NO20081167L - Fluoriseringsframgangsmate - Google Patents
FluoriseringsframgangsmateInfo
- Publication number
- NO20081167L NO20081167L NO20081167A NO20081167A NO20081167L NO 20081167 L NO20081167 L NO 20081167L NO 20081167 A NO20081167 A NO 20081167A NO 20081167 A NO20081167 A NO 20081167A NO 20081167 L NO20081167 L NO 20081167L
- Authority
- NO
- Norway
- Prior art keywords
- formula
- compound
- alkyl
- precursors
- fluoride
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
- C07C209/68—Preparation of compounds containing amino groups bound to a carbon skeleton from amines, by reactions not involving amino groups, e.g. reduction of unsaturated amines, aromatisation, or substitution of the carbon skeleton
- C07C209/74—Preparation of compounds containing amino groups bound to a carbon skeleton from amines, by reactions not involving amino groups, e.g. reduction of unsaturated amines, aromatisation, or substitution of the carbon skeleton by halogenation, hydrohalogenation, dehalogenation, or dehydrohalogenation
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C17/00—Preparation of halogenated hydrocarbons
- C07C17/093—Preparation of halogenated hydrocarbons by replacement by halogens
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
- A61K51/041—Heterocyclic compounds
- A61K51/044—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
- A61K51/0453—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J19/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
- B01J19/24—Stationary reactors without moving elements inside
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C211/00—Compounds containing amino groups bound to a carbon skeleton
- C07C211/43—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
- C07C211/44—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to only one six-membered aromatic ring
- C07C211/45—Monoamines
- C07C211/46—Aniline
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/64—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2
- C07D277/66—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2 with aromatic rings or ring systems directly attached in position 2
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
- B01J2219/24—Stationary reactors without moving elements inside
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Optics & Photonics (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- Physics & Mathematics (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
Oppfinnelsen angår en framgangsmåte for framstilling av en forbindelse av formel (I): der R1 er valgt blant C1-6-alkyl, C2-6-alkenyl, og C2-6-alkynyl, som omfatter: (i) reaksjon mellom fluorid, gjerne [18F]fluorid, og en tilsvarende forbindelse av formel (II): der R2 er valgt blant hydrogen, C1-10-alkyl, C1-10-halogenalkyl, C6-14-aryl, C6-14-arylalkyl, -(CH2CH2O)q-CH3 der q er et heltall fra 1 til 10, R1 er som definert for forbindelsen av formel (I), og R3 er en utgående gruppe. Visse nye forløpere av formel (II) og radiofarmasøytiske sett som inneholder slike forløpere er også omfattet av oppfinnelsen.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0516564.2A GB0516564D0 (en) | 2005-08-12 | 2005-08-12 | Fluorination process |
PCT/GB2006/003009 WO2007020400A1 (en) | 2005-08-12 | 2006-08-11 | Fluorination process of anilide derivatives and benzothiazole fluorinate derivatives as in vivo imaging agents |
Publications (2)
Publication Number | Publication Date |
---|---|
NO20081167L true NO20081167L (no) | 2008-03-05 |
NO341560B1 NO341560B1 (no) | 2017-12-04 |
Family
ID=35098197
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20081167A NO341560B1 (no) | 2005-08-12 | 2008-03-05 | Fluorineringsframgangsmåter, nye forbindelser, samt radiofarmasøytiske sett og kassetter |
Country Status (21)
Country | Link |
---|---|
US (3) | US8410312B2 (no) |
EP (1) | EP1915330B1 (no) |
JP (2) | JP5566605B2 (no) |
KR (2) | KR101409608B1 (no) |
CN (2) | CN101282920B (no) |
AU (1) | AU2006281216B2 (no) |
BR (1) | BRPI0614752B1 (no) |
CA (1) | CA2618448C (no) |
DK (1) | DK1915330T3 (no) |
ES (1) | ES2527864T3 (no) |
GB (1) | GB0516564D0 (no) |
HK (1) | HK1177463A1 (no) |
IL (1) | IL188933A0 (no) |
MX (2) | MX2008002068A (no) |
NO (1) | NO341560B1 (no) |
NZ (1) | NZ565333A (no) |
PL (1) | PL1915330T3 (no) |
PT (1) | PT1915330E (no) |
RU (1) | RU2419601C2 (no) |
WO (1) | WO2007020400A1 (no) |
ZA (1) | ZA200801860B (no) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0516564D0 (en) * | 2005-08-12 | 2005-09-21 | Ge Healthcare Ltd | Fluorination process |
US20100150835A1 (en) * | 2007-02-27 | 2010-06-17 | Bengt Langstrom | Synthesis of [18F] Fluoromethyl Benzene Using Benzyl Pentafluorobenzenesulfonate |
BRPI0815129B8 (pt) * | 2007-08-30 | 2021-05-25 | Ge Healthcare Ltd | composição radiofarmacêutica, e, métodos para preparação de uma composição radiofarmacêutica |
RU2475448C2 (ru) | 2008-01-03 | 2013-02-20 | ДжиИ ХЕЛТКЕР ЛИМИТЕД | Способ обработки фторида |
CA2737028C (en) | 2008-09-23 | 2017-06-27 | Wista Laboratories Ltd. | Ligands for aggregated tau molecules |
GB0921967D0 (en) * | 2009-12-17 | 2010-02-03 | Ge Healthcare Ltd | Novel Aryloxyanilide Derivatives |
GB201019303D0 (en) | 2010-11-15 | 2010-12-29 | Strom Hans E P | Agents and methods for visualising analytes |
CN103613589B (zh) * | 2013-11-29 | 2016-03-30 | 江苏华益科技有限公司 | 一种用于神经退行性疾病领域的新型pet显像剂前体及标准品的合成方法 |
CN106999603B (zh) | 2014-12-04 | 2022-05-27 | 通用电气健康护理有限公司 | 从放射性药物中除去乙醛的方法 |
JP6485914B2 (ja) * | 2015-10-28 | 2019-03-20 | 日本メジフィジックス株式会社 | フルテメタモルの製造方法 |
JP6955347B2 (ja) | 2017-02-28 | 2021-10-27 | 日本メジフィジックス株式会社 | フルテメタモルの製造方法 |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3878206A (en) * | 1973-06-06 | 1975-04-15 | Morton Norwich Products Inc | 9-(Substituted amino)imidazo{8 4,5-f{9 quinolines |
FR2449677B1 (fr) | 1979-02-26 | 1986-03-28 | Fabre Sa Pierre | Nouveaux derives de benzoyl-2 glycylanilides substitues, leur preparation et leur application en tant que medicaments anxiolytiques |
FR2693781B1 (fr) * | 1992-07-15 | 1994-10-28 | Otis Elevator Co | Dispositif de réglage de la tension d'un câble faisant boucle. |
DE4402056A1 (de) | 1994-01-25 | 1995-07-27 | Basf Ag | p-Phenylendiamin-Derivate und sie enthaltende fungizide Mittel |
US7270800B2 (en) * | 2000-08-24 | 2007-09-18 | University Of Pittsburgh | Thioflavin derivatives for use in antemortem diagnosis of Alzheimer's disease and in vivo imaging and prevention of amyloid deposition |
GB0229686D0 (en) * | 2002-12-20 | 2003-01-29 | Amersham Plc | Solid-phase fluorination of benzothiazoles |
PL1611115T3 (pl) * | 2003-03-14 | 2013-01-31 | Univ Pittsburgh Commonwealth Sys Higher Education | Związki pochodne benzotiazolu, kompozycje i zastosowania |
CA2438032C (en) * | 2003-03-14 | 2013-05-07 | University Of Pittsburgh | Benzothiazole derivative compounds, compositions and uses |
ES2427963T3 (es) * | 2004-07-02 | 2013-11-05 | University Of Pittsburgh - Of The Commonwealth System Of Higher Education | Uso de derivados de tioflavina radiomarcados en formación de imágenes de amiloide para evaluación de las terapias antiamiloide |
GB0516564D0 (en) * | 2005-08-12 | 2005-09-21 | Ge Healthcare Ltd | Fluorination process |
-
2005
- 2005-08-12 GB GBGB0516564.2A patent/GB0516564D0/en not_active Ceased
-
2006
- 2006-08-11 JP JP2008525644A patent/JP5566605B2/ja active Active
- 2006-08-11 PL PL06765263T patent/PL1915330T3/pl unknown
- 2006-08-11 CN CN200680037139.7A patent/CN101282920B/zh active Active
- 2006-08-11 AU AU2006281216A patent/AU2006281216B2/en active Active
- 2006-08-11 KR KR1020137025584A patent/KR101409608B1/ko active IP Right Grant
- 2006-08-11 PT PT67652636T patent/PT1915330E/pt unknown
- 2006-08-11 US US12/063,470 patent/US8410312B2/en active Active
- 2006-08-11 ES ES06765263.6T patent/ES2527864T3/es active Active
- 2006-08-11 BR BRPI0614752-6A patent/BRPI0614752B1/pt active IP Right Grant
- 2006-08-11 MX MX2008002068A patent/MX2008002068A/es active IP Right Grant
- 2006-08-11 RU RU2008103989/04A patent/RU2419601C2/ru active
- 2006-08-11 EP EP06765263.6A patent/EP1915330B1/en active Active
- 2006-08-11 CN CN201210177977.1A patent/CN102731432B/zh active Active
- 2006-08-11 NZ NZ565333A patent/NZ565333A/en unknown
- 2006-08-11 DK DK06765263.6T patent/DK1915330T3/en active
- 2006-08-11 WO PCT/GB2006/003009 patent/WO2007020400A1/en active Application Filing
- 2006-08-11 MX MX2013013741A patent/MX341173B/es unknown
- 2006-08-11 CA CA2618448A patent/CA2618448C/en active Active
-
2008
- 2008-01-22 IL IL188933A patent/IL188933A0/en active IP Right Grant
- 2008-02-11 KR KR1020087003263A patent/KR101392538B1/ko active Protection Beyond IP Right Term
- 2008-02-27 ZA ZA200801860A patent/ZA200801860B/xx unknown
- 2008-03-05 NO NO20081167A patent/NO341560B1/no unknown
-
2013
- 2013-03-22 US US13/848,877 patent/US9126961B2/en active Active
- 2013-04-17 HK HK13104661.5A patent/HK1177463A1/zh unknown
- 2013-09-24 JP JP2013196384A patent/JP2014028837A/ja not_active Withdrawn
-
2015
- 2015-07-27 US US14/809,497 patent/US9468694B2/en active Active
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
NO20081167L (no) | Fluoriseringsframgangsmate | |
TW200503724A (en) | Novel pharmaceuticals | |
MX2009013591A (es) | Proceso para la preparacion de pirazoles. | |
TW200510381A (en) | Novel 2-pyridinecarboxamide derivatives | |
MX2008010481A (es) | Compuestos que tienen afinado para el receptor f-ht6. | |
WO2006135641A3 (en) | PROCESS FOR THE SYNTHESIS OF 5- (METHYL-lH-IMIDAZOL-l-YL) -3- (TRI FLUOROME TH YL) -BENZENEAMINE | |
NO20091626L (no) | MGLUR5-modulatorer | |
MX2009004343A (es) | Compuestos organicos. | |
WO2005070884A3 (en) | Heterocyclic compounds useful as growth hormone secretagogues | |
NO20071242L (no) | Triazolpyridinylsulfanylderivater som P38-MAP-kinaseinhibitorer | |
NO20082116L (no) | Kjemisk fremgangsmate for fremstilling av en amido-fenoksybenzosyreforbindelse | |
NO20071012L (no) | Fremgangsmate for fremstilling av D-erytro-2,2-difluor-2-deoksy-1-oksoribosederivat | |
NO20091575L (no) | Hoyenhets massetilberedning av stannsoporfin | |
SG153856A1 (en) | Chemical process | |
NO20071253L (no) | Fremgangsmate for syntese av C-2, C-3 substituerte N-alkylerte indoler anvendbare som CPLA2-inhibitorer. | |
TW200619201A (en) | Process for the preparation of pyrazoles | |
WO2008103367A3 (en) | Method for assembling high-purity chemical libraries, proapoptotic compounds discovered by same | |
NO20076161L (no) | Fremgangsmater for fremstilling av 4-bifenylazetidin-2-oner | |
GB0327323D0 (en) | Novel pharmaceuticals | |
GB0215392D0 (en) | Chemical compounds | |
MX2010001512A (es) | Nuevo procedimiento de preparacion. | |
NO20052197L (no) | Fremgangsmate for fremstilling av pyrazol | |
IN2012DN02871A (no) | ||
NO20092210L (no) | Salter av dihydroksyantrakinon-karboksylsyrer og deres terapeutiske anvendelse | |
NO20073213L (no) | Fremgangsmate for fremstilling av tiofenglykosidderivater |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
CREP | Change of representative |
Representative=s name: ZACCO NORWAY AS, POSTBOKS 2003 VIKA |