MX2018006329A - Agente terapeutico para cancer de mama. - Google Patents

Agente terapeutico para cancer de mama.

Info

Publication number
MX2018006329A
MX2018006329A MX2018006329A MX2018006329A MX2018006329A MX 2018006329 A MX2018006329 A MX 2018006329A MX 2018006329 A MX2018006329 A MX 2018006329A MX 2018006329 A MX2018006329 A MX 2018006329A MX 2018006329 A MX2018006329 A MX 2018006329A
Authority
MX
Mexico
Prior art keywords
therapeutic agent
breast cancer
methoxyethoxy
benzamide
piperidin
Prior art date
Application number
MX2018006329A
Other languages
English (en)
Inventor
Yamamoto Yuji
Miyano Saori
Nakagawa Takayuki
Original Assignee
Eisai R&D Man Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eisai R&D Man Co Ltd filed Critical Eisai R&D Man Co Ltd
Publication of MX2018006329A publication Critical patent/MX2018006329A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/14Drugs for genital or sexual disorders; Contraceptives for lactation disorders, e.g. galactorrhoea
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente solicitud describe un agente terapéutico para el cáncer de mama que comprende 5-((2-(4-(1-(2-hidroxietil)piperidin- 4-il)benzamido)piridin-4-il)oxi)-6-(2-metoxietoxi)-N-metil-1H-ind ol-1-carboxamida o una sal farmacológicamente aceptable de esta.
MX2018006329A 2015-12-17 2016-12-15 Agente terapeutico para cancer de mama. MX2018006329A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2015246308 2015-12-17
PCT/JP2016/087349 WO2017104739A1 (ja) 2015-12-17 2016-12-15 乳がん治療剤

Publications (1)

Publication Number Publication Date
MX2018006329A true MX2018006329A (es) 2018-08-29

Family

ID=59056770

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2018006329A MX2018006329A (es) 2015-12-17 2016-12-15 Agente terapeutico para cancer de mama.

Country Status (13)

Country Link
US (1) US20180303817A1 (es)
EP (1) EP3391885B1 (es)
JP (1) JP6858132B2 (es)
KR (1) KR102486722B1 (es)
CN (2) CN108367000A (es)
AU (1) AU2016374441B2 (es)
CA (1) CA3001969C (es)
ES (1) ES2867804T3 (es)
IL (1) IL258671A (es)
MX (1) MX2018006329A (es)
RU (1) RU2730503C2 (es)
SG (2) SG10201913213WA (es)
WO (1) WO2017104739A1 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG11202001481PA (en) * 2017-10-12 2020-03-30 Eisai R&D Man Co Ltd Pharmaceutical composition comprising fgfr selective tyrosine kinase inhibitor
JPWO2019189241A1 (ja) 2018-03-28 2021-03-18 エーザイ・アール・アンド・ディー・マネジメント株式会社 肝細胞癌治療剤
EP4122465A4 (en) 2020-04-17 2024-03-20 Eisai R&D Man Co Ltd THERAPEUTIC AGENT AGAINST BREAST CANCER
AU2021315234A1 (en) * 2020-07-31 2023-01-19 Eisai R&D Management Co., Ltd. Therapeutic agent for breast cancer
JPWO2022092085A1 (es) 2020-10-28 2022-05-05

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7098332B2 (en) * 2002-12-20 2006-08-29 Hoffmann-La Roche Inc. 5,8-Dihydro-6H-pyrido[2,3-d]pyrimidin-7-ones
AR094812A1 (es) * 2013-02-20 2015-08-26 Eisai R&D Man Co Ltd Derivado de piridina monocíclico como inhibidor del fgfr
CA2956270C (en) * 2014-08-18 2022-08-09 Eisai R&D Management Co., Ltd. Salt of monocyclic pyridine derivative and crystal thereof

Also Published As

Publication number Publication date
RU2018119102A (ru) 2020-01-17
CN108367000A (zh) 2018-08-03
EP3391885B1 (en) 2021-03-17
CA3001969A1 (en) 2017-06-22
KR20180094862A (ko) 2018-08-24
CN115177619A (zh) 2022-10-14
AU2016374441B2 (en) 2021-10-21
SG11201803118WA (en) 2018-05-30
RU2018119102A3 (es) 2020-02-04
US20180303817A1 (en) 2018-10-25
EP3391885A4 (en) 2019-08-28
JPWO2017104739A1 (ja) 2018-10-04
EP3391885A1 (en) 2018-10-24
SG10201913213WA (en) 2020-03-30
ES2867804T3 (es) 2021-10-20
IL258671A (en) 2018-06-28
BR112018010103A2 (pt) 2018-11-21
CA3001969C (en) 2023-10-03
AU2016374441A1 (en) 2018-05-10
JP6858132B2 (ja) 2021-04-14
KR102486722B1 (ko) 2023-01-11
WO2017104739A1 (ja) 2017-06-22
RU2730503C2 (ru) 2020-08-24

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