NL180317B - PROCESS FOR PREPARING PENICILLANIC ACID-1,1-DIOXIDE AND ITS ESTERS AND PHARMACEUTICALLY ACCEPTABLE SALTS OF THE PENICILLANIC ACID-1,1-DIOXIDE. - Google Patents

PROCESS FOR PREPARING PENICILLANIC ACID-1,1-DIOXIDE AND ITS ESTERS AND PHARMACEUTICALLY ACCEPTABLE SALTS OF THE PENICILLANIC ACID-1,1-DIOXIDE.

Info

Publication number
NL180317B
NL180317B NLAANVRAGE8001285,A NL8001285A NL180317B NL 180317 B NL180317 B NL 180317B NL 8001285 A NL8001285 A NL 8001285A NL 180317 B NL180317 B NL 180317B
Authority
NL
Netherlands
Prior art keywords
dioxide
penicillanic acid
esters
pharmaceutically acceptable
acceptable salts
Prior art date
Application number
NLAANVRAGE8001285,A
Other languages
Dutch (nl)
Other versions
NL180317C (en
NL8001285A (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of NL8001285A publication Critical patent/NL8001285A/en
Publication of NL180317B publication Critical patent/NL180317B/en
Application granted granted Critical
Publication of NL180317C publication Critical patent/NL180317C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
NLAANVRAGE8001285,A 1979-03-05 1980-03-04 PROCESS FOR PREPARING PENICILLANIC ACID-1,1-DIOXIDE AND ITS ESTERS AND PHARMACEUTICALLY ACCEPTABLE SALTS OF THE PENICILLANIC ACID-1,1-DIOXIDE. NL180317C (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US1781079A 1979-03-05 1979-03-05
US1780879A 1979-03-05 1979-03-05
US1781079 1979-03-05
US1780879 1979-03-05

Publications (3)

Publication Number Publication Date
NL8001285A NL8001285A (en) 1980-09-09
NL180317B true NL180317B (en) 1986-09-01
NL180317C NL180317C (en) 1987-02-02

Family

ID=26690337

Family Applications (1)

Application Number Title Priority Date Filing Date
NLAANVRAGE8001285,A NL180317C (en) 1979-03-05 1980-03-04 PROCESS FOR PREPARING PENICILLANIC ACID-1,1-DIOXIDE AND ITS ESTERS AND PHARMACEUTICALLY ACCEPTABLE SALTS OF THE PENICILLANIC ACID-1,1-DIOXIDE.

Country Status (36)

Country Link
KR (1) KR850001339B1 (en)
AR (1) AR225031A1 (en)
AT (1) AT366693B (en)
AU (1) AU522572B2 (en)
BG (1) BG33292A3 (en)
CH (1) CH644608A5 (en)
CS (1) CS215130B2 (en)
DD (1) DD149367A5 (en)
DE (1) DE3008257C2 (en)
DK (2) DK159852C (en)
EG (1) EG14437A (en)
ES (1) ES8103094A1 (en)
FI (1) FI70024C (en)
FR (1) FR2450836B1 (en)
GB (1) GB2045755B (en)
GR (1) GR67234B (en)
HK (1) HK66587A (en)
HU (1) HU186304B (en)
IE (1) IE49535B1 (en)
IL (1) IL59515A (en)
IN (1) IN153685B (en)
IT (1) IT1130300B (en)
KE (1) KE3464A (en)
LU (1) LU82215A1 (en)
MX (1) MX6032E (en)
MY (1) MY8500319A (en)
NL (1) NL180317C (en)
NO (2) NO800618L (en)
PL (1) PL125197B1 (en)
PT (1) PT70897A (en)
RO (1) RO80112A (en)
SE (2) SE449103B (en)
SG (1) SG55884G (en)
SU (1) SU1192626A3 (en)
UA (1) UA6342A1 (en)
YU (1) YU42328B (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4419284A (en) * 1981-03-23 1983-12-06 Pfizer Inc. Preparation of halomethyl esters (and related esters) of penicillanic acid 1,1-dioxide
IN159362B (en) * 1981-03-23 1987-05-09 Pfizer
PT76526B (en) * 1982-04-19 1986-01-21 Gist Brocades Nv Preparation of 6-alpha-bromo- and/or 6,6-dibromopenicillanic acid 1,1-dioxides
IT1190897B (en) * 1982-06-29 1988-02-24 Opos Biochimica Srl PROCEDURE FOR THE PREPARATION OF THE 1-ETHOXYCARBONYLOXYETHYL ACID ACID 6- (D (-) - ALPHA AMINOALPHA-PHENYLACETAMIDE) -PENICILLANIC
US4606865A (en) * 1982-09-20 1986-08-19 Astra Lakemedel Aktiebolag Methods for the preparation of α-bromodiethylcarbonate
EP0139047A1 (en) * 1983-10-18 1985-05-02 Gist-Brocades N.V. Process for the preparation of 6,6-dibromopenicillanic acid 1,1-dioxide
EP0139048A1 (en) * 1983-10-18 1985-05-02 Gist-Brocades N.V. Process for the dehalogenation of 6,6-dibromopenicillanic acid 1,1-dioxide
US4596677A (en) * 1984-04-06 1986-06-24 Bristol-Myers Company Anhydropenicillin intermediates

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN149747B (en) * 1977-06-07 1982-04-03 Pfizer
CA1158639A (en) * 1978-12-11 1983-12-13 Eric M. Gordon 6-bromopenicillanic acid sulfone
DE3068390D1 (en) * 1979-01-10 1984-08-09 Beecham Group Plc Penicillin derivatives, process for their preparation and pharmaceutical compositions containing certain of these compounds
IE49881B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd B-lactam intermediates

Also Published As

Publication number Publication date
GB2045755A (en) 1980-11-05
GR67234B (en) 1981-06-25
IE49535B1 (en) 1985-10-16
AT366693B (en) 1982-04-26
SG55884G (en) 1985-03-08
DK159852C (en) 1991-05-06
EG14437A (en) 1984-09-30
PT70897A (en) 1980-04-01
FI800661A (en) 1980-09-06
DK145690D0 (en) 1990-06-14
SE8603309D0 (en) 1986-08-04
ATA119080A (en) 1981-09-15
RO80112A (en) 1982-10-26
LU82215A1 (en) 1980-09-24
SE8603309L (en) 1986-08-04
SE449103B (en) 1987-04-06
HK66587A (en) 1987-09-25
AR225031A1 (en) 1982-02-15
ES489185A0 (en) 1981-02-16
DK166353B (en) 1993-04-13
NO823127L (en) 1980-09-08
IT8020367A0 (en) 1980-03-05
IE800429L (en) 1980-09-05
YU42328B (en) 1988-08-31
IT1130300B (en) 1986-06-11
UA6342A1 (en) 1994-12-29
BG33292A3 (en) 1983-01-14
ES8103094A1 (en) 1981-02-16
AU5610480A (en) 1980-09-11
MY8500319A (en) 1985-12-31
DK166353C (en) 1993-09-06
DE3008257A1 (en) 1980-09-11
NL180317C (en) 1987-02-02
FR2450836B1 (en) 1986-03-21
FI70024C (en) 1986-09-12
IN153685B (en) 1984-08-04
KE3464A (en) 1984-10-12
DK145690A (en) 1990-06-14
MX6032E (en) 1984-10-04
DD149367A5 (en) 1981-07-08
DE3008257C2 (en) 1984-03-01
IL59515A (en) 1983-02-23
NL8001285A (en) 1980-09-09
SU1192626A3 (en) 1985-11-15
IL59515A0 (en) 1980-06-30
CH644608A5 (en) 1984-08-15
FI70024B (en) 1986-01-31
HU186304B (en) 1985-07-29
DK92680A (en) 1980-09-06
FR2450836A1 (en) 1980-10-03
PL125197B1 (en) 1983-04-30
DK159852B (en) 1990-12-17
SE8000512L (en) 1980-09-06
KR850001339B1 (en) 1985-09-19
PL222448A1 (en) 1981-01-02
YU58580A (en) 1983-02-28
AU522572B2 (en) 1982-06-17
CS215130B2 (en) 1982-07-30
NO800618L (en) 1980-09-08
GB2045755B (en) 1983-01-26

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Legal Events

Date Code Title Description
A1A A request for search or an international-type search has been filed
BB A search report has been drawn up
BC A request for examination has been filed
A85 Still pending on 85-01-01
V4 Discontinued because of reaching the maximum lifetime of a patent

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