MX2009004385A - Derivados de 2-[1-fenil-5-hidroxi-4alfa-metil-hexahidrociclopenta [f]indazol-5-il]etil fenilo como ligandos del receptor glucocorticoide. - Google Patents

Derivados de 2-[1-fenil-5-hidroxi-4alfa-metil-hexahidrociclopenta [f]indazol-5-il]etil fenilo como ligandos del receptor glucocorticoide.

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Publication number
MX2009004385A
MX2009004385A MX2009004385A MX2009004385A MX2009004385A MX 2009004385 A MX2009004385 A MX 2009004385A MX 2009004385 A MX2009004385 A MX 2009004385A MX 2009004385 A MX2009004385 A MX 2009004385A MX 2009004385 A MX2009004385 A MX 2009004385A
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MX
Mexico
Prior art keywords
phenyl
4alpha
indazol
hydroxy
methyl
Prior art date
Application number
MX2009004385A
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English (en)
Inventor
James J Perkins
Christopher J Bungard
Jesse J Manikowski
Robert Meissner
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Merck & Co Inc
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Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of MX2009004385A publication Critical patent/MX2009004385A/es

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    • A61K31/415—1,2-Diazoles
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Abstract

La presente invención se refiere a derivados de 2-[1-fenil-5-hidroxi-4alfa-metil-hexahidrociclopenta[f]indazol-5- il]etil fenilo como ligandos del receptor glucocorticoide útiles para el tratamiento de una variedad de enfermedades o afecciones autoinmunes e inflamatorias; también se incluyen composiciones farmacéuticas y procedimientos de uso.
MX2009004385A 2006-10-23 2007-10-23 Derivados de 2-[1-fenil-5-hidroxi-4alfa-metil-hexahidrociclopenta [f]indazol-5-il]etil fenilo como ligandos del receptor glucocorticoide. MX2009004385A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US85365506P 2006-10-23 2006-10-23
US92333707P 2007-04-13 2007-04-13
PCT/US2007/022449 WO2008060391A2 (en) 2006-10-23 2007-10-23 2- [l-phenyl-5-hydr0xy-4alpha-methyl-hexahydr0cycl0penta[f] indaz0l-5-yl] ethyl phenyl derivatives as glucocorticoid receptor ligands

Publications (1)

Publication Number Publication Date
MX2009004385A true MX2009004385A (es) 2009-05-22

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Family Applications (1)

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MX2009004385A MX2009004385A (es) 2006-10-23 2007-10-23 Derivados de 2-[1-fenil-5-hidroxi-4alfa-metil-hexahidrociclopenta [f]indazol-5-il]etil fenilo como ligandos del receptor glucocorticoide.

Country Status (19)

Country Link
US (1) US8119681B2 (es)
EP (2) EP2097385B1 (es)
JP (1) JP5271911B2 (es)
KR (1) KR20090068345A (es)
CN (1) CN101528707B (es)
AT (1) ATE538099T1 (es)
AU (1) AU2007309507A1 (es)
BR (1) BRPI0718505A2 (es)
CA (1) CA2667007A1 (es)
CO (1) CO6190517A2 (es)
CR (1) CR10771A (es)
EA (1) EA200970401A1 (es)
IL (1) IL198226A0 (es)
MA (1) MA30870B1 (es)
MX (1) MX2009004385A (es)
NO (1) NO20092004L (es)
SV (1) SV2009003233A (es)
TN (1) TN2009000149A1 (es)
WO (2) WO2008051532A1 (es)

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