MX2010008638A - Furo-[3,2-c]piridinas y tieno[3,2-c]piridinas. - Google Patents
Furo-[3,2-c]piridinas y tieno[3,2-c]piridinas.Info
- Publication number
- MX2010008638A MX2010008638A MX2010008638A MX2010008638A MX2010008638A MX 2010008638 A MX2010008638 A MX 2010008638A MX 2010008638 A MX2010008638 A MX 2010008638A MX 2010008638 A MX2010008638 A MX 2010008638A MX 2010008638 A MX2010008638 A MX 2010008638A
- Authority
- MX
- Mexico
- Prior art keywords
- furo
- thieno
- pyridines
- pyridine
- including conditions
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
- C07D491/044—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
- C07D491/048—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being five-membered
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
Compuestos de furo[3,2-c]piridina y tieno[3,2-c]piridina de la fórmula (I), y sales farmacéuticamente aceptables de los mismos, preparación, intermediarios, composiciones farmacéuticas y uso, tal como en tratamiento de enfermedad, incluyendo cánceres, incluyendo condiciones en las cuales EMT está implicado, incluyendo condiciones mediadas por actividad de proteína cinasa tal como RON y/o MET.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US6380008P | 2008-02-06 | 2008-02-06 | |
US11955308P | 2008-12-03 | 2008-12-03 | |
PCT/US2009/033311 WO2009100282A1 (en) | 2008-02-06 | 2009-02-06 | Furo-and thieno[3,2-c] pyridines |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2010008638A true MX2010008638A (es) | 2010-08-30 |
Family
ID=40524808
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2010008638A MX2010008638A (es) | 2008-02-06 | 2009-02-06 | Furo-[3,2-c]piridinas y tieno[3,2-c]piridinas. |
Country Status (19)
Country | Link |
---|---|
US (1) | US8022206B2 (es) |
EP (1) | EP2265616B8 (es) |
JP (1) | JP2011511094A (es) |
KR (1) | KR20110014971A (es) |
CN (1) | CN102007127A (es) |
AR (1) | AR070317A1 (es) |
AU (1) | AU2009212338A1 (es) |
BR (1) | BRPI0908050A2 (es) |
CA (1) | CA2711078A1 (es) |
CL (1) | CL2009000275A1 (es) |
EA (1) | EA201070929A1 (es) |
ES (1) | ES2451024T3 (es) |
IL (1) | IL206758A0 (es) |
MX (1) | MX2010008638A (es) |
PE (1) | PE20091414A1 (es) |
TW (1) | TW200944201A (es) |
UY (1) | UY31638A1 (es) |
WO (1) | WO2009100282A1 (es) |
ZA (1) | ZA201005554B (es) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2534156A1 (en) * | 2010-02-11 | 2012-12-19 | OSI Pharmaceuticals, LLC | 7-aminofuropyridine derivatives |
WO2011109593A1 (en) | 2010-03-03 | 2011-09-09 | OSI Pharmaceuticals, LLC | Substituted-5-aminopyrrolo/pyrazolopyridines |
US8916593B2 (en) * | 2010-05-04 | 2014-12-23 | Pfizer Inc. | Alkoxy-substituted 2-aminopyridines as ALK inhibitors |
WO2012003338A1 (en) | 2010-07-01 | 2012-01-05 | Takeda Pharmaceutical Company Limited | COMBINATION OF A cMET INHIBITOR AND AN ANTIBODY TO HGF AND/OR cMET |
TWI504350B (zh) * | 2010-09-01 | 2015-10-21 | Du Pont | 殺真菌吡唑及其混合物 |
US10614666B2 (en) | 2011-04-20 | 2020-04-07 | Video Gaming Technologies, Inc. | Gaming machines with free play bonus mode presenting only winning outcomes |
CN104136026B (zh) * | 2011-10-31 | 2018-03-02 | 卫理公会医院研究所 | 包含mao靶向/探寻器部分的人神经胶质瘤治疗用化合物 |
WO2013142253A2 (en) * | 2012-03-23 | 2013-09-26 | Memorial Sloan-Kettering Cancer Center | TREATMENT OF PANCREATIC AND RELATED CANCERS WITH 5-ACYL-6,7-DIHYDROTHIENO[3,2-c]PYRIDINES |
WO2013152252A1 (en) | 2012-04-06 | 2013-10-10 | OSI Pharmaceuticals, LLC | Combination anti-cancer therapy |
KR101582852B1 (ko) | 2012-05-24 | 2016-01-07 | 서울대학교 산학협력단 | 타우 단백질 매개 신경 퇴행성 질환 치료제 |
US9567339B2 (en) | 2013-06-26 | 2017-02-14 | Abbvie Inc. | Primary carboxamides as BTK inhibitors |
WO2015138925A1 (en) * | 2014-03-14 | 2015-09-17 | University Of Utah Research Foundation | Ron inhibitors for use in preventing and treating bone loss |
CN103923081B (zh) * | 2014-04-14 | 2017-06-27 | 武汉光谷人福生物医药有限公司 | 化合物及其制备方法和应用 |
EP3229836B1 (en) | 2014-12-09 | 2019-11-13 | Institut National de la Sante et de la Recherche Medicale (INSERM) | Human monoclonal antibodies against axl |
WO2016135041A1 (en) | 2015-02-26 | 2016-09-01 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Fusion proteins and antibodies comprising thereof for promoting apoptosis |
CN106866447A (zh) * | 2017-03-30 | 2017-06-20 | 成都绿林科技有限公司 | 一种合成对乙酰基苯甲酰胺的方法 |
US10957159B2 (en) | 2018-04-12 | 2021-03-23 | Aristocrat Technologies Australia Pty Limited | Gaming machine and method for displaying a free spin count-up |
US11427596B2 (en) * | 2019-07-19 | 2022-08-30 | Indian Institute of Technology Indore | Metal-free solvent-free synthesis of fused-pyrido heterocycles and biomedical applications |
Family Cites Families (33)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL159506A0 (en) * | 2001-06-23 | 2004-06-01 | Aventis Pharma Inc | Pyrrolopyrimidines as protein kinase inhibitors |
WO2003009852A1 (en) * | 2001-07-24 | 2003-02-06 | Merck & Co., Inc. | Tyrosine kinase inhibitors |
US20040014755A1 (en) * | 2002-01-10 | 2004-01-22 | Dhanapalan Nagarathnam | Rho-kinase inhibitors |
US7704995B2 (en) * | 2002-05-03 | 2010-04-27 | Exelixis, Inc. | Protein kinase modulators and methods of use |
US7276519B2 (en) * | 2002-11-25 | 2007-10-02 | Wyeth | Thieno[3,2-b]pyridine-6-carbonitriles and thieno[2,3-b]pyridine-5-carbonitriles as protein kinase inhibitors |
CL2003002287A1 (es) * | 2002-11-25 | 2005-01-14 | Wyeth Corp | COMPUESTOS DERIVADOS DE TIENO[3,2-b]-PIRIDINA-6-CARBONITRILOS Y TIENEO[2,3-b]-PIRIDINA-5-CARBONITRILOS, COMPOSICION FARMACEUTICA, PROCEDIMIENTO DE PREPARACION Y COMPUESTOS INTERMEDIARIOS, Y SU USO EN EL TRATAMIENTO DEL CANCER, APOPLEJIA, OSTEOPOROSIS |
EP1590339A4 (en) | 2003-01-28 | 2007-07-25 | Smithkline Beecham Corp | CHEMICAL COMPOUNDS |
ES2401330T3 (es) * | 2003-02-26 | 2013-04-18 | Sugen, Inc. | Compuesto de heteroarilamino inhibidores de proteín quinasas |
EP1620094A4 (en) * | 2003-05-06 | 2010-04-28 | Glaxosmithkline Llc | NEW CHEMICAL COMPOUNDS |
US20050026944A1 (en) * | 2003-07-24 | 2005-02-03 | Patrick Betschmann | Thienopyridine and furopyridine kinase inhibitors |
US7674907B2 (en) * | 2004-07-23 | 2010-03-09 | Amgen Inc. | Furanopyridine derivatives and methods of use |
US7361764B2 (en) * | 2004-07-27 | 2008-04-22 | Sgx Pharmaceuticals, Inc. | Pyrrolo-pyridine kinase modulators |
US7709645B2 (en) | 2004-07-27 | 2010-05-04 | Sgx Pharmaceuticals, Inc. | Pyrrolo-pyridine kinase modulators |
WO2006021886A1 (en) * | 2004-08-26 | 2006-03-02 | Pfizer Inc. | Aminoheteroaryl compounds as protein tyrosine kinase inhibitors |
BRPI0513915A (pt) * | 2004-08-26 | 2008-05-20 | Pfizer | compostos aminoeteroarila enantiomericamente puros como inibidores de proteìna quinase |
DK1784396T3 (da) | 2004-08-26 | 2011-02-14 | Pfizer | Pyrazol-substituerede aminoheteroaryl-forbindelser som proteinkinase-inhibitorer |
EP1869052A1 (en) * | 2005-04-06 | 2007-12-26 | AstraZeneca AB | Substituted heterocycles and their use as chk1, pdk1 and pak inhibitors |
KR100995790B1 (ko) * | 2005-08-16 | 2010-11-22 | 에프. 호프만-라 로슈 아게 | 신규한 4-아미노-티에노[3,2-c]피리딘-7-카르복실산아미드 |
RU2008112313A (ru) * | 2005-09-01 | 2009-10-10 | Эррэй Биофарма Инк. (Us) | Соединения ингибиторы raf и способы их применения |
EP1951728A4 (en) * | 2005-11-04 | 2011-04-20 | Glaxosmithkline Llc | THIENOPYRIDINES AS INHIBITORS OF B-RAF KINASE |
RU2387650C2 (ru) * | 2005-12-05 | 2010-04-27 | Пфайзер Продактс Инк. | Полиморфы с-met/hgfr ингибитора |
US7989461B2 (en) * | 2005-12-23 | 2011-08-02 | Amgen Inc. | Substituted quinazolinamine compounds for the treatment of cancer |
ATE453635T1 (de) | 2006-03-22 | 2010-01-15 | Vertex Pharma | C-met-proteinkinasehemmer zur behandlung proliferativer erkrankungen |
US7745449B2 (en) * | 2006-04-21 | 2010-06-29 | Amgen Inc. | Thieno-[2,3-d]pyrimidine and thieno-pyridazine compounds and methods of use |
US7601716B2 (en) * | 2006-05-01 | 2009-10-13 | Cephalon, Inc. | Pyridopyrazines and derivatives thereof as ALK and c-Met inhibitors |
PE20121126A1 (es) * | 2006-12-21 | 2012-08-24 | Plexxikon Inc | Compuestos pirrolo [2,3-b] piridinas como moduladores de quinasa |
RU2009122670A (ru) * | 2006-12-21 | 2011-01-27 | Плекссикон, Инк. (Us) | Соединения и способы для модуляции киназ и показания к их применению |
GB0625659D0 (en) | 2006-12-21 | 2007-01-31 | Cancer Rec Tech Ltd | Therapeutic compounds and their use |
CL2008001540A1 (es) * | 2007-05-29 | 2009-05-22 | Sgx Pharmaceuticals Inc | Compuestos derivados de pirrolopiridinas y pirazolopiridinas; composicion farmaceutica; y uso en el tratamiento del cancer. |
AU2008315746A1 (en) * | 2007-10-25 | 2009-04-30 | Astrazeneca Ab | Pyridine and pyrazine derivatives useful in the treatment of cell proliferative disorders |
UY31478A1 (es) | 2007-11-21 | 2009-07-17 | Inhibicion del receptor para la proteina estimulante del macrofago (ron) y métodos para el tratamiento de lo mismo | |
KR101034351B1 (ko) | 2008-05-14 | 2011-05-16 | 한국화학연구원 | 신규 벤즈옥사졸로 치환된 피리딘 유도체 또는 이의약학적으로 허용가능한 염, 이의 제조방법 및 이를유효성분으로 함유하는 이상세포 성장 질환의 예방 및치료용 약학적 조성물 |
WO2009140549A1 (en) | 2008-05-14 | 2009-11-19 | Amgen Inc. | Combinations vegf(r) inhibitors and hepatocyte growth factor (c-met) inhibitors for the treatment of cancer |
-
2009
- 2009-01-29 AR ARP090100283A patent/AR070317A1/es unknown
- 2009-02-04 TW TW098103558A patent/TW200944201A/zh unknown
- 2009-02-05 UY UY031638A patent/UY31638A1/es not_active Application Discontinuation
- 2009-02-05 PE PE2009000178A patent/PE20091414A1/es not_active Application Discontinuation
- 2009-02-06 ES ES09709265.4T patent/ES2451024T3/es active Active
- 2009-02-06 CL CL2009000275A patent/CL2009000275A1/es unknown
- 2009-02-06 BR BRPI0908050-3A patent/BRPI0908050A2/pt not_active IP Right Cessation
- 2009-02-06 KR KR1020107019308A patent/KR20110014971A/ko not_active Application Discontinuation
- 2009-02-06 JP JP2010546027A patent/JP2011511094A/ja not_active Ceased
- 2009-02-06 CA CA2711078A patent/CA2711078A1/en not_active Abandoned
- 2009-02-06 US US12/366,743 patent/US8022206B2/en not_active Expired - Fee Related
- 2009-02-06 WO PCT/US2009/033311 patent/WO2009100282A1/en active Application Filing
- 2009-02-06 CN CN2009801092027A patent/CN102007127A/zh active Pending
- 2009-02-06 EA EA201070929A patent/EA201070929A1/ru unknown
- 2009-02-06 MX MX2010008638A patent/MX2010008638A/es active IP Right Grant
- 2009-02-06 EP EP09709265.4A patent/EP2265616B8/en active Active
- 2009-02-06 AU AU2009212338A patent/AU2009212338A1/en not_active Abandoned
-
2010
- 2010-07-01 IL IL206758A patent/IL206758A0/en unknown
- 2010-08-04 ZA ZA2010/05554A patent/ZA201005554B/en unknown
Also Published As
Publication number | Publication date |
---|---|
KR20110014971A (ko) | 2011-02-14 |
UY31638A1 (es) | 2009-09-30 |
WO2009100282A1 (en) | 2009-08-13 |
EP2265616B1 (en) | 2013-11-20 |
ZA201005554B (en) | 2011-04-28 |
US8022206B2 (en) | 2011-09-20 |
CA2711078A1 (en) | 2009-08-13 |
JP2011511094A (ja) | 2011-04-07 |
ES2451024T3 (es) | 2014-03-26 |
PE20091414A1 (es) | 2009-09-23 |
AU2009212338A1 (en) | 2009-08-13 |
EA201070929A1 (ru) | 2011-04-29 |
US20090197864A1 (en) | 2009-08-06 |
TW200944201A (en) | 2009-11-01 |
CL2009000275A1 (es) | 2009-06-12 |
IL206758A0 (en) | 2010-12-30 |
BRPI0908050A2 (pt) | 2015-08-11 |
AR070317A1 (es) | 2010-03-31 |
EP2265616A1 (en) | 2010-12-29 |
EP2265616B8 (en) | 2014-01-08 |
CN102007127A (zh) | 2011-04-06 |
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