MX9706912A - Inhibidores de protesa retroviral de sulfonamida de hidroxietilamino de amino acido y uso de los mismos. - Google Patents

Inhibidores de protesa retroviral de sulfonamida de hidroxietilamino de amino acido y uso de los mismos.

Info

Publication number
MX9706912A
MX9706912A MX9706912A MX9706912A MX9706912A MX 9706912 A MX9706912 A MX 9706912A MX 9706912 A MX9706912 A MX 9706912A MX 9706912 A MX9706912 A MX 9706912A MX 9706912 A MX9706912 A MX 9706912A
Authority
MX
Mexico
Prior art keywords
amino acid
protease inhibitors
retroviral
retroviral protease
protease
Prior art date
Application number
MX9706912A
Other languages
English (en)
Inventor
Daniel P Getman
Gary A Decrescenzo
John N Freskos
Michael L Vazquez
James A Sikorski
Balekudru Devadas
Srinivasan Nagarajan
David L Brown
Joseph J Macdonald
Original Assignee
Searle & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Searle & Co filed Critical Searle & Co
Priority claimed from PCT/US1996/002684 external-priority patent/WO1996028463A1/en
Publication of MX9706912A publication Critical patent/MX9706912A/es

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  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Compuestos de hidroxietilamino sulfonamida de amino ácido seleccionados son efectivos como inhibidores de protesa retroviral, y en particular como inhibidores de proteasa de VIH, y la presente invencion se refiere a dichos inhibidores de protesa retroviral y, más en particular, se refiere a compuestos novedosos seleccionados, a la composicion y el uso de los mismos en la preparacion de composiciones y medicamentos para inhibir las proteasas retrovirales, tales como protesa de virus de inmunodeficiencia humana (VIH), prevenir profilácticamente la infeccion retroviral o la expansion de un retrovirus, y el tratamiento de una infeccion retroviral.
MX9706912A 1996-03-07 1996-03-07 Inhibidores de protesa retroviral de sulfonamida de hidroxietilamino de amino acido y uso de los mismos. MX9706912A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US1996/002684 WO1996028463A1 (en) 1995-03-10 1996-03-07 Amino acid hydroxyethylamino sulfonamide retroviral protease inhibitors

Publications (1)

Publication Number Publication Date
MX9706912A true MX9706912A (es) 1998-01-31

Family

ID=39165645

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9706912A MX9706912A (es) 1996-03-07 1996-03-07 Inhibidores de protesa retroviral de sulfonamida de hidroxietilamino de amino acido y uso de los mismos.

Country Status (1)

Country Link
MX (1) MX9706912A (es)

Similar Documents

Publication Publication Date Title
MX9706913A (es) Compuestos de bis-aminacido-hidroxietilamina-sulfonamida inhibidoresde proteasan retroviral, composiciones que los contienen y ek uso de los mismos.
PL322784A1 (en) Amino acid hydroxyethylaminosulphonamides as inhibitors of retroviral protease
MX9706947A (es) Inhibidores de proteasa retroviral de sulfonilalcanoilamino-hidroxietilamino-sulfonamida y uso de los mismos.
DE69625183D1 (en) Heterocyclocarbonyl-aminosäure-hydroxyethylamino-sulfonamid inhibitoren retroviraler proteasen
MX9706912A (es) Inhibidores de protesa retroviral de sulfonamida de hidroxietilamino de amino acido y uso de los mismos.

Legal Events

Date Code Title Description
FG Grant or registration
MM Annulment or lapse due to non-payment of fees