MX2023005761A - Pirrolo [2,3-b] piridina sustituida y derivados de pirazolo [3,4-b] piridina como inhibidores de proteinas quinasas. - Google Patents
Pirrolo [2,3-b] piridina sustituida y derivados de pirazolo [3,4-b] piridina como inhibidores de proteinas quinasas.Info
- Publication number
- MX2023005761A MX2023005761A MX2023005761A MX2023005761A MX2023005761A MX 2023005761 A MX2023005761 A MX 2023005761A MX 2023005761 A MX2023005761 A MX 2023005761A MX 2023005761 A MX2023005761 A MX 2023005761A MX 2023005761 A MX2023005761 A MX 2023005761A
- Authority
- MX
- Mexico
- Prior art keywords
- pyridine
- pyrazolo
- protein kinase
- kinase inhibitors
- substituted pyrrolo
- Prior art date
Links
- MVXVYAKCVDQRLW-UHFFFAOYSA-N 1h-pyrrolo[2,3-b]pyridine Chemical class C1=CN=C2NC=CC2=C1 MVXVYAKCVDQRLW-UHFFFAOYSA-N 0.000 title 2
- 229940045988 antineoplastic drug protein kinase inhibitors Drugs 0.000 title 1
- 239000003909 protein kinase inhibitor Substances 0.000 title 1
- 150000005230 pyrazolo[3,4-b]pyridines Chemical class 0.000 title 1
- 229940124291 BTK inhibitor Drugs 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Hematology (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Se proporcionan ciertos inhibidores de BTK, sus composiciones farmacéuticas, y métodos de uso de los mismos.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US202063115027P | 2020-11-17 | 2020-11-17 | |
PCT/CN2021/130897 WO2022105746A1 (en) | 2020-11-17 | 2021-11-16 | SUBSTITUTED PYRROLO [2, 3-b] PYRIDINE AND PYRAZOLO [3, 4-b] PYRIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2023005761A true MX2023005761A (es) | 2023-05-29 |
Family
ID=81708347
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2023005761A MX2023005761A (es) | 2020-11-17 | 2021-11-16 | Pirrolo [2,3-b] piridina sustituida y derivados de pirazolo [3,4-b] piridina como inhibidores de proteinas quinasas. |
Country Status (10)
Country | Link |
---|---|
US (1) | US20230406856A1 (es) |
EP (1) | EP4247812A1 (es) |
JP (1) | JP2023549273A (es) |
KR (1) | KR20230110286A (es) |
CN (1) | CN116568686A (es) |
AU (1) | AU2021383227A1 (es) |
CA (1) | CA3198254A1 (es) |
MX (1) | MX2023005761A (es) |
TW (1) | TW202227437A (es) |
WO (1) | WO2022105746A1 (es) |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102603581B (zh) * | 2005-06-22 | 2015-06-24 | 普莱希科公司 | 作为蛋白质激酶抑制剂的吡咯并[2,3-b]吡啶衍生物 |
WO2008080001A2 (en) * | 2006-12-21 | 2008-07-03 | Plexxikon, Inc. | Compounds and methods for kinase modulation, and indications therefor |
BR112021023607A2 (pt) * | 2019-05-31 | 2022-01-04 | Fochon Pharmaceuticals Ltd | Derivados de pirrolo[2,3-b]piridina e pirazolo[3,4-b]piridina substituídos por inibidores de proteína quinase |
CN112608318B (zh) * | 2019-12-16 | 2023-09-08 | 成都海博为药业有限公司 | 一种作为蛋白质激酶抑制剂的化合物及其用途 |
CN112574200B (zh) * | 2021-02-26 | 2021-06-11 | 安润医药科技(苏州)有限公司 | Btk和/或btk的突变体c481s的小分子抑制剂 |
-
2021
- 2021-11-16 AU AU2021383227A patent/AU2021383227A1/en active Pending
- 2021-11-16 TW TW110142640A patent/TW202227437A/zh unknown
- 2021-11-16 KR KR1020237019390A patent/KR20230110286A/ko unknown
- 2021-11-16 CA CA3198254A patent/CA3198254A1/en active Pending
- 2021-11-16 MX MX2023005761A patent/MX2023005761A/es unknown
- 2021-11-16 JP JP2023529093A patent/JP2023549273A/ja active Pending
- 2021-11-16 US US18/253,252 patent/US20230406856A1/en active Pending
- 2021-11-16 CN CN202180077389.8A patent/CN116568686A/zh active Pending
- 2021-11-16 WO PCT/CN2021/130897 patent/WO2022105746A1/en active Application Filing
- 2021-11-16 EP EP21893893.4A patent/EP4247812A1/en active Pending
Also Published As
Publication number | Publication date |
---|---|
AU2021383227A1 (en) | 2023-06-22 |
CA3198254A1 (en) | 2022-05-27 |
WO2022105746A1 (en) | 2022-05-27 |
KR20230110286A (ko) | 2023-07-21 |
AU2021383227A9 (en) | 2024-05-02 |
TW202227437A (zh) | 2022-07-16 |
US20230406856A1 (en) | 2023-12-21 |
CN116568686A (zh) | 2023-08-08 |
EP4247812A1 (en) | 2023-09-27 |
JP2023549273A (ja) | 2023-11-22 |
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