NO20071095L - Hittil ukjente tiofenderivater - Google Patents

Hittil ukjente tiofenderivater

Info

Publication number
NO20071095L
NO20071095L NO20071095A NO20071095A NO20071095L NO 20071095 L NO20071095 L NO 20071095L NO 20071095 A NO20071095 A NO 20071095A NO 20071095 A NO20071095 A NO 20071095A NO 20071095 L NO20071095 L NO 20071095L
Authority
NO
Norway
Prior art keywords
thiophene derivatives
hitherto unknown
derivatives
hitherto
unknown
Prior art date
Application number
NO20071095A
Other languages
English (en)
Norwegian (no)
Inventor
Martin Bolli
Thomas Weller
Walter Fischli
Martine Clozel
Oliver Nayler
Daniel Bur
Claus Mueller
Michael Scherz
David Lehmann
Boris Mathys
Original Assignee
Actelion Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Actelion Pharmaceuticals Ltd filed Critical Actelion Pharmaceuticals Ltd
Publication of NO20071095L publication Critical patent/NO20071095L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/78Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems condensed with rings other than six-membered or with ring systems containing such rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/14Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Immunology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Transplantation (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
NO20071095A 2004-07-29 2007-02-27 Hittil ukjente tiofenderivater NO20071095L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
PCT/EP2004/008501 WO2006010379A1 (fr) 2004-07-29 2004-07-29 Nouveaux derives du thiophene utilises comme agents immunosupresseurs
PCT/EP2005/007892 WO2006010544A2 (fr) 2004-07-29 2005-07-20 Nouveaux derives du thiophene

Publications (1)

Publication Number Publication Date
NO20071095L true NO20071095L (no) 2007-02-27

Family

ID=34958296

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20071095A NO20071095L (no) 2004-07-29 2007-02-27 Hittil ukjente tiofenderivater

Country Status (23)

Country Link
US (1) US7750040B2 (fr)
EP (1) EP1805163B1 (fr)
JP (1) JP4807884B2 (fr)
KR (1) KR20070046849A (fr)
CN (1) CN1993346B (fr)
AR (1) AR050273A1 (fr)
AT (1) ATE409697T1 (fr)
AU (1) AU2005266529A1 (fr)
BR (1) BRPI0513841A (fr)
CA (1) CA2574305A1 (fr)
DE (1) DE602005010109D1 (fr)
DK (1) DK1805163T3 (fr)
ES (1) ES2313391T3 (fr)
IL (1) IL180962A0 (fr)
MX (1) MX2007000972A (fr)
NO (1) NO20071095L (fr)
PL (1) PL1805163T3 (fr)
PT (1) PT1805163E (fr)
RU (1) RU2386626C2 (fr)
SI (1) SI1805163T1 (fr)
TW (1) TW200616994A (fr)
WO (2) WO2006010379A1 (fr)
ZA (1) ZA200700535B (fr)

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BRPI0609668A2 (pt) 2005-03-23 2011-10-18 Actelion Pharmaceuticals Ltd composto, composição farmacêutica, e, uso de um composto
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CN101180290B (zh) * 2005-03-23 2012-12-12 埃科特莱茵药品有限公司 氢化苯并〔c〕噻吩衍生物作为免疫调节剂
RU2008101805A (ru) * 2005-06-24 2009-07-27 Актелион Фармасьютиклз Лтд (Ch) Новые производные тиофена
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TWI404706B (zh) * 2006-01-11 2013-08-11 Actelion Pharmaceuticals Ltd 新穎噻吩衍生物
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TWI408139B (zh) * 2006-09-07 2013-09-11 Actelion Pharmaceuticals Ltd 新穎噻吩衍生物
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ES2389042T3 (es) * 2008-03-06 2012-10-22 Actelion Pharmaceuticals Ltd. Compuestos de piridina
BRPI0909055A2 (pt) * 2008-03-07 2019-02-26 Actelion Pharmaceuticals Ltd composto derivado de piridin-2-il, composição farmacêutica que o contém e uso desse composto.
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DE102014222629A1 (de) 2014-11-05 2016-05-12 Carl Zeiss Meditec Ag Untersuchen eines Objekts mit OCT-Abtastlichtstrahlen
DE202014011051U1 (de) 2014-11-05 2017-07-26 Carl Zeiss Meditec Ag Vorrichtung für das Untersuchen eines Patientenauges
DE202014011050U1 (de) 2014-11-05 2017-07-26 Carl Zeiss Meditec Ag Vorrichtung für das Untersuchen eines Patientenauges
MX2017008925A (es) 2015-01-06 2017-10-11 Arena Pharm Inc Metodos de condiciones de tratamiento relacionadas con el receptor s1p1.
US10385043B2 (en) 2015-05-20 2019-08-20 Idorsia Pharmaceuticals Ltd Crystalline form of the compound (S)-3-{4-[5-(2-cyclopentyl-6-methoxy-pyridin-4-yl)-[1,2,4]oxadiazol-3-yl]-2-ethyl-6-methyl-phenoxy}-propane-1,2-diol
US10111841B2 (en) 2015-06-19 2018-10-30 University Of South Florida Stabilization of alcohol intoxication-induced cardiovascular instability
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JP2020507610A (ja) 2017-02-16 2020-03-12 アリーナ ファーマシューティカルズ, インコーポレイテッド 腸管外症状を伴う炎症性腸疾患の治療のための化合物および方法
JP2020507611A (ja) 2017-02-16 2020-03-12 アリーナ ファーマシューティカルズ, インコーポレイテッド 原発性胆汁性胆管炎の治療のための化合物および方法
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Also Published As

Publication number Publication date
RU2386626C2 (ru) 2010-04-20
PL1805163T3 (pl) 2009-04-30
CN1993346B (zh) 2011-04-27
JP4807884B2 (ja) 2011-11-02
AR050273A1 (es) 2006-10-11
SI1805163T1 (sl) 2009-02-28
KR20070046849A (ko) 2007-05-03
US7750040B2 (en) 2010-07-06
CN1993346A (zh) 2007-07-04
AU2005266529A1 (en) 2006-02-02
DE602005010109D1 (de) 2008-11-13
US20080064740A1 (en) 2008-03-13
BRPI0513841A (pt) 2008-05-20
WO2006010379A1 (fr) 2006-02-02
DK1805163T3 (da) 2008-12-15
ATE409697T1 (de) 2008-10-15
ZA200700535B (en) 2008-10-29
IL180962A0 (en) 2007-07-04
ES2313391T3 (es) 2009-03-01
TW200616994A (en) 2006-06-01
WO2006010544A3 (fr) 2006-03-30
CA2574305A1 (fr) 2006-02-02
PT1805163E (pt) 2008-12-05
WO2006010544A2 (fr) 2006-02-02
MX2007000972A (es) 2007-04-10
JP2008508210A (ja) 2008-03-21
EP1805163A2 (fr) 2007-07-11
RU2007107164A (ru) 2008-09-10
EP1805163B1 (fr) 2008-10-01

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