MXPA03004166A - Nuevos usos de combinaciones de agonistas de 5-ht1a e inhibidores de la recaptacion de serotonina. - Google Patents

Nuevos usos de combinaciones de agonistas de 5-ht1a e inhibidores de la recaptacion de serotonina.

Info

Publication number
MXPA03004166A
MXPA03004166A MXPA03004166A MXPA03004166A MXPA03004166A MX PA03004166 A MXPA03004166 A MX PA03004166A MX PA03004166 A MXPA03004166 A MX PA03004166A MX PA03004166 A MXPA03004166 A MX PA03004166A MX PA03004166 A MXPA03004166 A MX PA03004166A
Authority
MX
Mexico
Prior art keywords
ht1a
combined
novel uses
novel
Prior art date
Application number
MXPA03004166A
Other languages
English (en)
Inventor
Gerd Bartoszyk
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of MXPA03004166A publication Critical patent/MXPA03004166A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Indole Compounds (AREA)
MXPA03004166A 2000-11-14 2001-10-16 Nuevos usos de combinaciones de agonistas de 5-ht1a e inhibidores de la recaptacion de serotonina. MXPA03004166A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP00124815 2000-11-14
PCT/EP2001/011952 WO2002040024A1 (en) 2000-11-14 2001-10-16 Novel uses of combined 5-ht1a agonists and serotonin reuptake inhibitors

Publications (1)

Publication Number Publication Date
MXPA03004166A true MXPA03004166A (es) 2003-09-22

Family

ID=8170369

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA03004166A MXPA03004166A (es) 2000-11-14 2001-10-16 Nuevos usos de combinaciones de agonistas de 5-ht1a e inhibidores de la recaptacion de serotonina.

Country Status (22)

Country Link
US (1) US20040082594A1 (es)
EP (1) EP1333832B1 (es)
JP (1) JP2004513924A (es)
KR (1) KR20030059244A (es)
CN (1) CN1222291C (es)
AR (1) AR031335A1 (es)
AU (2) AU2002215027B2 (es)
BR (1) BR0115296A (es)
CA (1) CA2428511C (es)
CZ (1) CZ302484B6 (es)
DE (1) DE60131675T2 (es)
ES (1) ES2296820T3 (es)
HK (1) HK1060697A1 (es)
HU (1) HUP0302751A3 (es)
MX (1) MXPA03004166A (es)
NO (1) NO20032148D0 (es)
PL (1) PL204331B1 (es)
RU (1) RU2288719C2 (es)
SK (1) SK287337B6 (es)
UA (1) UA79583C2 (es)
WO (1) WO2002040024A1 (es)
ZA (1) ZA200304606B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10305739A1 (de) * 2003-02-11 2004-08-19 Merck Patent Gmbh Benzofuranderivate
PL1701940T3 (pl) 2003-12-23 2008-11-28 H Lundbeck As Pochodne 2-(1H-indolilosulfanylo)benzyloaminy jako SSRI
EP1732610A2 (en) 2004-03-26 2006-12-20 Baylor University Targeted serotonin reuptake inhibitors
AR052308A1 (es) 2004-07-16 2007-03-14 Lundbeck & Co As H Derivados de 2-(1h-indolilsulfanil)-arilamina y una composicion farmaceutica que contiene al compuesto
WO2006034788A1 (en) * 2004-09-28 2006-04-06 Merck Patent Gmbh Combinations of n-(indolecarbonyl-)piperazine derivatives and serotonin reuptake inhibitors
AR054393A1 (es) 2005-06-17 2007-06-20 Lundbeck & Co As H Derivados de benzo(b)furano y benzo(b)tiofeno, composiciones farmaceuticas que los contienen y su uso en la fabricacion de un medicamento para el tratamiento de enfermedades mediadas por la inhibicion de la reabsorcion de neurotransmisores de amina biogenicos.
US7629473B2 (en) 2005-06-17 2009-12-08 H. Lundbeck A/S 2-(1H-indolylsulfanyl)-aryl amine derivatives
EP2068863B1 (en) * 2006-08-11 2010-12-15 DSM IP Assets B.V. Ligustilide for the treatment of disorders of the central nervous system

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4333254A1 (de) * 1993-09-30 1995-04-06 Merck Patent Gmbh Piperidine und Piperazine
DE19512639A1 (de) * 1995-04-05 1996-10-10 Merck Patent Gmbh Benzonitrile und -fluoride
DE19637237A1 (de) * 1996-09-13 1998-03-19 Merck Patent Gmbh Piperazin-Derivate
DE19730989A1 (de) * 1997-07-18 1999-01-21 Merck Patent Gmbh Piperazin-Derivate
AU5033899A (en) * 1998-07-20 2000-02-14 Merck Patent Gmbh Biphenyl derivatives

Also Published As

Publication number Publication date
JP2004513924A (ja) 2004-05-13
PL360310A1 (en) 2004-09-06
ZA200304606B (en) 2004-09-13
CZ302484B6 (cs) 2011-06-08
CN1222291C (zh) 2005-10-12
DE60131675T2 (de) 2008-11-20
CA2428511A1 (en) 2002-05-23
HK1060697A1 (en) 2004-08-20
PL204331B1 (pl) 2010-01-29
SK287337B6 (sk) 2010-07-07
ES2296820T3 (es) 2008-05-01
EP1333832A1 (en) 2003-08-13
DE60131675D1 (de) 2008-01-10
WO2002040024A1 (en) 2002-05-23
HUP0302751A3 (en) 2007-06-28
AU1502702A (en) 2002-05-27
CN1474691A (zh) 2004-02-11
KR20030059244A (ko) 2003-07-07
CA2428511C (en) 2009-12-29
BR0115296A (pt) 2003-09-02
EP1333832B1 (en) 2007-11-28
NO20032148L (no) 2003-05-13
NO20032148D0 (no) 2003-05-13
HUP0302751A2 (hu) 2003-11-28
AU2002215027B2 (en) 2006-10-05
US20040082594A1 (en) 2004-04-29
AR031335A1 (es) 2003-09-17
RU2288719C2 (ru) 2006-12-10
UA79583C2 (en) 2007-07-10
CZ20031433A3 (cs) 2003-09-17
SK6382003A3 (en) 2003-11-04

Similar Documents

Publication Publication Date Title
ZA200204020B (en) Use of anti-CTLA-4-antibodies.
ZA200205479B (en) Novel biarylcarboxamides.
MXPA03007093A (es) Nueva composicion.
MXPA03007043A (es) Nueva sal de succinato de o-desmetil-venlafaxina.
HK1055955A1 (en) Methanesulphonamido-benzofuran, preparation methodand use thereof as synthesis intermediate.
ZA200206198B (en) New aza-indolyl derivatives.
MXPA03009558A (es) Compuestos novedosos.
MXPA03007834A (es) Uso de agonistas inversos de gabaa, en combinacion con agonistas parciales del receptor de nicotina, estrogenos, moduladores selectivos de estrogenos o vitamina e, para el tratamiento de transtornos cognitivos.
ZA200307102B (en) The use of enmantiomeric pure escitalopram.
EG23361A (en) High utility tissue.
EP1254140A4 (en) SAFRAMYCIN-ECTEINASCIDIN SERIES COMPOUNDS, USES AND SYNTHESIS
MXPA03006603A (es) Agonista de subtipo de receptor 5-ht1a.
MXPA03009698A (es) Vacuna multivalente que comprende un antigeno vih y un antigeno vsh y/o un antigeno vph.
MXPA03007693A (es) Composicion para la piel.
MXPA03008139A (es) Fluoralcoxifenilsulfonilureas sustituidas.
HK1050610A1 (en) Microemulsion aerosol composition.
MXPA03001991A (es) Novedosas arilalcano-sulfonamidas.
MXPA03000914A (es) Sintesis de (r)-3-(4 -bromobencil) -1-(3, 5-diclorofenil) -5-yodo-3 -metil-1-h -imidazo[1, 2-a]imidazol -2-ona.
MXPA03007314A (es) Composicion para la piel para reducir aceites y grasa de la piel.
EG23378A (en) Composition.
MXPA03004166A (es) Nuevos usos de combinaciones de agonistas de 5-ht1a e inhibidores de la recaptacion de serotonina.
MXPA03004341A (es) Nuevo uso de combinaciones de agonsitas de 5-ht1a e inhibidores selectivos de la recaptacion de serotonina.
GB0104554D0 (en) New uses
HK1066022A1 (en) Use of 1,1,1,3,3-pentafluorobutan
MXPA01000464A (es) Composicion.

Legal Events

Date Code Title Description
FG Grant or registration
GD Licence granted
GD Licence granted