Treatments not provided for in C07F7/20
- C07F7/188—Preparation; Treatments not provided for in C07F7/20 by reactions involving the formation of Si-O linkages

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Epoxy Compounds (AREA)
Crystals, And After-Treatments Of Crystals (AREA)
Silicon Compounds (AREA)
Saccharide Compounds (AREA)
Peptides Or Proteins (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Liquid Deposition Of Substances Of Which Semiconductor Devices Are Composed (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Silicon Polymers (AREA)
Cephalosporin Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Steroid Compounds (AREA)
Magnetic Resonance Imaging Apparatus (AREA)
Processes Of Treating Macromolecular Substances (AREA)
Internal Circuitry In Semiconductor Integrated Circuit Devices (AREA)

NO964103A 1994-04-05 1996-09-27 FremgangsmÕte for fremstilling av 7-trialkylsilyl-baccatin-III NO305839B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR9403979A FR2718137B1 (fr)	1994-04-05	1994-04-05	Procédé de préparation de trialcoylsilyl-7 baccatine III.
PCT/FR1995/000419 WO1995026967A1 (fr)	1994-04-05	1995-04-03	Procede de preparation de trialcoylsilyl-7 baccatine iii

Publications (3)

Publication Number	Publication Date
NO964103D0 NO964103D0 (no)	1996-09-27
NO964103L NO964103L (no)	1996-09-27
NO305839B1 true NO305839B1 (no)	1999-08-02

Family

ID=9461745

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO964103A NO305839B1 (no)	1994-04-05	1996-09-27	FremgangsmÕte for fremstilling av 7-trialkylsilyl-baccatin-III

Country Status (33)

Country	Link
US (1)	US5670658A (ja)
EP (1)	EP0754185B1 (ja)
JP (1)	JP3718225B2 (ja)
KR (1)	KR100399246B1 (ja)
CN (1)	CN1058497C (ja)
AT (1)	ATE160351T1 (ja)
AU (1)	AU683560B2 (ja)
BG (1)	BG62735B1 (ja)
BR (1)	BR9507444A (ja)
CA (1)	CA2186916C (ja)
CZ (1)	CZ288397B6 (ja)
DE (1)	DE69501080T2 (ja)
DK (1)	DK0754185T3 (ja)
EE (1)	EE03240B1 (ja)
ES (1)	ES2109103T3 (ja)
FI (1)	FI115970B (ja)
FR (1)	FR2718137B1 (ja)
GE (1)	GEP19991537B (ja)
GR (1)	GR3025448T3 (ja)
HU (1)	HU214158B (ja)
LT (1)	LT4185B (ja)
LV (1)	LV11691B (ja)
MX (1)	MX9604466A (ja)
NO (1)	NO305839B1 (ja)
NZ (1)	NZ284490A (ja)
PL (1)	PL316588A1 (ja)
RO (1)	RO115631B1 (ja)
RU (1)	RU2127729C1 (ja)
SK (1)	SK280448B6 (ja)
TW (1)	TW284765B (ja)
UA (1)	UA44730C2 (ja)
WO (1)	WO1995026967A1 (ja)
ZA (1)	ZA952733B (ja)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5973160A (en) *	1992-12-23	1999-10-26	Poss; Michael A.	Methods for the preparation of novel sidechain-bearing taxanes
US7288665B1 (en) *	1997-08-18	2007-10-30	Florida State University	Process for selective derivatization of taxanes
ES2195378T3 (es)	1997-08-21	2003-12-01	Univ Florida State	Procedimiento para la sintesis de taxanos.
JP2004525860A (ja)	2000-09-22	2004-08-26	ブリストル−マイヤーズスクイブカンパニー	併用化学療法剤の毒性を低下させる方法
ATE431343T1 (de) *	2002-10-09	2009-05-15	Chatham Biotec Ltd	Thio-analoga von paclitaxel und deren vorprodukte
US7202370B2 (en) *	2003-10-27	2007-04-10	Conor Medsystems, Inc.	Semi-synthesis of taxane intermediates from 9-dihydro-13-acetylbaccatin III
MXPA06012606A (es) *	2004-05-14	2007-01-31	Immunogen Inc	Un metodo facil para sintetizar compuestos de bacatina iii.
CZ298333B6 (cs) *	2005-09-26	2007-08-29	Zentiva, A. S	Zpusob prípravy 7-trialkylsilylbaccatinu III
JP5588983B2 (ja)	2008-08-11	2014-09-10	ウェルズファーゴバンクナショナルアソシエイション	マルチアームポリマーアルカノエートコンジュゲート
US9199954B2 (en)	2010-12-22	2015-12-01	Nektar Therapeutics	Non-ring hydroxy substituted taxanes and methods for synthesizing the same
US10894087B2 (en)	2010-12-22	2021-01-19	Nektar Therapeutics	Multi-arm polymeric prodrug conjugates of cabazitaxel-based compounds
US20130331443A1 (en)	2010-12-22	2013-12-12	Nektar Therapeutics	Multi-arm polymeric prodrug conjugates of taxane-based compounds

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4823167A (en) *	1986-12-16	1989-04-18	Baxter International Inc.	Catheter calibration device
FR2629818B1 (fr) *	1988-04-06	1990-11-16	Centre Nat Rech Scient	Procede de preparation du taxol
MX9102128A (es)	1990-11-23	1992-07-08	Rhone Poulenc Rorer Sa	Derivados de taxano,procedimiento para su preparacion y composicion farmaceutica que los contiene
US5229526A (en) *	1991-09-23	1993-07-20	Florida State University	Metal alkoxides
US5597931A (en) *	1992-03-30	1997-01-28	Sloan-Kettering Institute For Cancer Research	Total synthesis of taxol and analogues thereof
US5475011A (en) *	1993-03-26	1995-12-12	The Research Foundation Of State University Of New York	Anti-tumor compounds, pharmaceutical compositions, methods for preparation thereof and for treatment
US5405972A (en) *	1993-07-20	1995-04-11	Florida State University	Synthetic process for the preparation of taxol and other tricyclic and tetracyclic taxanes
US5449790A (en) *	1994-04-06	1995-09-12	Hauser Chemical Research, Inc.	Preparation of 10-deacetylbaccatin III and 7-protected-10-deacetylbaccatin III derivatives from 10-deacetyl taxol A, 10-deacetyl taxol B, and 10-deacetyl taxol C

1994
- 1994-04-05 FR FR9403979A patent/FR2718137B1/fr not_active Expired - Fee Related
1995
- 1995-03-22 TW TW084102793A patent/TW284765B/zh not_active IP Right Cessation
- 1995-04-03 UA UA96093735A patent/UA44730C2/uk unknown
- 1995-04-03 CA CA002186916A patent/CA2186916C/fr not_active Expired - Lifetime
- 1995-04-03 DE DE69501080T patent/DE69501080T2/de not_active Expired - Lifetime
- 1995-04-03 GE GEAP19953433A patent/GEP19991537B/en unknown
- 1995-04-03 CN CN95192429A patent/CN1058497C/zh not_active Expired - Lifetime
- 1995-04-03 AU AU23096/95A patent/AU683560B2/en not_active Expired
- 1995-04-03 ES ES95916696T patent/ES2109103T3/es not_active Expired - Lifetime
- 1995-04-03 WO PCT/FR1995/000419 patent/WO1995026967A1/fr active IP Right Grant
- 1995-04-03 PL PL95316588A patent/PL316588A1/xx unknown
- 1995-04-03 CZ CZ19962900A patent/CZ288397B6/cs not_active IP Right Cessation
- 1995-04-03 BR BR9507444A patent/BR9507444A/pt not_active IP Right Cessation
- 1995-04-03 HU HU9602735A patent/HU214158B/hu unknown
- 1995-04-03 MX MX9604466A patent/MX9604466A/es unknown
- 1995-04-03 RO RO96-01921A patent/RO115631B1/ro unknown
- 1995-04-03 RU RU96120192/04A patent/RU2127729C1/ru active
- 1995-04-03 JP JP52546695A patent/JP3718225B2/ja not_active Expired - Lifetime
- 1995-04-03 KR KR1019960705642A patent/KR100399246B1/ko not_active IP Right Cessation
- 1995-04-03 AT AT95916696T patent/ATE160351T1/de active
- 1995-04-03 US US08/722,103 patent/US5670658A/en not_active Expired - Lifetime
- 1995-04-03 DK DK95916696.8T patent/DK0754185T3/da active
- 1995-04-03 ZA ZA952733A patent/ZA952733B/xx unknown
- 1995-04-03 EP EP95916696A patent/EP0754185B1/fr not_active Expired - Lifetime
- 1995-04-03 SK SK1265-96A patent/SK280448B6/sk not_active IP Right Cessation
- 1995-04-03 NZ NZ284490A patent/NZ284490A/en not_active IP Right Cessation
- 1995-04-03 EE EE9600143A patent/EE03240B1/xx unknown
1996
- 1996-09-24 LT LT96-137A patent/LT4185B/lt not_active IP Right Cessation
- 1996-09-27 NO NO964103A patent/NO305839B1/no not_active IP Right Cessation
- 1996-10-04 BG BG100886A patent/BG62735B1/bg unknown
- 1996-10-04 FI FI964001A patent/FI115970B/fi not_active IP Right Cessation
- 1996-10-07 LV LVP-96-392A patent/LV11691B/lv unknown
1997
- 1997-11-20 GR GR970401504T patent/GR3025448T3/el unknown

Also Published As

Publication number	Publication date
FI964001A0 (fi)	1996-10-04
BG100886A (en)	1998-01-30
FR2718137B1 (fr)	1996-04-26
SK126596A3 (en)	1997-04-09
ZA952733B (en)	1996-01-09
NZ284490A (en)	1998-08-26
AU683560B2 (en)	1997-11-13
DE69501080T2 (de)	1998-04-02
JP3718225B2 (ja)	2005-11-24
HU214158B (hu)	1998-01-28
ATE160351T1 (de)	1997-12-15
LT4185B (en)	1997-07-25
HU9602735D0 (en)	1996-11-28
GR3025448T3 (en)	1998-02-27
AU2309695A (en)	1995-10-23
KR100399246B1 (ko)	2004-02-11
WO1995026967A1 (fr)	1995-10-12
PL316588A1 (en)	1997-01-20
HUT76035A (en)	1997-06-30
RO115631B1 (ro)	2000-04-28
LT96137A (en)	1997-02-25
BG62735B1 (bg)	2000-06-30
GEP19991537B (en)	1999-03-05
LV11691B (en)	1997-06-20
NO964103D0 (no)	1996-09-27
EE03240B1 (et)	1999-12-15
DE69501080D1 (de)	1998-01-02
MX9604466A (es)	1997-07-31
CA2186916C (fr)	2004-05-25
LV11691A (lv)	1997-02-20
BR9507444A (pt)	1997-09-16
DK0754185T3 (da)	1998-01-26
US5670658A (en)	1997-09-23
RU2127729C1 (ru)	1999-03-20
NO964103L (no)	1996-09-27
TW284765B (ja)	1996-09-01
EP0754185B1 (fr)	1997-11-19
FI964001A (fi)	1996-10-04
UA44730C2 (uk)	2002-03-15
JPH09512522A (ja)	1997-12-16
CN1058497C (zh)	2000-11-15
CA2186916A1 (fr)	1995-10-12
CZ290096A3 (en)	1997-01-15
ES2109103T3 (es)	1998-01-01
CZ288397B6 (en)	2001-06-13
FI115970B (fi)	2005-08-31
FR2718137A1 (fr)	1995-10-06
SK280448B6 (sk)	2000-02-14
EP0754185A1 (fr)	1997-01-22
CN1145073A (zh)	1997-03-12

Legal Events

Date	Code	Title	Description
2015-04-13	MK1K	Patent expired

Publication	Publication Date	Title
GB9412590D0 (en)	1994-08-10	Organic compounds
ATE187445T1 (de)	1999-12-15	Verfahren zur herstellung von chinazolinderivaten
NO964103D0 (no)	1996-09-27	Fremgangsmåte for fremstilling av 7-trialkylsilyl-baccatin-III
EP0994106A4 (en)	2002-08-07	METHOD FOR PRODUCING CARBAMOYL-SUBSTITUTED IMIDAZOLE DERIVATIVES
DE69926223D1 (de)	2005-08-25	Verfahren zur herstellung von zwischenprodukten
ATE363460T1 (de)	2007-06-15	Verfahren zur herstellung von fluorhalogenalkanen
LT96138A (en)	1997-02-25	Processfor the preparation of 7-hydroxy taxanes
DE60110019D1 (de)	2005-05-19	Verfahren zur Herstellung von Cyclopropancarboxylaten
ATE188694T1 (de)	2000-01-15	Verfahren zur herstellung von benzopyranderivaten
MX9804255A (es)	1998-09-30	Ditiazoldioxidos y su uso como microbicidas.
ATE208388T1 (de)	2001-11-15	Eintopfverfahren zur herstellung von 2- oxazolidinonderivate
DE50114223D1 (de)	2008-09-25	Verfahren zur herstellung von 1-substituierten 5-chlor-4methylpyrazolen
DE69620244T2 (de)	2002-10-24	Verfahren zur herstellung von prostaglandin e1
DE69712474T2 (de)	2003-01-16	Verfahren zur Herstellung von Diphosphonat-Derivaten
YU49004B (sh)	2003-04-30	LANOSTA-7,9-DIEN-3Гџ, 32-DIOL I POSTUPAK ZA NJEGOVO DOBIJANJE
ATE244217T1 (de)	2003-07-15	Herstellung von beta-mehtylcarbapenem- zwischenprodukten