NO174206C - Fremgangsmåte til fremstilling av deoksyfluornukleorider, samt utgangsmaterialer til fremstilling av slike - Google Patents
Fremgangsmåte til fremstilling av deoksyfluornukleorider, samt utgangsmaterialer til fremstilling av slikeInfo
- Publication number
- NO174206C NO174206C NO904870A NO904870A NO174206C NO 174206 C NO174206 C NO 174206C NO 904870 A NO904870 A NO 904870A NO 904870 A NO904870 A NO 904870A NO 174206 C NO174206 C NO 174206C
- Authority
- NO
- Norway
- Prior art keywords
- nucleorides
- deoxyfluoro
- preparing
- preparation
- starting materials
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/16—Purine radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H1/00—Processes for the preparation of sugar derivatives
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US43585289A | 1989-11-13 | 1989-11-13 |
Publications (4)
Publication Number | Publication Date |
---|---|
NO904870D0 NO904870D0 (no) | 1990-11-09 |
NO904870L NO904870L (no) | 1991-05-14 |
NO174206B NO174206B (no) | 1993-12-20 |
NO174206C true NO174206C (no) | 1994-04-06 |
Family
ID=23730082
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO904870A NO174206C (no) | 1989-11-13 | 1990-11-09 | Fremgangsmåte til fremstilling av deoksyfluornukleorider, samt utgangsmaterialer til fremstilling av slike |
Country Status (12)
Country | Link |
---|---|
EP (1) | EP0428109A3 (no) |
JP (1) | JPH03170496A (no) |
KR (1) | KR910009717A (no) |
AU (1) | AU6596590A (no) |
CA (1) | CA2029301A1 (no) |
FI (1) | FI905536A0 (no) |
HU (4) | HU906976D0 (no) |
IE (1) | IE904070A1 (no) |
IL (1) | IL96306A0 (no) |
NO (1) | NO174206C (no) |
PT (1) | PT95861A (no) |
ZA (1) | ZA909042B (no) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
UA41261C2 (uk) * | 1992-06-22 | 2001-09-17 | Елі Ліллі Енд Компані | Спосіб одержання збагачених бета-аномером нуклеозидів |
US5426183A (en) * | 1992-06-22 | 1995-06-20 | Eli Lilly And Company | Catalytic stereoselective glycosylation process for preparing 2'-deoxy-2',2'-difluoronucleosides and 2'-deoxy-2'-fluoronucleosides |
US5821357A (en) * | 1992-06-22 | 1998-10-13 | Eli Lilly And Company | Stereoselective glycosylation process for preparing 2'-deoxy-2',2'-difluoropurine and triazole nucleosides |
AU659009B2 (en) * | 1992-06-22 | 1995-05-04 | Eli Lilly And Company | Stereoselective glycosylation process |
US5401838A (en) * | 1992-06-22 | 1995-03-28 | Eli Lilly And Company | Stereoselective fusion glycosylation process for preparing 2'-deoxy-2',2'-difluoronucleosides and 2'-deoxy-2'-fluoronucleosides |
SG94686A1 (en) * | 1992-06-22 | 2003-03-18 | Lilly Co Eli | Stereoselective gylcosylation process |
JPH0673086A (ja) * | 1992-06-22 | 1994-03-15 | Eli Lilly & Co | 立体選択的な陰イオングリコシル化法 |
US5371210A (en) * | 1992-06-22 | 1994-12-06 | Eli Lilly And Company | Stereoselective fusion glycosylation process for preparing 2'-deoxy-2',2'-difluoronucleosides and 2'-deoxy-2'-fluoronucleosides |
AU659008B2 (en) * | 1992-06-22 | 1995-05-04 | Eli Lilly And Company | Stereoselective anion glycosylation process |
US5594124A (en) * | 1992-06-22 | 1997-01-14 | Eli Lilly And Company | Stereoselective glycosylation process for preparing 2'-Deoxy-2',2'-difluoropyrimidine nucleosides and 2'-deoxy-2'-fluoropyrimidine nucleosides and intermediates thereof |
US5606048A (en) * | 1992-06-22 | 1997-02-25 | Eli Lilly And Company | Stereoselective glycosylation process for preparing 2'-Deoxy-2', 2'-difluoronucleosides and 2'-deoxy-2'-fluoronucleosides |
US5424416A (en) * | 1993-08-25 | 1995-06-13 | Eli Lilly And Company | Process for preparation of 2-deoxy-2,2-difluoro-D-ribofuranosyl-3,5-hydroxy protected-1-alkyl and aryl sulfonates and their use in preparation of 2',2'-difluoro-2'-deoxy nucleosides |
AT400953B (de) * | 1994-08-25 | 1996-05-28 | Joern Saischek | Pentofuranosid-derivate, deren herstellung und verwendung |
JPH11217396A (ja) * | 1998-01-30 | 1999-08-10 | Ajinomoto Co Inc | ヌクレオシド誘導体の製造方法 |
US6949640B2 (en) * | 2000-02-18 | 2005-09-27 | Southern Research Institute | Method for synthesizing 2-chloro-9-(2-fluoro-β-D-arabinofuranosyl)-9H-purin-6-amine |
EP1412369B1 (en) | 2001-08-02 | 2008-05-07 | Ilex Oncology, Inc. | Process for preparing purine nucleosides |
EP3450438A1 (en) | 2011-05-19 | 2019-03-06 | Gilead Sciences, Inc. | Processes and intermediates for preparing anti-hiv agents |
SI3661937T1 (sl) | 2017-08-01 | 2021-11-30 | Gilead Sciences, Inc. | Kristalinične oblike etil((S)-((((2R,5R)-5-(6-amino-9H-purin-9-IL)-4- fluoro-2,5-dihidrofuran-2-IL)oksi)metil)(fenoksi)fosforil)-L-alaninata (GS-9131) za zdravljenje virusnih okužb |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4751221A (en) * | 1985-10-18 | 1988-06-14 | Sloan-Kettering Institute For Cancer Research | 2-fluoro-arabinofuranosyl purine nucleosides |
CA1340645C (en) * | 1987-04-17 | 1999-07-13 | Victor E. Marquez | Acid stable dideoxynucleosides active against the cytopathic effects of human immunodeficiency virus |
NZ226672A (en) * | 1987-10-30 | 1991-07-26 | Hoffmann La Roche | 6-amino-9-(2,3-dideoxy-2-fluoro-b-d-threopentofuranosyl)-9h-purine derivatives and pharmaceutical compositions |
GB8816345D0 (en) * | 1988-07-08 | 1988-08-10 | Hoffmann La Roche | Purine derivatives |
-
1990
- 1990-11-01 HU HU906976A patent/HU906976D0/hu unknown
- 1990-11-05 CA CA002029301A patent/CA2029301A1/en not_active Abandoned
- 1990-11-08 FI FI905536A patent/FI905536A0/fi not_active IP Right Cessation
- 1990-11-09 NO NO904870A patent/NO174206C/no unknown
- 1990-11-12 AU AU65965/90A patent/AU6596590A/en not_active Abandoned
- 1990-11-12 KR KR1019900018266A patent/KR910009717A/ko not_active Application Discontinuation
- 1990-11-12 IL IL96306A patent/IL96306A0/xx unknown
- 1990-11-12 PT PT95861A patent/PT95861A/pt not_active Application Discontinuation
- 1990-11-12 IE IE407090A patent/IE904070A1/en unknown
- 1990-11-12 EP EP19900121636 patent/EP0428109A3/en not_active Withdrawn
- 1990-11-12 ZA ZA909042A patent/ZA909042B/xx unknown
- 1990-11-13 HU HU907113A patent/HU208149B/hu not_active IP Right Cessation
- 1990-11-13 JP JP2304179A patent/JPH03170496A/ja active Pending
- 1990-11-13 HU HU9303049A patent/HU9303049D0/hu unknown
- 1990-11-13 HU HU9303048A patent/HU9303048D0/hu unknown
Also Published As
Publication number | Publication date |
---|---|
KR910009717A (ko) | 1991-06-28 |
PT95861A (pt) | 1991-09-13 |
HU906976D0 (en) | 1991-05-28 |
FI905536A0 (fi) | 1990-11-08 |
JPH03170496A (ja) | 1991-07-24 |
AU6596590A (en) | 1991-05-16 |
NO904870L (no) | 1991-05-14 |
EP0428109A3 (en) | 1991-09-11 |
HU9303049D0 (en) | 1994-01-28 |
IE904070A1 (en) | 1991-05-22 |
NO174206B (no) | 1993-12-20 |
NO904870D0 (no) | 1990-11-09 |
HUT57790A (en) | 1991-12-30 |
HU208149B (en) | 1993-08-30 |
CA2029301A1 (en) | 1991-05-14 |
EP0428109A2 (en) | 1991-05-22 |
HU907113D0 (en) | 1991-05-28 |
HU9303048D0 (en) | 1994-01-28 |
ZA909042B (en) | 1991-09-25 |
IL96306A0 (en) | 1991-08-16 |
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